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Ales Machara - Publications

Affiliations: 
2009- Brock University, Saint Catharines, Ontario, Canada 
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23/40 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2018 Machara A, Křivánek J, Dolejšová K, Havlíčková J, Bednárová L, Hanus R, Majer P, Kyjaková P. Identification and Enantiodivergent Synthesis of (5 Z,9 S)-Tetradec-5-en-9-olide, a Queen-Specific Volatile of the Termite Silvestritermes minutus. Journal of Natural Products. PMID 30299957 DOI: 10.1021/Acs.Jnatprod.8B00632  0.307
2016 Kožíšek M, Štěpánek O, Parkan K, Berenguer Albiñana C, Pávová M, Weber J, Krӓusslich HG, Konvalinka J, Machara A. Synthesis and evaluation of 2-pyridinylpyrimidines as inhibitors of HIV-1 structural protein assembly. Bioorganic & Medicinal Chemistry Letters. PMID 27353536 DOI: 10.1016/J.Bmcl.2016.06.039  0.343
2016 Hudlicky T, Ann A. Endoma-Arias M, Machara A, Phillip Cox D. Synthesis of Noroxymorphone by N-Demethylation/ Intramolecular Acylation of Oxymorphone Catalyzed by Iron(II) Chloride Heterocycles. 93: 824. DOI: 10.3987/Com-15-S(T)63  0.535
2016 Machara A, Hudlický T, Endoma-Arias M, Císařova I, Cox D. Synthesis of Nororipavine and Noroxymorphone via N- and O-Demethylation of Iron Tricarbonyl Complex of Thebaine Synthesis. 48: e1-e1. DOI: 10.1055/S-0035-1562345  0.582
2016 Albiñana CB, Hayward JJ, Hudlicky T, Machara A. Reinvestigation of acetylation of 3,4-dihydroxybenzaldehyde and reconciliation of previously reported analytical data Tetrahedron Letters. 57: 1019-1021. DOI: 10.1016/J.Tetlet.2016.01.075  0.377
2016 Machara A, Konvalinka J, Kotora M. A MODULAR SYNTHESIS OFN-BENZOTRIAZOLE UREAS USING ALKYLATION OF 5-NITROBENZOTRIAZOLE Chemistryselect. 1: 101-107. DOI: 10.1002/slct.201600025  0.391
2016 Machara A, Endoma-Arias MAA, Císařová I, Cox DP, Hudlicky T. Direct Synthesis of Noroxymorphone from Thebaine: Unusual CeIV Oxidation of a Methoxydiene-Iron Complex to an Enone-γ-Nitrate European Journal of Organic Chemistry. 2016: 1500-1503. DOI: 10.1002/Ejoc.201600153  0.523
2016 Machara A, Konvalinka J, Kotora M. ChemInform Abstract: A Modular Synthesis of N-Benzotriazole Ureas Using Alkylation of 5-Nitrobenzotriazole. Cheminform. 47. DOI: 10.1002/chin.201626113  0.419
2016 Machara A, Endoma-Arias MAA, Cisarova I, Cox DP, Hudlicky T. ChemInform Abstract: Direct Synthesis of Noroxymorphone from Thebaine: Unusual CeIVOxidation of a Methoxydiene-Iron Complex to an Enone-γ-nitrate. Cheminform. 47. DOI: 10.1002/chin.201619181  0.401
2015 Machara A, Werner L, Leisch H, Carroll RJ, Adams DR, Haque DM, Cox DP, Hudlicky T. Synthesis of Naltrexone and (R)-Methylnaltrexone from Oripavine via Direct Oxidation of Its Quaternary Salts Synlett. 26: 2101-2108. DOI: 10.1055/S-0034-1378808  0.596
2014 Murphy B, Šnajdr I, Machara A, Endoma-Arias MAA, Stamatatos TC, Cox DP, Hudlický T. Conversion of thebaine to oripavine and other useful intermediates for the semisynthesis of opiate-derived agents: Synthesis of hydromorphone Advanced Synthesis and Catalysis. 356: 2679-2687. DOI: 10.1002/Adsc.201400445  0.546
2013 MacHara A, Svoboda J. Thiophenium-ylides: Synthesis and reactivity Chemical Papers. 67: 59-65. DOI: 10.2478/s11696-012-0222-7  0.314
2012 MacHara A, Cox DP, Hudlicky T. Direct synthesis of naltrexone by palladium-catalyzed N-demethylation/ acylation of oxymorphone: The benefit of C-H activation and the intramolecular acyl transfer from C-14 hydroxy Advanced Synthesis and Catalysis. 354: 2713-2718. DOI: 10.1002/Adsc.201200677  0.537
2012 Werner L, Wernerova M, MacHara A, Endoma-Arias MA, Duchek J, Adams DR, Cox DP, Hudlicky T. Unexpected N-demethylation of oxymorphone and oxycodone N-oxides mediated by the burgess reagent: Direct synthesis of naltrexone, naloxone, and other antagonists from oxymorphone Advanced Synthesis and Catalysis. 354: 2706-2712. DOI: 10.1002/Adsc.201200676  0.671
2012 MacHara A, Werner L, Endoma-Arias MA, Cox DP, Hudlicky T. Improved synthesis of buprenorphine from thebaine and/or oripavine via palladium-catalyzed N-demethylation/acylation and/or concomitant O-demethylation Advanced Synthesis and Catalysis. 354: 613-626. DOI: 10.1002/Adsc.201100807  0.663
2011 Werner L, Machara A, Sullivan B, Carrera I, Moser M, Adams DR, Hudlicky T, Andraos J. Several generations of chemoenzymatic synthesis of oseltamivir (Tamiflu): evolution of strategy, quest for a process-quality synthesis, and evaluation of efficiency metrics. The Journal of Organic Chemistry. 76: 10050-67. PMID 22007598 DOI: 10.1021/Jo2018872  0.62
2011 Werner L, Machara A, Adams DR, Cox DP, Hudlicky T. Synthesis of buprenorphine from oripavine via N-demethylation of oripavine quaternary salts. The Journal of Organic Chemistry. 76: 4628-34. PMID 21495679 DOI: 10.1021/Jo200567N  0.665
2011 Machara A, Cox DP, Hudlicky T. Synthesis of nalbuphine from oripavine via N-demethylation of N-cyclobutylmethyl oripavine Heterocycles. 84: 615-623. DOI: 10.3987/Com-11-S(P)32  0.523
2011 Werner L, Machara A, Adams DR, Cox DP, Hudlicky T. Synthesis of Buprenorphine Synfacts. 2011: 817-817. DOI: 10.1055/S-0030-1260675  0.63
2010 Werner L, Machara A, Hudlicky T. Short chemoenzymatic azide-free synthesis of oseltamivir (tamiflu): Approaching the potential for process efficiency Advanced Synthesis and Catalysis. 352: 195-200. DOI: 10.1002/Adsc.200900844  0.638
2009 Machara A, Kozmík V, Pojarová M, Dvořáková H, Svoboda J. Preparation and rearrangement study of novel thiophenium-and selenophenium-ylides Collection of Czechoslovak Chemical Communications. 74: 785-798. DOI: 10.1135/Cccc2009001  0.337
2007 Machara A, Pojarová M, Svoboda J. Synthesis and cycloaddition reaction of 3-vinylthieno[3,2-b][1] benzothiophene Collection of Czechoslovak Chemical Communications. 72: 952-964. DOI: 10.1135/Cccc20070952  0.378
2004 Machara A, Kurfürst M, Kozmík V, Petříčková H, Dvořáková H, Svoboda J. A nonconcerted cycloaddition of fused 2-vinylthiophenes with dimethyl acetylenedicarboxylate Tetrahedron Letters. 45: 2189-2192. DOI: 10.1016/J.Tetlet.2004.01.030  0.302
Low-probability matches (unlikely to be authored by this person)
2017 Zábranský M, Machara A, Císařová I, Štěpnička P. Palladium(II) Complexes of Homologated Ferrocene Phosphanylether and Thioether Ligands European Journal of Inorganic Chemistry. 2017: 4850-4860. DOI: 10.1002/Ejic.201701057  0.295
2019 Zima V, Albiñana CB, Rojíková K, Pokorná J, Pachl P, Řezáčová P, Hudlicky J, Navrátil V, Majer P, Konvalinka J, Kožíšek M, Machara A. Investigation of flexibility of neuraminidase 150-loop using tamiflu derivatives in influenza A viruses H1N1 and H5N1. Bioorganic & Medicinal Chemistry. PMID 31128993 DOI: 10.1016/J.Bmc.2019.05.024  0.265
2018 Kožíšek M, Navrátil V, Rojíková K, Pokorná J, Albiňana CB, Pachl P, Zemanová J, Machara A, Šácha P, Hudlický J, Císařová I, Řezáčová P, Konvalinka J. DNA-linked inhibitor antibody assay (DIANA) as a new method for screening influenza neuraminidase inhibitors. The Biochemical Journal. PMID 30404922 DOI: 10.2210/Pdb6G01/Pdb  0.265
2016 Albiñana CB, Machara A, Řezáčová P, Pachl P, Konvalinka J, Kožíšek M. Kinetic, thermodynamic and structural analysis of tamiphosphor binding to neuraminidase of H1N1 (2009) pandemic influenza. European Journal of Medicinal Chemistry. 121: 100-109. PMID 27236066 DOI: 10.1016/J.Ejmech.2016.05.016  0.264
2020 Zima V, Radilová K, Kožíšek M, Albiñana CB, Karlukova E, Brynda J, Fanfrlík J, Flieger M, Hodek J, Weber J, Majer P, Konvalinka J, Machara A. Unraveling the anti-influenza effect of flavonoids: Experimental validation of luteolin and its congeners as potent influenza endonuclease inhibitors. European Journal of Medicinal Chemistry. 208: 112754. PMID 32883638 DOI: 10.1016/J.Ejmech.2020.112754  0.253
2015 Machara A, Lux V, Kozisek M, Grantz-Saskova K, Stepanek O, Kotora M, Parkan K, Pavova M, Glass B, Sehr P, Lewis J, Muller B, Kraeusslich HG, Konvalinka J. Specific inhibitors of HIV capsid assembly binding to the C-terminal domain of the capsid protein: evaluation of 2-arylquinazolines as potential antiviral compounds. Journal of Medicinal Chemistry. PMID 26685880 DOI: 10.1021/Acs.Jmedchem.5B01089  0.238
2018 Pokorná J, Pachl P, Karlukova E, Hejdánek J, Řezáčová P, Machara A, Hudlický J, Konvalinka J, Kožíšek M. Kinetic, Thermodynamic, and Structural Analysis of Drug Resistance Mutations in Neuraminidase from the 2009 Pandemic Influenza Virus. Viruses. 10. PMID 29933553 DOI: 10.2210/Pdb5Nzf/Pdb  0.224
2021 Reiberger R, Radilová K, Kráľ M, Zima V, Majer P, Brynda J, Dračínský M, Konvalinka J, Kožíšek M, Machara A. Synthesis and In Vitro Evaluation of C-7 and C-8 Luteolin Derivatives as Influenza Endonuclease Inhibitors. International Journal of Molecular Sciences. 22. PMID 34299354 DOI: 10.3390/ijms22147735  0.195
2022 Tupec M, Culka M, Machara A, Macháček S, Bím D, Svatoš A, Rulíšek L, Pichová I. Understanding desaturation/hydroxylation activity of castor stearoyl Δ-Desaturase through rational mutagenesis. Computational and Structural Biotechnology Journal. 20: 1378-1388. PMID 35386101 DOI: 10.1016/j.csbj.2022.03.010  0.156
2022 Osifová Z, Reiberger R, Císařová I, Machara A, Dračínský M. Diketo-Ketoenol Tautomers in Curcuminoids: Synthesis, Separation of Tautomers, and Kinetic and Structural Studies. The Journal of Organic Chemistry. 87: 10309-10318. PMID 35895908 DOI: 10.1021/acs.joc.2c01357  0.154
2022 Radilová K, Zima V, Kráľ M, Machara A, Majer P, Hodek J, Weber J, Brynda J, Strmeň T, Konvalinka J, Kožíšek M. Thermodynamic and structural characterization of an optimized peptide-based inhibitor of the influenza polymerase PA-PB1 subunit interaction. Antiviral Research. 208: 105449. PMID 36265804 DOI: 10.1016/j.antiviral.2022.105449  0.108
2020 Hejdánek J, Radilová K, Pachl P, Hodek J, Machara A, Weber J, Řezáčová P, Konvalinka J, Kožíšek M. structural characterization of the interaction between the C-terminal domain of the influenza polymerase PA subunit and an optimized small peptide inhibitor. Antiviral Research. 185: 104971. PMID 33166574 DOI: 10.1016/j.antiviral.2020.104971  0.097
2021 Milacek M, Bittova L, Tumova S, Luksan O, Hanus R, Kyjakova P, Machara A, Marek A, Jindra M. Binding of de novo synthesized radiolabeled juvenile hormone (JH III) by JH receptors from the Cuban subterranean termite Prorhinotermes simplex and the German cockroach Blattella germanica. Insect Biochemistry and Molecular Biology. 139: 103671. PMID 34656795 DOI: 10.1016/j.ibmb.2021.103671  0.094
2023 Cudlman L, Machara A, Vrkoslav V, Polášek M, Bosáková Z, Blanksby SJ, Cvačka J. Characterization of Triacylglycerol Estolide Isomers Using High-Resolution Tandem Mass Spectrometry with Nanoelectrospray Ionization. Biomolecules. 13. PMID 36979410 DOI: 10.3390/biom13030475  0.085
2021 Yuvaraj JK, Roberts RE, Sonntag Y, Hou XQ, Grosse-Wilde E, Machara A, Zhang DD, Hansson BS, Johanson U, Löfstedt C, Andersson MN. Putative ligand binding sites of two functionally characterized bark beetle odorant receptors. Bmc Biology. 19: 16. PMID 33499862 DOI: 10.1186/s12915-020-00946-6  0.067
2023 Macháček S, Tupec M, Horáček N, Halmová M, Roy A, Machara A, Kyjaková P, Lukšan O, Pichová I, Hanus R. Evolution of Linoleic Acid Biosynthesis Paved the Way for Ecological Success of Termites. Molecular Biology and Evolution. 40. PMID 37043525 DOI: 10.1093/molbev/msad087  0.062
2000 Machara A, Fitzgerald PJ. Coronary calcification: Assessment by intravascular ultrasound imaging Zeitschrift Fur Kardiologie. 89: II112-II116. PMID 10769413  0.027
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