Jeffrey L. Gustafson - Publications

Affiliations: 
2011 Yale University, New Haven, CT 

33 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Basilaia M, Chen MH, Secka J, Gustafson JL. Atropisomerism in the Pharmaceutically Relevant Realm. Accounts of Chemical Research. PMID 36153960 DOI: 10.1021/acs.accounts.2c00500  0.342
2021 Cardenas MM, Saputra MA, Gordon DA, Sanchez AN, Yamamoto N, Gustafson JL. Catalytic atroposelective dynamic kinetic resolutions and kinetic resolutions towards 3-arylquinolines SAr. Chemical Communications (Cambridge, England). PMID 34515276 DOI: 10.1039/d1cc04335h  0.318
2020 Dinh AN, Maddox SM, Vaidya SD, Saputra MA, Nalbandian CJ, Gustafson JL. Catalyst-Controlled Regioselective Chlorination of Phenols and Anilines through a Lewis Basic Selenoether Catalyst. The Journal of Organic Chemistry. PMID 33044067 DOI: 10.1021/acs.joc.0c01917  0.323
2020 Ortiz MA, Michaels H, Molina B, Toenjes S, Davis J, Diletta Marconi G, Hecht D, Gustafson JL, Javier Piedrafita F, Nefzi A. Discovery of cyclic guanidine-linked sulfonamides as inhibitors of LMTK3 kinase. Bioorganic & Medicinal Chemistry Letters. 127108. PMID 32192797 DOI: 10.1016/J.Bmcl.2020.127108  0.326
2020 Vaidya SD, Toenjes ST, Yamamoto N, Maddox SM, Gustafson JL. Catalytic Atroposelective Synthesis of N-Aryl Quinoid Compounds. Journal of the American Chemical Society. PMID 31944689 DOI: 10.1021/Jacs.9B12994  0.448
2020 Dinh A, Gustafson JL. A Catalytic Cycle of Discovery: Asymmetric Catalysis Gives Rise to New Chiral Catalyst Scaffolds Chem. 6: 810-812. DOI: 10.1016/J.Chempr.2020.03.020  0.439
2019 Toenjes ST, Garcia V, Maddox SM, Dawson GA, Ortiz MA, Piedrafita FJ, Gustafson JL. Leveraging atropisomerism to obtain a selective inhibitor of RET kinase with secondary activities towards EGFR mutants. Acs Chemical Biology. PMID 31424197 DOI: 10.1021/Acschembio.9B00407  0.408
2019 Dinh AN, Nguyen AD, Aceves EM, Albright ST, Cedano MR, Smith DK, Gustafson JL. Photocatalytic Oxidative C–H Thiolation: Synthesis of Benzothiazoles and Sulfenylated Indoles Synlett. 30: 1648-1655. DOI: 10.1055/S-0039-1690107  0.309
2018 Dinh AN, Noorbehesht RR, Toenjes ST, Jackson AC, Saputra MA, Maddox SM, Gustafson JL. Towards a Catalytic Atroposelective Synthesis of Diaryl Ethers via C()-H Alkylation Using Nitroalkanes. Synlett : Accounts and Rapid Communications in Synthetic Organic Chemistry. 29: 2155-2160. PMID 31178629 DOI: 10.1055/S-0037-1609581  0.363
2018 Maddox SM, Dawson GA, Rochester NC, Ayonon AB, Moore CE, Rheingold AL, Gustafson JL. Enantioselective Synthesis of Biaryl Atropisomers via the Addition of Thiophenols into Aryl-Naphthoquinones. Acs Catalysis. 8: 5443-5447. PMID 30455999 DOI: 10.1021/Acscatal.8B00906  0.411
2018 Nalbandian CJ, Brown ZE, Alvarez E, Gustafson JL. Lewis Base/Bronsted Acid Dual-Catalytic C-H Sulfenylation of Aromatics. Organic Letters. PMID 29762039 DOI: 10.1021/Acs.Orglett.8B01066  0.359
2018 Cardenas MM, Toenjes ST, Nalbandian CJ, Gustafson JL. Enantioselective Synthesis of Pyrrolopyrimidine Scaffolds through Cation-Directed Nucleophilic Aromatic Substitution. Organic Letters. PMID 29561161 DOI: 10.1021/Acs.Orglett.8B00579  0.465
2018 Toenjes ST, Gustafson JL. Atropisomerism in medicinal chemistry: challenges and opportunities. Future Medicinal Chemistry. PMID 29380622 DOI: 10.4155/Fmc-2017-0152  0.416
2017 Ottis P, Toure M, Cromm PM, Ko E, Gustafson JL, Crews CM. Assessing Different E3 Ligases for Small Molecule-induced Protein Ubiquitination and Degradation. Acs Chemical Biology. PMID 28767222 DOI: 10.1021/Acschembio.7B00485  0.357
2017 Nalbandian CJ, Miller EM, Toenjes ST, Gustafson JL. A conjugate Lewis base-Brønsted acid catalyst for the sulfenylation of nitrogen containing heterocycles under mild conditions. Chemical Communications (Cambridge, England). PMID 28084476 DOI: 10.1039/C6Cc09998J  0.375
2017 Ayonon A, Nalbandian C, Guillemard L, Gustafson J. Benzylic bromination catalyzed by triphenylphosphine selenide via Lewis basic activation Tetrahedron Letters. 58: 2940-2943. DOI: 10.1016/J.Tetlet.2017.06.042  0.436
2016 Maddox SM, Dinh AN, Armenta F, Um J, Gustafson JL. The Catalyst-Controlled Regiodivergent Chlorination of Phenols. Organic Letters. PMID 27754679 DOI: 10.1021/Acs.Orglett.6B02650  0.415
2016 Maddox S, Hecht D, Gustafson JL. Enhancing the selectivity of kinase inhibitors in oncology: a chemical biology perspective. Future Medicinal Chemistry. PMID 26898835 DOI: 10.4155/Fmc.15.193  0.324
2016 Maligal-Ganesh RV, Xiao C, Goh TW, Wang LL, Gustafson J, Pei Y, Qi Z, Johnson DD, Zhang S, Tao F, Huang W. A Ship-in-a-Bottle Strategy to Synthesize Encapsulated Intermetallic Nanoparticle Catalysts: Exemplified for Furfural Hydrogenation Acs Catalysis. 6: 1754-1763. DOI: 10.1021/Acscatal.5B02281  0.338
2016 Kelly MJB, Fallot LB, Gustafson JL, Bergdahl BM. Water Mediated Wittig Reactions of Aldehydes in the Teaching Laboratory: Using Sodium Bicarbonate for the in Situ Formation of Stabilized Ylides Journal of Chemical Education. 93: 1631-1636. DOI: 10.1021/Acs.Jchemed.6B00206  0.321
2015 Smith DE, Marquez I, Lokensgard ME, Rheingold AL, Hecht DA, Gustafson JL. Exploiting Atropisomerism to Increase the Target Selectivity of Kinase Inhibitors. Angewandte Chemie (International Ed. in English). PMID 26276764 DOI: 10.1002/Anie.201506085  0.397
2015 Bondeson DP, Mares A, Smith IE, Ko E, Campos S, Miah AH, Mulholland KE, Routly N, Buckley DL, Gustafson JL, Zinn N, Grandi P, Shimamura S, Bergamini G, Faelth-Savitski M, et al. Catalytic in vivo protein knockdown by small-molecule PROTACs. Nature Chemical Biology. 11: 611-7. PMID 26075522 DOI: 10.1038/Nchembio.1858  0.4
2015 Buckley DL, Raina K, Darricarrere N, Hines J, Gustafson JL, Smith IE, Miah AH, Harling JD, Crews CM. HaloPROTACS: Use of Small Molecule PROTACs to Induce Degradation of HaloTag Fusion Proteins. Acs Chemical Biology. PMID 26070106 DOI: 10.1021/Acschembio.5B00442  0.398
2015 Maddox SM, Nalbandian CJ, Smith DE, Gustafson JL. A practical Lewis base catalyzed electrophilic chlorination of arenes and heterocycles. Organic Letters. 17: 1042-5. PMID 25671756 DOI: 10.1021/Acs.Orglett.5B00186  0.4
2015 Nalbandian CJ, Hecht DE, Gustafson JL. The Preorganization of Atropisomers to Increase Target Selectivity Synlett. DOI: 10.1055/S-0035-1561314  0.433
2015 Luca OR, Gustafson JL, Maddox SM, Fenwick AQ, Smith DC. Catalysis by electrons and holes: Formal potential scales and preparative organic electrochemistry Organic Chemistry Frontiers. 2: 823-848. DOI: 10.1039/C5Qo00075K  0.318
2012 Buckley DL, Gustafson JL, Van Molle I, Roth AG, Tae HS, Gareiss PC, Jorgensen WL, Ciulli A, Crews CM. Small-molecule inhibitors of the interaction between the E3 ligase VHL and HIF1α. Angewandte Chemie (International Ed. in English). 51: 11463-7. PMID 23065727 DOI: 10.1002/Anie.201206231  0.373
2012 Tae HS, Sundberg TB, Neklesa TK, Noblin DJ, Gustafson JL, Roth AG, Raina K, Crews CM. Identification of hydrophobic tags for the degradation of stabilized proteins. Chembiochem : a European Journal of Chemical Biology. 13: 538-41. PMID 22271667 DOI: 10.1002/Cbic.201100793  0.323
2011 Gustafson JL, Lim D, Barrett KT, Miller SJ. Synthesis of atropisomerically defined, highly substituted biaryl scaffolds through catalytic enantioselective bromination and regioselective cross-coupling. Angewandte Chemie (International Ed. in English). 50: 5125-9. PMID 21520374 DOI: 10.1002/Anie.201101147  0.634
2010 Gustafson JL, Lim D, Miller SJ. Dynamic kinetic resolution of biaryl atropisomers via peptide-catalyzed asymmetric bromination. Science (New York, N.Y.). 328: 1251-5. PMID 20522769 DOI: 10.1126/Science.1188403  0.641
2010 Gustafson JL, Sigman MS, Miller SJ. Linear free-energy relationship analysis of a catalytic desymmetrization reaction of a diarylmethane-bis(phenol). Organic Letters. 12: 2794-7. PMID 20486656 DOI: 10.1021/Ol100927M  0.463
2008 Lewis CA, Gustafson JL, Chiu A, Balsells J, Pollard D, Murry J, Reamer RA, Hansen KB, Miller SJ. A case of remote asymmetric induction in the peptide-catalyzed desymmetrization of a bis(phenol). Journal of the American Chemical Society. 130: 16358-65. PMID 19006301 DOI: 10.1021/Ja807120Z  0.631
2007 Grotjahn DB, Larsen CR, Gustafson JL, Nair R, Sharma A. Extensive isomerization of alkenes using a bifunctional catalyst: an alkene zipper. Journal of the American Chemical Society. 129: 9592-3. PMID 17636924 DOI: 10.1021/Ja073457I  0.398
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