| Year |
Citation |
Score |
| 2020 |
Jaime-Figueroa S, Buhimschi AD, Toure M, Hines J, Crews CM. Design, synthesis and biological evaluation of Proteolysis Targeting Chimeras (PROTACs) as a BTK degraders with improved pharmacokinetic properties. Bioorganic & Medicinal Chemistry Letters. 30: 126877. PMID 31879210 DOI: 10.1016/J.Bmcl.2019.126877 |
0.643 |
|
| 2018 |
Burslem GM, Ottis P, Jaime-Figueroa S, Morgan A, Cromm P, Toure M, Crews C. Efficient Synthesis of Immunomodulatory Drug Analogues Enables Exploration of Structure Degradation Relationships. Chemmedchem. PMID 29870139 DOI: 10.1002/Cmdc.201800271 |
0.705 |
|
| 2018 |
Serebrenik YV, Hellerschmied D, Toure M, López-Giráldez F, Brookner D, Crews CM. Targeted protein unfolding uncovers a Golgi-specific transcriptional stress response. Molecular Biology of the Cell. 29: 1284-1298. PMID 29851555 DOI: 10.1091/Mbc.E17-11-0693 |
0.676 |
|
| 2018 |
Buhimschi AD, Armstrong HA, Toure M, Jaime-Figueroa S, Chen TL, Lehman AM, Woyach JA, Johnson AJ, Byrd JC, Crews CM. Targeting the C481S Ibrutinib-Resistance Mutation in Bruton's Tyrosine Kinase using PROTAC-mediated Degradation. Biochemistry. PMID 29851337 DOI: 10.1021/Acs.Biochem.8B00391 |
0.57 |
|
| 2017 |
Burslem GM, Smith BE, Lai AC, Jaime-Figueroa S, McQuaid DC, Bondeson DP, Toure M, Dong H, Qian Y, Wang J, Crew AP, Hines J, Crews CM. The Advantages of Targeted Protein Degradation Over Inhibition: An RTK Case Study. Cell Chemical Biology. PMID 29129716 DOI: 10.1016/J.Chembiol.2017.09.009 |
0.669 |
|
| 2017 |
Ottis P, Toure M, Cromm PM, Ko E, Gustafson JL, Crews CM. Assessing Different E3 Ligases for Small Molecule-induced Protein Ubiquitination and Degradation. Acs Chemical Biology. PMID 28767222 DOI: 10.1021/Acschembio.7B00485 |
0.716 |
|
| 2016 |
Toure M, Jaime-Figueroa S, Burslem GM, Crews CM. Expeditious Synthesis of Isoquinolones and Isocoumarins with a Vinyl Borane as an Acetylene Equivalent. European Journal of Organic Chemistry. 2016: 4171-4175. PMID 28781577 DOI: 10.1002/Ejoc.201600575 |
0.53 |
|
| 2016 |
Toure M, Crews CM. Small-Molecule PROTACS: New Approaches to Protein Degradation. Angewandte Chemie (International Ed. in English). PMID 26756721 DOI: 10.1002/Anie.201507978 |
0.678 |
|
| 2016 |
Toure M, Crews CM. Niedermolekulare PROTACs: neue Wege zum Abbau von Proteinen Angewandte Chemie. 128: 2002-2010. DOI: 10.1002/Ange.201507978 |
0.59 |
|
| 2015 |
Lai AC, Toure M, Hellerschmied D, Salami J, Jaime-Figueroa S, Ko E, Hines J, Crews CM. Modular PROTAC Design for the Degradation of Oncogenic BCR-ABL. Angewandte Chemie (International Ed. in English). PMID 26593377 DOI: 10.1002/Anie.201507634 |
0.716 |
|
| 2015 |
Lai AC, Toure M, Hellerschmied D, Salami J, Jaime-Figueroa S, Ko E, Hines J, Crews CM. Modulares PROTAC-Design zum Abbau von onkogenem BCR-ABL Angewandte Chemie. 128: 818-821. DOI: 10.1002/Ange.201507634 |
0.555 |
|
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