Vincent P. Santarelli, PhD - Publications

Affiliations: 
Physiology  Thomas Jefferson University, Philadelphia, PA, United States 
Area:
Ion channels, sodium channels, potassium channels

11 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Chen YT, Hong MR, Zhang XJ, Kostas J, Li Y, Kraus RL, Santarelli VP, Wang D, Gomez-Llorente Y, Brooun A, Strickland C, Soisson SM, Klein DJ, Ginnetti AT, Marino MJ, et al. Identification, structural, and biophysical characterization of a positive modulator of human Kv3.1 channels. Proceedings of the National Academy of Sciences of the United States of America. 120: e2220029120. PMID 37812700 DOI: 10.1073/pnas.2220029120  0.42
2017 Yao J, McHedlishvili D, McIntire WE, Guagliardo NA, Erisir A, Coburn CA, Santarelli VP, Bayliss DA, Barrett PQ. Functional TASK-3-Like Channels in Mitochondria of Aldosterone-Producing Zona Glomerulosa Cells. Hypertension (Dallas, Tex. : 1979). PMID 28630209 DOI: 10.1161/Hypertensionaha.116.08871  0.384
2017 Roecker AJ, Egbertson M, Jones KL, Gomez R, Kraus RL, Li Y, Koser AJ, Urban MO, Klein R, Clements M, Panigel J, Daley C, Wang J, Finger EN, Majercak J, ... Santarelli V, et al. Discovery of selective, orally bioavailable, N-linked arylsulfonamide Nav1.7 inhibitors with pain efficacy in mice. Bioorganic & Medicinal Chemistry Letters. PMID 28389149 DOI: 10.1016/J.Bmcl.2017.03.085  0.303
2012 Coburn CA, Luo Y, Cui M, Wang J, Soll R, Dong J, Hu B, Lyon MA, Santarelli VP, Kraus RL, Gregan Y, Wang Y, Fox SV, Binns J, Doran SM, et al. Discovery of a pharmacologically active antagonist of the two-pore-domain potassium channel K2P9.1 (TASK-3). Chemmedchem. 7: 123-33. PMID 21916012 DOI: 10.1002/Cmdc.201100351  0.447
2009 Uebele VN, Nuss CE, Fox SV, Garson SL, Cristescu R, Doran SM, Kraus RL, Santarelli VP, Li Y, Barrow JC, Yang ZQ, Schlegel KA, Rittle KE, Reger TS, Bednar RA, et al. Positive allosteric interaction of structurally diverse T-type calcium channel antagonists. Cell Biochemistry and Biophysics. 55: 81-93. PMID 19582593 DOI: 10.1007/S12013-009-9057-4  0.47
2009 Uebele VN, Nuss CE, Santarelli VP, Garson SL, Kraus RL, Barrow JC, Stauffer SR, Koblan KS, Renger JJ, Aton S, Seibt J, Dumoulin M, Jha SK, Coleman T, Frank MG. T-type calcium channels regulate cortical plasticity in-vivo. [corrected]. Neuroreport. 20: 257-62. PMID 19212242 DOI: 10.1097/Wnr.0B013E3283200111  0.469
2007 Santarelli VP, Eastwood AL, Dougherty DA, Ahern CA, Horn R. Calcium block of single sodium channels: role of a pore-lining aromatic residue. Biophysical Journal. 93: 2341-9. PMID 17545248 DOI: 10.1529/Biophysj.107.106856  0.399
2007 Santarelli VP, Eastwood AL, Dougherty DA, Horn R, Ahern CA. A cation-pi interaction discriminates among sodium channels that are either sensitive or resistant to tetrodotoxin block. The Journal of Biological Chemistry. 282: 8044-51. PMID 17237232 DOI: 10.1074/Jbc.M611334200  0.425
2003 Xia M, Imredy JP, Santarelli VP, Liang HA, Condra CL, Bennett P, Koblan KS, Connolly TM. Generation and characterization of a cell line with inducible expression of Ca(v)3.2 (T-type) channels. Assay and Drug Development Technologies. 1: 637-45. PMID 15090236 DOI: 10.1089/154065803770380995  0.409
1997 Sheng Z, Skach W, Santarelli V, Deutsch C. Evidence for interaction between transmembrane segments in assembly of Kv1.3. Biochemistry. 36: 15501-13. PMID 9398279 DOI: 10.1021/Bi971490J  0.391
1996 Tu L, Santarelli V, Sheng Z, Skach W, Pain D, Deutsch C. Voltage-gated K+ channels contain multiple intersubunit association sites. The Journal of Biological Chemistry. 271: 18904-11. PMID 8702552 DOI: 10.1074/Jbc.271.31.18904  0.369
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