Year |
Citation |
Score |
2024 |
Tang SA, Fults A, Boyd SR, Gattu N, Tran KA, Fan J, MacKenzie KR, Palzkill T, Young DW, Chamakuri S. Expanding Complex Morpholines Using Systematic Chemical Diversity. Organic Letters. PMID 38506470 DOI: 10.1021/acs.orglett.4c00528 |
0.318 |
|
2023 |
Jimmidi R, Chamakuri S, Lu S, Ucisik MN, Chen PJ, Bohren KM, Moghadasi SA, Versteeg L, Nnabuife C, Li JY, Qin X, Chen YC, Faver JC, Nyshadham P, Sharma KL, et al. DNA-encoded chemical libraries yield non-covalent and non-peptidic SARS-CoV-2 main protease inhibitors. Communications Chemistry. 6: 164. PMID 37542196 DOI: 10.1038/s42004-023-00961-y |
0.774 |
|
2021 |
Chamakuri S, Lu S, Ucisik MN, Bohren KM, Chen YC, Du HC, Faver JC, Jimmidi R, Li F, Li JY, Nyshadham P, Palmer SS, Pollet J, Qin X, Ronca SE, et al. DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 M inhibitors. Proceedings of the National Academy of Sciences of the United States of America. 118. PMID 34426525 DOI: 10.1073/pnas.2111172118 |
0.768 |
|
2019 |
Chamakuri S, Jain P, Guduru SRK, Arney JW, MacKenzie KR, Santini C, Young DW. Correction to Synthesis of Enantiomerically Pure 6-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production. The Journal of Organic Chemistry. PMID 30855144 DOI: 10.1021/Acs.Joc.9B00594 |
0.374 |
|
2019 |
Jain P, Raji IO, Chamakuri S, MacKenzie KR, Ebright BT, Santini C, Young DW. Synthesis of Enantiomerically Pure 5-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production. The Journal of Organic Chemistry. PMID 30848904 DOI: 10.1021/Acs.Joc.9B00148 |
0.414 |
|
2018 |
Guduru SKR, Chamakuri S, Raji IO, MacKenzie KR, Santini C, Young DW. Synthesis of Enantiomerically Pure 3-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production. The Journal of Organic Chemistry. PMID 30180575 DOI: 10.1021/Acs.Joc.8B01708 |
0.43 |
|
2018 |
Chamakuri S, Jain P, Guduru SKR, Arney JW, MacKenzie K, Santini C, Young DW. Synthesis of Enantiomerically Pure 6-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production. The Journal of Organic Chemistry. PMID 29751727 DOI: 10.1021/Acs.Joc.8B00854 |
0.466 |
|
2017 |
Jogula S, Soorneedi AR, Gaddam J, Chamakuri S, Deora GS, Indarapu RK, Ramgopal MK, Dravida S, Arya P. Geldanamycin-inspired compounds induce direct trans-differentiation of human mesenchymal stem cells to neurons. European Journal of Medicinal Chemistry. 135: 110-116. PMID 28441579 DOI: 10.1016/J.Ejmech.2017.03.082 |
0.604 |
|
2015 |
Chamakuri S, Jogula S, Arya P. Regio- and Stereocontrolled Dieckmann Approach to Treprostinil-Inspired, Polycyclic Scaffold For Building Macrocyclic Diversity. Acs Combinatorial Science. 17: 437-41. PMID 26167941 DOI: 10.1021/Acscombsci.5B00076 |
0.712 |
|
2014 |
Aeluri M, Chamakuri S, Dasari B, Guduru SK, Jimmidi R, Jogula S, Arya P. Small molecule modulators of protein-protein interactions: selected case studies. Chemical Reviews. 114: 4640-94. PMID 24673632 DOI: 10.1021/Cr4004049 |
0.419 |
|
2013 |
Reddy Guduru SK, Chamakuri S, Chandrasekar G, Kitambi SS, Arya P. Tetrahydroquinoline-derived macrocyclic toolbox: the discovery of antiangiogenesis agents in zebrafish assay. Acs Medicinal Chemistry Letters. 4: 666-70. PMID 24900727 DOI: 10.1021/Ml400026N |
0.726 |
|
2013 |
Chamakuri S, Guduru SKR, Pamu S, Chandrasekar G, Kitambi SS, Arya P. A Modular Approach to Build Macrocyclic Diversity in Aminoindoline Scaffolds Identifies Antiangiogenesis Agents from a Zebrafish Assay European Journal of Organic Chemistry. 2013: 3959-3964. DOI: 10.1002/Ejoc.201300409 |
0.658 |
|
2010 |
Kumar KS, Chamakuri S, Vishweshwar P, Iqbal J, Pal M. AlCl3-induced (hetero)arylation of thienopyrimidine ring: a new synthesis of 4-substituted thieno[2,3-d]pyrimidines Tetrahedron Letters. 51: 3269-3273. DOI: 10.1016/J.Tetlet.2010.04.057 |
0.387 |
|
Low-probability matches (unlikely to be authored by this person) |
2022 |
Moghadasi SA, Esler MA, Otsuka Y, Becker JT, Moraes SN, Anderson CB, Chamakuri S, Belica C, Wick C, Harki DA, Young DW, Scampavia L, Spicer TP, Shi K, Aihara H, et al. Gain-of-Signal Assays for Probing Inhibition of SARS-CoV-2 M/3CL in Living Cells. Mbio. e0078422. PMID 35471084 DOI: 10.1128/mbio.00784-22 |
0.3 |
|
2023 |
Viveki A, Mansfield T, Tran K, Lenkeit E, MacKenzie K, Young DW, Chamakuri S. Heterocyclic Merging of Stereochemically Diverse Chiral Piperazines and Morpholines with Indazoles. Chemistry (Weinheim An Der Bergstrasse, Germany). e202301888. PMID 37462979 DOI: 10.1002/chem.202301888 |
0.279 |
|
2024 |
Holmes S, Jain P, Rodriguez KG, Williams J, Yu Z, Cerda-Smith C, Samuel ELG, Campbell J, Hakenjos JM, Monsivais D, Li F, Chamakuri S, Matzuk MM, Santini C, MacKenzie KR, et al. Chemical Catalysis Guides Structural Identification for the Major Metabolite of the BET Inhibitor JQ1. Acs Medicinal Chemistry Letters. 15: 107-115. PMID 38229743 DOI: 10.1021/acsmedchemlett.3c00464 |
0.263 |
|
2021 |
Chamakuri S, Chung MK, Samuel ELG, Tran KA, Chen YC, Nyshadham P, Santini C, Matzuk MM, Young DW. Design and construction of a stereochemically diverse piperazine-based DNA-encoded chemical library. Bioorganic & Medicinal Chemistry. 48: 116387. PMID 34571488 DOI: 10.1016/j.bmc.2021.116387 |
0.259 |
|
2010 |
Kumar KS, Chamakuri S, Vishweshwar P, Iqbal J, Pal M. ChemInform Abstract: AlCl3-Induced (Hetero)arylation of Thienopyrimidine Ring: A New Synthesis of 4-Substituted Thieno[2,3-d]pyrimidines. Cheminform. 41. DOI: 10.1002/CHIN.201042159 |
0.246 |
|
2022 |
Chamakuri S, Tang SA, Tran KA, Guduru SKR, Bolin PK, MacKenzie KR, Young DW. A Concise Synthetic Method for Constructing 3-Substituted Piperazine-2-Acetic Acid Esters from 1,2-Diamines. Molecules (Basel, Switzerland). 27. PMID 35684357 DOI: 10.3390/molecules27113419 |
0.245 |
|
2020 |
Monty OBC, Simmons N, Chamakuri S, Matzuk MM, Young DW. Solution-Phase Fmoc-Based Peptide Synthesis for DNA-Encoded Chemical Libraries: Reaction Conditions, Protecting Group Strategies, and Pitfalls. Acs Combinatorial Science. PMID 33074645 DOI: 10.1021/acscombsci.0c00144 |
0.242 |
|
2020 |
Chamakuri S, Shah MM, Yang DCH, Santini C, Young DW. Practical and scalable synthesis of orthogonally protected-2-substituted chiral piperazines. Organic & Biomolecular Chemistry. PMID 33118584 DOI: 10.1039/d0ob01713b |
0.231 |
|
2023 |
Park S, Fan J, Chamakuri S, Palaniappan M, Sharma K, Qin X, Wang J, Tan Z, Judge A, Hu L, Sankaran B, Li F, Prasad BVV, Matzuk MM, Palzkill T. Exploiting the Carboxylate-Binding Pocket of β-Lactamase Enzymes Using a Focused DNA-Encoded Chemical Library. Journal of Medicinal Chemistry. PMID 38117688 DOI: 10.1021/acs.jmedchem.3c01834 |
0.211 |
|
2022 |
Young DW, Chamakuri S. Trisubstituted triumph. Nature Chemistry. 14: 595-597. PMID 35668207 DOI: 10.1038/s41557-022-00959-4 |
0.195 |
|
2022 |
Kandel P, Semerci F, Mishra R, Choi W, Bajic A, Baluya D, Ma L, Chen K, Cao AC, Phongmekhin T, Matinyan N, Jiménez-Panizo A, Chamakuri S, Raji IO, Chang L, et al. Oleic acid is an endogenous ligand of TLX/NR2E1 that triggers hippocampal neurogenesis. Proceedings of the National Academy of Sciences of the United States of America. 119: e2023784119. PMID 35333654 DOI: 10.1073/pnas.2023784119 |
0.103 |
|
2021 |
Bowling EA, Wang JH, Gong F, Wu W, Neill NJ, Kim IS, Tyagi S, Orellana M, Kurley SJ, Dominguez-Vidaña R, Chung HC, Hsu TY, Dubrulle J, Saltzman AB, Li H, ... ... Chamakuri S, et al. Spliceosome-targeted therapies trigger an antiviral immune response in triple-negative breast cancer. Cell. PMID 33450205 DOI: 10.1016/j.cell.2020.12.031 |
0.073 |
|
Hide low-probability matches. |