Year |
Citation |
Score |
2015 |
Cushing TD, Hao X, Shin Y, Andrews K, Brown M, Cardozo M, Chen Y, Duquette J, Fisher B, Gonzalez-Lopez de Turiso F, He X, Henne KR, Hu YL, Hungate R, Johnson MG, ... ... Reichelt A, et al. Discovery and in vivo evaluation of (S)-N-(1-(7-fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and related PI3Kδ inhibitors for inflammation and autoimmune disease. Journal of Medicinal Chemistry. 58: 480-511. PMID 25469863 DOI: 10.1021/Jm501624R |
0.322 |
|
2014 |
Rzasa RM, Frohn MJ, Andrews KL, Chmait S, Chen N, Clarine JG, Davis C, Eastwood HA, Horne DB, Hu E, Jones AD, Kaller MR, Kunz RK, Miller S, Monenschein H, ... ... Reichelt A, et al. Synthesis and preliminary biological evaluation of potent and selective 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors with improved solubility. Bioorganic & Medicinal Chemistry. 22: 6570-85. PMID 25456383 DOI: 10.1016/J.Bmc.2014.10.013 |
0.354 |
|
2014 |
Reichelt A, Bailis JM, Bartberger MD, Yao G, Shu H, Kaller MR, Allen JG, Weidner MF, Keegan KS, Dao JH. Synthesis and structure-activity relationship of trisubstituted thiazoles as Cdc7 kinase inhibitors. European Journal of Medicinal Chemistry. 80: 364-82. PMID 24793884 DOI: 10.1016/J.Ejmech.2014.04.013 |
0.346 |
|
2013 |
Bryan MC, Falsey JR, Frohn M, Reichelt A, Yao G, Bartberger MD, Bailis JM, Zalameda L, Miguel TS, Doherty EM, Allen JG. N-substituted azaindoles as potent inhibitors of Cdc7 kinase. Bioorganic & Medicinal Chemistry Letters. 23: 2056-60. PMID 23481650 DOI: 10.1016/J.Bmcl.2013.02.007 |
0.384 |
|
2010 |
Thiel OR, Achmatowicz MM, Reichelt A, Larsen RD. Palladium-catalyzed coupling of aldehyde-derived hydrazones: practical synthesis of triazolopyridines and related heterocycles. Angewandte Chemie (International Ed. in English). 49: 8395-8. PMID 20661974 DOI: 10.1002/Anie.201001999 |
0.417 |
|
2010 |
Reichelt A, Falsey JR, Rzasa RM, Thiel OR, Achmatowicz MM, Larsen RD, Zhang D. Palladium-catalyzed chemoselective monoarylation of hydrazides for the synthesis of [1,2,4]triazolo[4,3-a]pyridines. Organic Letters. 12: 792-5. PMID 20099864 DOI: 10.1021/Ol902868Q |
0.482 |
|
2010 |
Reichelt A, Falsey JR, Rzasa RM, Thiel OR, Achmatowicz MM, Larsen RD, Zhang D. Triazolopyridines via Selective Palladium-Catalyzed Monoarylationof Hydrazides Synfacts. 2010: 522-522. DOI: 10.1055/S-0029-1219725 |
0.322 |
|
2010 |
Reichelt A, Bur SK, Martin SF. ChemInform Abstract: Applications of Vinylogous Mannich Reactions. Total Synthesis of the Angiotensin Converting Enzyme Inhibitor (-)-A58365A. Cheminform. 33: no-no. DOI: 10.1002/CHIN.200250181 |
0.493 |
|
2010 |
Thiel OR, Achmatowicz MM, Reichelt A, Larsen RD. Cover Picture: Palladium-Catalyzed Coupling of Aldehyde-Derived Hydrazones: Practical Synthesis of Triazolopyridines and Related Heterocycles (Angew. Chem. Int. Ed. 45/2010) Angewandte Chemie International Edition. 49: 8277-8277. DOI: 10.1002/Anie.201004361 |
0.409 |
|
2010 |
Thiel OR, Achmatowicz MM, Reichelt A, Larsen RD. Titelbild: Palladium-Catalyzed Coupling of Aldehyde-Derived Hydrazones: Practical Synthesis of Triazolopyridines and Related Heterocycles (Angew. Chem. 45/2010) Angewandte Chemie. 122: 8453-8453. DOI: 10.1002/Ange.201004361 |
0.416 |
|
2009 |
Evans DA, Welch DS, Speed AW, Moniz GA, Reichelt A, Ho S. An aldol-based synthesis of (+)-peloruside a, a potent microtubule stabilizing agent. Journal of the American Chemical Society. 131: 3840-1. PMID 19249829 DOI: 10.1021/Ja900020A |
0.438 |
|
2009 |
Evans DA, Welch DS, Speed AWH, Moniz GA, Reichelt A, Ho S. Synthesis of (+)-Peloruside A Synfacts. 2009: 945-945. DOI: 10.1055/S-0029-1217617 |
0.465 |
|
2008 |
Herberich B, Cao GQ, Chakrabarti PP, Falsey JR, Pettus L, Rzasa RM, Reed AB, Reichelt A, Sham K, Thaman M, Wurz RP, Xu S, Zhang D, Hsieh F, Lee MR, et al. Discovery of highly selective and potent p38 inhibitors based on a phthalazine scaffold. Journal of Medicinal Chemistry. 51: 6271-9. PMID 18817365 DOI: 10.1021/Jm8005417 |
0.358 |
|
2006 |
Reichelt A, Martin SF. Synthesis and properties of cyclopropane-derived peptidomimetics. Accounts of Chemical Research. 39: 433-42. PMID 16846207 DOI: 10.1021/Ar030255S |
0.516 |
|
2006 |
Simila ST, Reichelt A, Martin SF. Synthetic studies toward the immunosuppressant FR901483. Facile construction of the azatricyclic skeleton Tetrahedron Letters. 47: 2933-2936. DOI: 10.1016/J.Tetlet.2006.02.116 |
0.484 |
|
2002 |
Reichelt A, Gaul C, Frey RR, Kennedy A, Martin SF. Design, synthesis, and evaluation of matrix metalloprotease inhibitors bearing cyclopropane-derived peptidomimetics as P1' and P2' replacements. The Journal of Organic Chemistry. 67: 4062-75. PMID 12054939 DOI: 10.1021/Jo0110698 |
0.472 |
|
2002 |
Reichelt A, Bur SK, Martin SF. Applications of vinylogous Mannich reactions. Total synthesis of the angiotensin converting enzyme inhibitor (-)-A58365A Tetrahedron. 58: 6323-6328. DOI: 10.1016/S0040-4020(02)00631-2 |
0.663 |
|
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