C. Robin Ganellin, Ph.D.

Affiliations: 
1958-1986 Smith Kline and French 
 1986- University College London, London, United Kingdom 
Area:
histamines, Tagamet
Website:
https://www.acsmedchem.org/?nd=Ganellin
Google:
"C. Ganellin"
Bio:

1980 ACS Medicinal Chemistry Hall of Fame

Mean distance: 7.96
 
SNBCP
BETA: Related publications

Publications

You can help our author matching system! If you notice any publications incorrectly attributed to this author, please sign in and mark matches as correct or incorrect.

Yang D, Arifhodzic L, Ganellin CR, et al. (2013) Further studies on bis-charged tetraazacyclophanes as potent inhibitors of small conductance Ca(2+)-activated K+ channels. European Journal of Medicinal Chemistry. 63: 907-23
Ganellin CR. (2011) Personal reflections on Sir James Black (1924-2010) and histamine. Inflammation Research : Official Journal of the European Histamine Research Society ... [Et Al.]. 60: 103-10
Levoin N, Calmels T, Poupardin-Olivier O, et al. (2008) Refined docking as a valuable tool for lead optimization: application to histamine H3 receptor antagonists. Archiv Der Pharmazie. 341: 610-23
Das BC, Madhukumar AV, Anguiano J, et al. (2008) Synthesis of novel ketoconazole derivatives as inhibitors of the human Pregnane X Receptor (PXR; NR1I2; also termed SXR, PAR). Bioorganic & Medicinal Chemistry Letters. 18: 3974-7
Fletcher DI, Ganellin CR, Piergentili A, et al. (2007) Synthesis and pharmacological testing of polyaminoquinolines as blockers of the apamin-sensitive Ca2+-activated K+ channel (SK(Ca)). Bioorganic & Medicinal Chemistry. 15: 5457-79
Shah MM, Javadzadeh-Tabatabaie M, Benton DC, et al. (2006) Enhancement of hippocampal pyramidal cell excitability by the novel selective slow-afterhyperpolarization channel blocker 3-(triphenylmethylaminomethyl)pyridine (UCL2077). Molecular Pharmacology. 70: 1494-502
Parsons ME, Ganellin CR. (2006) Histamine and its receptors. British Journal of Pharmacology. 147: S127-35
Power EC, Ganellin CR, Benton DC. (2006) Partial structures of ketoconazole as modulators of the large conductance calcium-activated potassium channel (BK(Ca)). Bioorganic & Medicinal Chemistry Letters. 16: 887-90
Apelt J, Grassmann S, Ligneau X, et al. (2005) Search for histamine H3 receptor antagonists with combined inhibitory potency at Ntau-methyltransferase: ether derivatives. Die Pharmazie. 60: 97-106
Grassmann S, Apelt J, Ligneau X, et al. (2004) Search for histamine H(3) receptor ligands with combined inhibitory potency at histamine N-methyltransferase: omega-piperidinoalkanamine derivatives. Archiv Der Pharmazie. 337: 533-45
See more...