☰

Kevin George Pinney - Publications

Affiliations: 
1993- Chemistry Baylor University, Waco, TX 
Area:
total synthesis of natural products
Website:
https://www.baylor.edu/chemistry/index.php?id=950871
Tree Info Similar researchers PubMed Report error

70 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Ren W, Deng Y, Ward JD, Vairin R, Bai R, Wanniarachchi HI, Hamal KB, Tankoano PE, Tamminga CS, Bueno LMA, Hamel E, Mason RP, Trawick ML, Pinney KG. Synthesis and biological evaluation of structurally diverse 6-aryl-3-aroyl-indole analogues as inhibitors of tubulin polymerization. European Journal of Medicinal Chemistry. 263: 115794. PMID 37984295 DOI: 10.1016/j.ejmech.2023.115794  0.471
2023 Ren W, Vairin R, Ward JD, Francis R, VanNatta J, Bai R, Tankoano PE, Deng Y, Hamel E, Trawick ML, Pinney KG. Structure Guided Design, Synthesis, and Biological Evaluation of Oxetane-Containing Indole Analogues. Bioorganic & Medicinal Chemistry. 92: 117400. PMID 37556912 DOI: 10.1016/j.bmc.2023.117400  0.454
2022 Liu L, Schuetze R, Gerberich JL, Lopez R, Odutola SO, Tanpure RP, Charlton-Sevcik AK, Tidmore JK, Taylor EA, Kapur P, Hammers H, Trawick ML, Pinney KG, Mason RP. Demonstrating Tumor Vascular Disrupting Activity of the Small-Molecule Dihydronaphthalene Tubulin-Binding Agent OXi6196 as a Potential Therapeutic for Cancer Treatment. Cancers. 14. PMID 36077745 DOI: 10.3390/cancers14174208  0.792
2021 Guo Y, Wang H, Gerberich JL, Odutola SO, Charlton-Sevcik AK, Li M, Tanpure RP, Tidmore JK, Trawick ML, Pinney KG, Mason RP, Liu L. Imaging-Guided Evaluation of the Novel Small-Molecule Benzosuberene Tubulin-Binding Agent KGP265 as a Potential Therapeutic Agent for Cancer Treatment. Cancers. 13. PMID 34638255 DOI: 10.3390/cancers13194769  0.787
2020 Winn BA, Devkota L, Kuch B, MacDonough MT, Strecker TE, Wang Y, Shi Z, Gerberich JL, Mondal D, Ramirez AJ, Hamel E, Chaplin DJ, Davis P, Mason RP, Trawick ML, ... Pinney KG, et al. Bioreductively Activatable Prodrug Conjugates of Combretastatin A-1 and Combretastatin A-4 as Anticancer Agents Targeted toward Tumor-Associated Hypoxia. Journal of Natural Products. PMID 32196334 DOI: 10.1021/Acs.Jnatprod.9B00773  0.472
2019 Maguire CJ, Carlson GJ, Ford JW, Strecker TE, Hamel E, Trawick ML, Pinney KG. Synthesis and biological evaluation of structurally diverse α-conformationally restricted chalcones and related analogues. Medchemcomm. 10: 1445-1456. PMID 31534659 DOI: 10.1039/C9Md00127A  0.528
2019 Mondal D, Niu H, Pinney KG. Efficient Synthetic Methodology for the Construction of Dihydronaphthalene and Benzosuberene Molecular Frameworks. Tetrahedron Letters. 60: 397-401. PMID 31061544 DOI: 10.1016/J.Tetlet.2018.12.033  0.562
2019 Niu H, Strecker TE, Gerberich JL, Campbell J, Saha D, Mondal D, Hamel E, Chaplin DJ, Mason RP, Trawick ML, Pinney KG. Structure Guided Design, Synthesis, and Biological Evaluation of Novel Benzosuberene Analogues as Inhibitors of Tubulin Polymerization. Journal of Medicinal Chemistry. PMID 31059248 DOI: 10.1021/Acs.Jmedchem.9B00551  0.545
2018 Mondal D, Ford J, Pinney KG. Improved Methodology for the Synthesis of a Cathepsin B Cleavable Dipeptide Linker, Widely Used in Antibody-Drug Conjugate Research. Tetrahedron Letters. 59: 3594-3599. PMID 31156276 DOI: 10.1016/J.Tetlet.2018.08.021  0.415
2018 Maguire CJ, Chen Z, Mocharla VP, Sriram M, Strecker TE, Hamel E, Zhou H, Lopez R, Wang Y, Mason RP, Chaplin DJ, Trawick ML, Pinney KG. Synthesis of dihydronaphthalene analogues inspired by combretastatin A-4 and their biological evaluation as anticancer agents. Medchemcomm. 9: 1649-1662. PMID 30429970 DOI: 10.1039/C8Md00322J  0.839
2017 Pinney KG, Trawick ML, Mason RP, Liu L, Chaplin DJ, Winn BA, Devkota L, Strecker TE, Gerberich J, Winters A, Wang Y, MacDonough MT. Abstract 3203: Targeting tumor hypoxia with prodrug conjugates of potent small-molecule inhibitors of tubulin polymerization Cancer Research. 77: 3203-3203. DOI: 10.1158/1538-7445.Am2017-3203  0.386
2016 Herdman CA, Strecker TE, Tanpure RP, Chen Z, Winters A, Gerberich J, Liu L, Hamel E, Mason RP, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and Biological Evaluation of Benzocyclooctene-based and Indene-based Anticancer Agents that Function as Inhibitors of Tubulin Polymerization. Medchemcomm. 7: 2418-2427. PMID 28217276 DOI: 10.1039/C6Md00459H  0.853
2016 Parker EN, Odutola SO, Wang Y, Strecker TE, Mukherjee R, Shi Z, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and biological evaluation of a water-soluble phosphate prodrug salt and structural analogues of KGP94, a lead inhibitor of cathepsin L. Bioorganic & Medicinal Chemistry Letters. PMID 28117205 DOI: 10.1016/J.Bmcl.2016.12.039  0.479
2016 Winn BA, Shi Z, Carlson GJ, Wang Y, Nguyen BL, Kelly EM, Ross RD, Hamel E, Chaplin DJ, Trawick ML, Pinney KG. Bioreductively activatable prodrug conjugates of phenstatin designed to target tumor hypoxia. Bioorganic & Medicinal Chemistry Letters. PMID 28007448 DOI: 10.1016/J.Bmcl.2016.11.093  0.738
2016 Devkota L, Lin CM, Strecker TE, Wang Y, Tidmore JK, Chen Z, Guddneppanavar R, Jelinek CJ, Lopez R, Liu L, Hamel E, Mason RP, Chaplin DJ, Trawick ML, Pinney KG. Design, synthesis, and biological evaluation of water-soluble amino acid prodrug conjugates derived from combretastatin, dihydronaphthalene, and benzosuberene-based parent vascular disrupting agents. Bioorganic & Medicinal Chemistry. PMID 26852340 DOI: 10.1016/J.Bmc.2016.01.007  0.531
2016 Liu L, Trawick ML, Pinney K, Mason RP. Abstract 4194: Assessment of novel benzosuberene-based vascular disrupting agents (VDA) on diverse tumor lines Cancer Research. 76: 4194-4194. DOI: 10.1158/1538-7445.Am2016-4194  0.357
2015 MacDonough MT, Shi Z, Pinney KG. Mechanistic Considerations in the Synthesis of 2-Aryl-Indole Analogues under Bischler-Mohlau Conditions. Tetrahedron Letters. 56: 3624-3629. PMID 26973358 DOI: 10.1016/J.Tetlet.2015.01.129  0.383
2015 Herdman CA, Devkota L, Lin CM, Niu H, Strecker TE, Lopez R, Liu L, George CS, Tanpure RP, Hamel E, Chaplin DJ, Mason RP, Trawick ML, Pinney KG. Structural interrogation of benzosuberene-based inhibitors of tubulin polymerization. Bioorganic & Medicinal Chemistry. PMID 26775540 DOI: 10.1016/J.Bmc.2015.10.012  0.844
2015 Parker EN, Song J, Kishore Kumar GD, Odutola SO, Chavarria GE, Charlton-Sevcik AK, Strecker TE, Barnes AL, Sudhan DR, Wittenborn TR, Siemann DW, Horsman MR, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L. Bioorganic & Medicinal Chemistry. PMID 26462052 DOI: 10.1016/J.Bmc.2015.09.036  0.828
2015 Strecker TE, Odutola SO, Lopez R, Cooper MS, Tidmore JK, Charlton-Sevcik AK, Li L, MacDonough MT, Hadimani MB, Ghatak A, Liu L, Chaplin DJ, Mason RP, Pinney KG, Trawick ML. The vascular disrupting activity of OXi8006 in endothelial cells and its phosphate prodrug OXi8007 in breast tumor xenografts. Cancer Letters. 369: 229-41. PMID 26325604 DOI: 10.1016/J.Canlet.2015.08.021  0.788
2014 Wittenborn TR, Stratford M, Trawick ML, Pinney KG, Chaplin DJ, Siemann DW, Horsman MR. Abstract 1816: Assessment of anti-tumor activity of the cathepsin L inhibitor, KGP94 Cancer Research. 74: 1816-1816. DOI: 10.1158/1538-7445.Am2014-1816  0.326
2013 Tanpure RP, George CS, Strecker TE, Devkota L, Tidmore JK, Lin CM, Herdman CA, Macdonough MT, Sriram M, Chaplin DJ, Trawick ML, Pinney KG. Synthesis of structurally diverse benzosuberene analogues and their biological evaluation as anti-cancer agents. Bioorganic & Medicinal Chemistry. 21: 8019-32. PMID 24183586 DOI: 10.1016/J.Bmc.2013.08.035  0.813
2013 Hadimani MB, Macdonough MT, Ghatak A, Strecker TE, Lopez R, Sriram M, Nguyen BL, Hall JJ, Kessler RJ, Shirali AR, Liu L, Garner CM, Pettit GR, Hamel E, Chaplin DJ, ... ... Pinney KG, et al. Synthesis of a 2-aryl-3-aroyl indole salt (OXi8007) resembling combretastatin A-4 with application as a vascular disrupting agent. Journal of Natural Products. 76: 1668-78. PMID 24016002 DOI: 10.1021/Np400374W  0.81
2013 Macdonough MT, Strecker TE, Hamel E, Hall JJ, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and biological evaluation of indole-based, anti-cancer agents inspired by the vascular disrupting agent 2-(3'-hydroxy-4'-methoxyphenyl)-3-(3″,4″,5″-trimethoxybenzoyl)-6-methoxyindole (OXi8006). Bioorganic & Medicinal Chemistry. 21: 6831-43. PMID 23993969 DOI: 10.1016/J.Bmc.2013.07.028  0.74
2013 Song J, Jones LM, Chavarria GE, Charlton-Sevcik AK, Jantz A, Johansen A, Bayeh L, Soeung V, Snyder LK, Lade SD, Chaplin DJ, Trawick ML, Pinney KG. Small-molecule inhibitors of cathepsin L incorporating functionalized ring-fused molecular frameworks. Bioorganic & Medicinal Chemistry Letters. 23: 2801-7. PMID 23540644 DOI: 10.1016/J.Bmcl.2012.12.025  0.82
2013 Wittenborn T, Trawick ML, Pinney KG, Chaplin DJ, Siemann DW, Horsman MR. Abstract 5071: KGP94, a small-molecule cathepsin L inhibitor with antitumor activity. Cancer Research. 73: 5071-5071. DOI: 10.1158/1538-7445.Am2013-5071  0.353
2012 Song J, Jones LM, Kumar GD, Conner ES, Bayeh L, Chavarria GE, Charlton-Sevcik AK, Chen SE, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and biochemical evaluation of thiochromanone thiosemicarbazone analogues as inhibitors of cathepsin L. Acs Medicinal Chemistry Letters. 3: 450-3. PMID 24900494 DOI: 10.1021/Ml200299G  0.81
2012 Tanpure RP, George CS, Sriram M, Strecker TE, Tidmore JK, Hamel E, Charlton-Sevcik AK, Chaplin DJ, Trawick ML, Pinney KG. An Amino-Benzosuberene Analogue That Inhibits Tubulin Assembly and Demonstrates Remarkable Cytotoxicity. Medchemcomm. 3: 720-724. PMID 23772309 DOI: 10.1039/C2Md00318J  0.815
2012 Chavarria GE, Horsman MR, Arispe WM, Kumar GD, Chen SE, Strecker TE, Parker EN, Chaplin DJ, Pinney KG, Trawick ML. Initial evaluation of the antitumour activity of KGP94, a functionalized benzophenone thiosemicarbazone inhibitor of cathepsin L. European Journal of Medicinal Chemistry. 58: 568-72. PMID 23168380 DOI: 10.1016/J.Ejmech.2012.10.039  0.425
2011 Tanpure RP, Nguyen BL, Strecker TE, Aguirre S, Sharma S, Chaplin DJ, Siim BG, Hamel E, Lippert JW, Pettit GR, Trawick ML, Pinney KG. Regioselective synthesis of water-soluble monophosphate derivatives of combretastatin A-1. Journal of Natural Products. 74: 1568-74. PMID 21718055 DOI: 10.1021/Np200104T  0.827
2011 Mason RP, Zhao D, Liu L, Trawick ML, Pinney KG. A perspective on vascular disrupting agents that interact with tubulin: preclinical tumor imaging and biological assessment. Integrative Biology : Quantitative Biosciences From Nano to Macro. 3: 375-87. PMID 21321746 DOI: 10.1039/C0Ib00135J  0.407
2011 Trawick ML, Pinney KG, Chaplin DJ, Horsman MR, Chavarria GE, Arispe WM, Kumar GDK. Abstract 1416: Development and initial evaluation of the antitumor activity of a functionalized benzophenone thiosemicarbazone inhibitor of cathepsin L Cancer Research. 71: 1416-1416. DOI: 10.1158/1538-7445.Am2011-1416  0.508
2011 Allen PH, Bloom AJ, Bragg R, Brown RT, Burgos A, Bushby N, Clarke ML, Dudin LF, Ellames GJ, Gee AD, Gouverneur V, Harding JR, Harrowven DC, Herbert JM, Hickey MJ, ... ... Pinney KG, et al. 19th international isotope society (UK group) symposium: synthesis & applications of labelled compounds 2010 Journal of Labelled Compounds and Radiopharmaceuticals. 54: 387-398. DOI: 10.1002/jlcr.1878  0.792
2010 Kumar GD, Chavarria GE, Charlton-Sevcik AK, Yoo GK, Song J, Strecker TE, Siim BG, Chaplin DJ, Trawick ML, Pinney KG. Functionalized benzophenone, thiophene, pyridine, and fluorene thiosemicarbazone derivatives as inhibitors of cathepsin L. Bioorganic & Medicinal Chemistry Letters. 20: 6610-5. PMID 20933415 DOI: 10.1016/J.Bmcl.2010.09.026  0.82
2010 Tanpure RP, Strecker TE, Chaplin DJ, Siim BG, Trawick ML, Pinney KG. Regio- and stereospecific synthesis of mono-beta-d-glucuronic acid derivatives of combretastatin A-1. Journal of Natural Products. 73: 1093-101. PMID 20496923 DOI: 10.1021/Np100108E  0.807
2010 Kishore Kumar GD, Chavarria GE, Charlton-Sevcik AK, Arispe WM, Macdonough MT, Strecker TE, Chen SE, Siim BG, Chaplin DJ, Trawick ML, Pinney KG. Design, synthesis, and biological evaluation of potent thiosemicarbazone based cathepsin L inhibitors. Bioorganic & Medicinal Chemistry Letters. 20: 1415-9. PMID 20089402 DOI: 10.1016/J.Bmcl.2009.12.090  0.479
2010 MARSHALL JA, PINNEY KG. ChemInform Abstract: Stereoselective Synthesis of 2,5-Dihydrofurans by Sequential SN2′ Cleavage of Alkynyloxiranes and Ag+-Catalyzed Cyclization of the Allenylcarbinol Products. Cheminform. 25: no-no. DOI: 10.1002/chin.199416140  0.419
2009 Tanpure RP, Harkrider AR, Strecker TE, Hamel E, Trawick ML, Pinney KG. Application of the McMurry coupling reaction in the synthesis of tri- and tetra-arylethylene analogues as potential cancer chemotherapeutic agents. Bioorganic & Medicinal Chemistry. 17: 6993-7001. PMID 19733085 DOI: 10.1016/J.Bmc.2009.08.011  0.85
2009 Shirali A, Sriram M, Hall JJ, Nguyen BL, Guddneppanavar R, Hadimani MB, Ackley JF, Siles R, Jelinek CJ, Arthasery P, Brown RC, Murrell VL, McMordie A, Sharma S, Chaplin DJ, ... Pinney KG, et al. Development of synthetic methodology suitable for the radiosynthesis of combretastatin A-1 (CA1) and its corresponding prodrug CA1P. Journal of Natural Products. 72: 414-21. PMID 19161336 DOI: 10.1021/Np800661R  0.751
2009 Brown RT, Murrell VL, McMordie A, Sriram M, Pinney KG, Sharma S, Chaplinc DJ. Carbon-14 radiosynthesis of combretastatin A-1 (CA1) and its corresponding phosphate prodrug (CA1P) Journal of Labelled Compounds and Radiopharmaceuticals. 52: 567-570. DOI: 10.1002/Jlcr.1676  0.813
2008 Sriram M, Hall JJ, Grohmann NC, Strecker TE, Wootton T, Franken A, Trawick ML, Pinney KG. Design, synthesis and biological evaluation of dihydronaphthalene and benzosuberene analogs of the combretastatins as inhibitors of tubulin polymerization in cancer chemotherapy. Bioorganic & Medicinal Chemistry. 16: 8161-71. PMID 18722127 DOI: 10.1016/J.Bmc.2008.07.050  0.842
2008 Hall JJ, Sriram M, Strecker TE, Tidmore JK, Jelinek CJ, Kumar GD, Hadimani MB, Pettit GR, Chaplin DJ, Trawick ML, Pinney KG. Design, synthesis, biochemical, and biological evaluation of nitrogen-containing trifluoro structural modifications of combretastatin A-4. Bioorganic & Medicinal Chemistry Letters. 18: 5146-9. PMID 18710804 DOI: 10.1016/J.Bmcl.2008.07.070  0.831
2008 Siles R, Ackley JF, Hadimani MB, Hall JJ, Mugabe BE, Guddneppanavar R, Monk KA, Chapuis JC, Pettit GR, Chaplin DJ, Edvardsen K, Trawick ML, Garner CM, Pinney KG. Combretastatin dinitrogen-substituted stilbene analogues as tubulin-binding and vascular-disrupting agents. Journal of Natural Products. 71: 313-20. PMID 18303849 DOI: 10.1021/Np070377J  0.839
2007 Trawick ML, Arispe‐Angulo WM, Chen S, Siles R, Zhou M, Pinney KG. Kinetics of Thiosemicarbazone‐Based Inhibitors of Cathepsin L The Faseb Journal. 21. DOI: 10.1096/Fasebj.21.5.A642-A  0.774
2007 Chen S, Siles RE, Zhou M, Arispe WM, Lee H, Pinney KG, Trawick ML. Kinetic Studies of Potent Thiosemicarbazone Inhibitors of Cruzain The Faseb Journal. 21. DOI: 10.1096/Fasebj.21.5.A641-D  0.374
2006 Siles R, Chen SE, Zhou M, Pinney KG, Trawick ML. Design, synthesis, and biochemical evaluation of novel cruzain inhibitors with potential application in the treatment of Chagas' disease. Bioorganic & Medicinal Chemistry Letters. 16: 4405-9. PMID 16781147 DOI: 10.1016/J.Bmcl.2006.05.041  0.833
2006 Monk KA, Siles R, Hadimani MB, Mugabe BE, Ackley JF, Studerus SW, Edvardsen K, Trawick ML, Garner CM, Rhodes MR, Pettit GR, Pinney KG. Design, synthesis, and biological evaluation of combretastatin nitrogen-containing derivatives as inhibitors of tubulin assembly and vascular disrupting agents. Bioorganic & Medicinal Chemistry. 14: 3231-44. PMID 16442292 DOI: 10.1016/J.Bmc.2005.12.033  0.838
2006 Brien KA, Garner CM, Pinney KG. Synthesis and characterization of 2,6-bis-hydrazinopyridine, and its conversion to 2,6-bis-pyrazolylpyridines Tetrahedron. 62: 3663-3666. DOI: 10.1016/J.Tet.2006.01.086  0.371
2006 Miranda MG, Norton EJ, Feazell RP, Klausmeyer KK, Pinney KG. Synthesis and crystal structures of two novel 3,4,5-trimethoxyphenyl derivatives from (Z)-1-[(2′,3′-dinitro-4′-methoxy)-phenyl]-2- [(3″,4″,5″-trimethoxy)-phenyl]ethene Journal of Chemical Crystallography. 36: 309-314. DOI: 10.1007/S10870-005-9065-1  0.396
2004 Sheng Y, Hua J, Pinney KG, Garner CM, Kane RR, Prezioso JA, Chaplin DJ, Edvardsen K. Combretastatin family member OXI4503 induces tumor vascular collapse through the induction of endothelial apoptosis. International Journal of Cancer. Journal International Du Cancer. 111: 604-10. PMID 15239140 DOI: 10.1002/Ijc.20297  0.316
2004 Dorsey JM, Miranda MG, Cozzi NV, Pinney KG. Synthesis and biological evaluation of 2-(4-fluorophenoxy)-2-phenyl-ethyl piperazines as serotonin-selective reuptake inhibitors with a potentially improved adverse reaction profile. Bioorganic & Medicinal Chemistry. 12: 1483-91. PMID 15018922 DOI: 10.1016/J.Bmc.2003.12.021  0.555
2003 Hadimani MB, Hua J, Jonklaas MD, Kessler RJ, Sheng Y, Olivares A, Tanpure RP, Weiser A, Zhang J, Edvardsen K, Kane RR, Pinney KG. Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4. Bioorganic & Medicinal Chemistry Letters. 13: 1505-8. PMID 12699742 DOI: 10.1016/S0960-894X(03)00206-3  0.82
2003 Monk KA, Siles R, Pinney KG, Garner CM. Synthesis of 4-methoxy-3,5-dinitrobenzaldehyde: A correction to supposed tele nucleophilic aromatic substitution Tetrahedron Letters. 44: 3759-3761. DOI: 10.1016/S0040-4039(03)00751-2  0.797
2003 Ghatak A, Dorsey JM, Garner CM, Pinney KG. Synthesis of methoxy and hydroxy containing tetralones: Versatile intermediates for the preparation of biologically relevant molecules Tetrahedron Letters. 44: 4145-4148. DOI: 10.1016/S0040-4039(03)00715-9  0.388
2002 Hadimani MB, Kessler RJ, Kautz JA, Ghatak A, Shirali AR, O'Dell H, Garner CM, Pinney KG. 2-(3-tert-Butyldimethylsiloxy-4-methoxyphenyl)-6-methoxy-3-(3,4,5-trimethoxybenzoyl)indole. Acta Crystallographica. Section C, Crystal Structure Communications. 58: o330-2. PMID 12050432 DOI: 10.1107/S0108270102003669  0.759
2002 Hadimani MB, Kessler RJ, Kautz JA, Ghatak A, Shirali AR, O'Dell H, Garner CM, Pinney KG. 2-(3-tert-butyldimethylsiloxy-4-methoxyphenyl)-6-methoxy-3-(3,4, 5-trimethoxybenzoyl)indole Acta Crystallographica Section C: Crystal Structure Communications. 58: o330-o332. DOI: 10.1107/S0108270102003669  0.802
2000 Pinney KG, Mejia MP, Villalobos VM, Rosenquist BE, Pettit GR, Verdier-Pinard P, Hamel E. Synthesis and biological evaluation of aryl azide derivatives of combretastatin A-4 as molecular probes for tubulin. Bioorganic & Medicinal Chemistry. 8: 2417-25. PMID 11058036 DOI: 10.1016/S0968-0896(00)00176-0  0.519
1999 Pinney KG, Bounds AD, Dingeman KM, Mocharla VP, Pettit GR, Bai R, Hamel E. A new anti-tubulin agent containing the benzo[b]thiophene ring system. Bioorganic & Medicinal Chemistry Letters. 9: 1081-6. PMID 10328289 DOI: 10.1016/S0960-894X(99)00143-2  0.5
1998 Mullica DF, Pinney KG, Mejia P, Rosenquist BE, Sappenfield EL. (E)-1-(3-Methoxy-4-nitrophenyl)-2-(3,4,5-trimethoxyphenyl)ethene Acta Crystallographica Section C: Crystal Structure Communications. 54: 695-697. DOI: 10.1107/S0108270197019902  0.354
1998 Mullica DF, Pinney KG, Mocharla VP, Dingeman KM, Bounds AD, Sappenfield EL. Characterization and structural analyses of trimethoxy and triethoxybenzo[b]thiophene Journal of Chemical Crystallography. 28: 289-295. DOI: 10.1023/A:1021853320007  0.314
1996 Mullica DF, Pinney KG, Dingeman KM, Bounds AD, Sappenfield EL. X-ray structures of two methoxybenzo[b]thiophenes Journal of Chemical Crystallography. 26: 801-806. DOI: 10.1007/Bf01670312  0.303
1993 Kym PR, Anstead GM, Pinney KG, Wilson SR, Katzenellenbogen JA. Molecular structures, conformational analysis, and preferential modes of binding of 3-aroyl-2-arylbenzo[b]thiophene estrogen receptor ligands: LY117018 and aryl azide photoaffinity labeling analogs. Journal of Medicinal Chemistry. 36: 3910-22. PMID 8254621 DOI: 10.1021/Jm00076A020  0.523
1993 Marshall JA, Pinney KG. Stereoselective synthesis of 2,5-dihydrofurans by sequential SN2' cleavage of alkynyloxiranes and silver(I)-catalyzed cyclization of the allenylcarbinol products Journal of Organic Chemistry. 58: 7180-7184. DOI: 10.1021/Jo00077A048  0.469
1992 Pinney KG, Carlson KE, Katzenellenbogen JA. Nonsteroidal estrogens bearing acyl azide functions: potential electrophilic and photoaffinity labeling agents for the estrogen receptor. Steroids. 57: 222-32. PMID 1488784 DOI: 10.1016/0039-128X(92)90106-J  0.508
1991 Pinney KG, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Efficient and selective photoaffinity labeling of the estrogen receptor using two nonsteroidal ligands that embody aryl azide or tetrafluoroaryl azide photoreactive functions. Biochemistry. 30: 2421-31. PMID 2001370 DOI: 10.1021/Bi00223A018  0.486
1991 Pinney KG, Katzenellenbogen JA. Synthesis of a tetrafluoro-substituted aryl azide and its protio analog as photoaffinity labeling reagents for the estrogen receptor The Journal of Organic Chemistry. 56: 3125-3133. DOI: 10.1021/Jo00009A037  0.56
1991 Pinney KG, Katzenellenbogen JA. Synthesis of a tetrafluoro-substituted aryl azide and its protio analogue as photoaffinity labeling reagents for the estrogen receptor Journal of Organic Chemistry. 56: 3125-3133.  0.421
1990 Pomper MG, Pinney KG, Carlson KE, van Brocklin H, Mathias CJ, Welch MJ, Katzenellenbogen JA. Target tissue uptake selectivity of three fluorine-substituted progestins: potential imaging agents for receptor-positive breast tumors. International Journal of Radiation Applications and Instrumentation. Part B, Nuclear Medicine and Biology. 17: 309-19. PMID 2341287 DOI: 10.1016/0883-2897(90)90058-9  0.614
1990 Pinney KG, Carlson KE, Katzenellenbogen JA. [3H]DU41165: a high affinity ligand and novel photoaffinity labeling reagent for the progesterone receptor. Journal of Steroid Biochemistry. 35: 179-89. PMID 2308335 DOI: 10.1016/0022-4731(90)90272-T  0.457
1990 Anstead GM, Peterson CS, Pinney KG, Wilson SR, Katzenellenbogen JA. Torsionally and hydrophobically modified 2,3-diarylindenes as estrogen receptor ligands. Journal of Medicinal Chemistry. 33: 2726-34. PMID 2213825 DOI: 10.1021/Jm00172A008  0.53
Show low-probability matches.