Mikael Bols - Publications

Affiliations: 
Chemistry University of Aarhus, Denmark 

152 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Jessen CH, Bendix J, Nannestad TB, Bordallo H, Pedersen MJ, Pedersen CM, Bols M. CO complexation with cyclodextrins. Beilstein Journal of Organic Chemistry. 19: 1021-1027. PMID 37497051 DOI: 10.3762/bjoc.19.78  0.402
2020 Bols M, Matassini C, Warren J, Wang B, Goti A, Cardona F, Morrone A. Imino- and azasugar protonation inside human acid β-glucosidase, the enzyme defective in Gaucher disease. Angewandte Chemie (International Ed. in English). PMID 32191378 DOI: 10.1002/Anie.202002850  0.309
2019 Madsen J, Viuf C, Bols M. A new method for the deprotection of benzyl ethers or the selective protection of alcohols Chemistry (Weinheim An Der Bergstrasse, Germany). 6: 1140-6. PMID 10785798 DOI: 10.1002/(Sici)1521-3765(20000403)6:7<1140::Aid-Chem1140>3.0.Co;2-6  0.318
2018 Jørgensen FP, Bols M. An inexpensive and scalable synthesis of Shld. The Journal of Organic Chemistry. PMID 29749733 DOI: 10.1021/Acs.Joc.8B00698  0.361
2017 Wang B, Olsen JI, Laursen BW, Navarro Poulsen JC, Bols M. Determination of protonation states of iminosugar-enzyme complexes using photoinduced electron transfer. Chemical Science. 8: 7383-7393. PMID 29163889 DOI: 10.1039/C7Sc01540B  0.355
2017 Bols M, Pedersen CM. Silyl-protective groups influencing the reactivity and selectivity in glycosylations. Beilstein Journal of Organic Chemistry. 13: 93-105. PMID 28228850 DOI: 10.3762/Bjoc.13.12  0.499
2017 Pedersen CM, Bols M. On the nature of the electronic effect of multiple hydroxyl groups in the 6-membered ring - the effects are additive but steric hindrance plays a role too. Organic & Biomolecular Chemistry. PMID 28084490 DOI: 10.1039/C6Ob02427K  0.51
2017 Nielsen MM, Stougaard BA, Bols M, Glibstrup E, Pedersen CM. Glycosyl Fluorides as Intermediates in BF3·OEt2-Promoted Glycosylation with Trichloroacetimidates European Journal of Organic Chemistry. 2017: 1281-1284. DOI: 10.1002/Ejoc.201601439  0.502
2016 Bandara MD, Yasomanee JP, Rath NP, Pedersen CM, Bols M, Demchenko AV. Conformationally superarmed S-ethyl glycosyl donors as effective building blocks for chemoselective oligosaccharide synthesis in one pot. Organic & Biomolecular Chemistry. PMID 27942674 DOI: 10.1039/C6Ob02498J  0.556
2016 Olsen JI, Plata GB, Padrón JM, López Ó, Bols M, Fernández-Bolaños JG. Selenoureido-iminosugars: A new family of multitarget drugs. European Journal of Medicinal Chemistry. 123: 155-160. PMID 27474931 DOI: 10.1016/J.Ejmech.2016.07.021  0.312
2016 Olsen JI, Kowalska K, Pedersen CM, Bols M. Super arming of a glycosyl donor using a molecular lever Tetrahedron Letters. 57: 35-38. DOI: 10.1016/J.Tetlet.2015.11.052  0.5
2016 Frihed TG, Bols M, Pedersen CM. C-H Functionalization on Carbohydrates European Journal of Organic Chemistry. 2016: 2740-2756. DOI: 10.1002/Ejoc.201600121  0.466
2016 Frihed TG, Bols M, Pedersen CM. ChemInform Abstract: C-H Functionalization on Carbohydrates Cheminform. 47. DOI: 10.1002/CHIN.201635168  0.37
2015 Heuckendorff M, Bols PS, Barry CB, Frihed TG, Pedersen CM, Bols M. β-Mannosylation with 4,6-benzylidene protected mannosyl donors without preactivation. Chemical Communications (Cambridge, England). 51: 13283-5. PMID 26197760 DOI: 10.1039/C5Cc04716A  0.517
2015 Lindbäck E, Laursen BW, Poulsen JC, Kilså K, Pedersen CM, Bols M. A fluorescence study of isofagomine protonation in β-glucosidase. Organic & Biomolecular Chemistry. 13: 6562-6. PMID 25978843 DOI: 10.1039/C5Ob00624D  0.515
2015 Frihed TG, Bols M, Pedersen CM. Mechanisms of Glycosylation Reactions Studied by Low-Temperature Nuclear Magnetic Resonance. Chemical Reviews. 115: 4963-5013. PMID 25923428 DOI: 10.1021/Cr500434X  0.442
2015 Frihed TG, Bols M, Pedersen CM. Synthesis of L-Hexoses. Chemical Reviews. 115: 3615-76. PMID 25893557 DOI: 10.1021/Acs.Chemrev.5B00104  0.474
2015 Heuckendorff M, Bols PS, Barry CB, Frihed TG, Pedersen CM, Bols M. β-Mannosylation with 4,6-benzylidene protected mannosyl donors without preactivation Chemical Communications. 51: 13283-13285. DOI: 10.1039/c5cc04716a  0.432
2015 Frihed TG, Bols M, Pedersen CM. ChemInform Abstract: Mechanisms of Glycosylation Reactions Studied by Low-Temperature Nuclear Magnetic Resonance Cheminform. 46: no-no. DOI: 10.1002/CHIN.201533305  0.379
2015 Frihed TG, Bols M, Pedersen CM. ChemInform Abstract: Synthesis of L-Hexoses Cheminform. 46: no-no. DOI: 10.1002/CHIN.201532248  0.418
2014 Frihed TG, Pedersen CM, Bols M. Synthesis of all eight L-glycopyranosyl donors using C-H activation. Angewandte Chemie (International Ed. in English). 53: 13889-93. PMID 25303081 DOI: 10.1002/Ange.201408209  0.518
2014 Hogendorf WF, Gisch N, Schwudke D, Heine H, Bols M, Pedersen CM. Total Synthesis of Five Lipoteichoic acids of Clostridium difficile. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 13511-6. PMID 25168290 DOI: 10.1002/Chem.201404336  0.483
2014 Heuckendorff M, Bendix J, Pedersen CM, Bols M. β-Selective mannosylation with a 4,6-silylene-tethered thiomannosyl donor. Organic Letters. 16: 1116-9. PMID 24502365 DOI: 10.1021/Ol403722F  0.526
2014 Zhou Y, Lindbäck E, Pedersen CM, Bols M. Cyclodextrin-based artificial oxidases with high rate accelerations and selectivity Tetrahedron Letters. 55: 2304-2307. DOI: 10.1016/J.Tetlet.2014.02.100  0.507
2014 Frihed TG, Pedersen CM, Bols M. Synthesis of All Eight Stereoisomeric 6-Deoxy-L-hexopyranosyl Donors - Trends in Using Stereoselective Reductions or Mitsunobu Epimerizations European Journal of Organic Chemistry. 2014: 7924-7939. DOI: 10.1002/Ejoc.201403074  0.494
2014 Frihed TG, Pedersen CM, Bols M. Synthesis of All EightL-Glycopyranosyl Donors Using CH Activation Angewandte Chemie. 126: 14109-14113. DOI: 10.1002/ANGE.201408209  0.443
2013 Hogendorf WF, Jagalski V, Pomorski TG, Bols M, Cárdenas M, Pedersen CM. Synthesis and thermotropic phase behavior of four glycoglycerolipids. Molecules (Basel, Switzerland). 18: 13546-73. PMID 24189295 DOI: 10.3390/Molecules181113546  0.482
2013 Heuckendorff M, Premathilake HD, Pornsuriyasak P, Madsen AØ, Pedersen CM, Bols M, Demchenko AV. Superarming of glycosyl donors by combined neighboring and conformational effects. Organic Letters. 15: 4904-7. PMID 24006853 DOI: 10.1021/Ol402371B  0.494
2013 Heuckendorff M, Pedersen CM, Bols M. Conformationally armed 3,6-tethered glycosyl donors: synthesis, conformation, reactivity, and selectivity. The Journal of Organic Chemistry. 78: 7234-48. PMID 23786671 DOI: 10.1021/Jo4012464  0.548
2013 López Ó, Qing FL, Pedersen CM, Bols M. Enzyme inhibition by iminosugars: analysis and insight into the glycosidase-iminosugar dependency of pH. Bioorganic & Medicinal Chemistry. 21: 4755-61. PMID 23583693 DOI: 10.1016/J.Bmc.2013.03.003  0.484
2013 Frihed TG, Walvoort MT, Codée JD, van der Marel GA, Bols M, Pedersen CM. Influence of O6 in mannosylations using benzylidene protected donors: stereoelectronic or conformational effects? The Journal of Organic Chemistry. 78: 2191-205. PMID 23336427 DOI: 10.1021/Jo302455D  0.541
2013 Zhou Y, Pedersen CM, Bols M. Artificial enzyme activity from cyclodextrins with cyanohydrins on the secondary rim Tetrahedron Letters. 54: 2458-2461. DOI: 10.1016/J.Tetlet.2013.02.091  0.554
2013 Pedersen CM, Bols M, Qiao Y. ChemInform Abstract: Total Synthesis of Biologically Active Lipoteichoic Acids Cheminform. 44: no-no. DOI: 10.1002/chin.201316228  0.435
2012 Frihed TG, Heuckendorff M, Pedersen CM, Bols M. Easy access to L-mannosides and L-galactosides by using C-H activation of the corresponding 6-deoxysugars. Angewandte Chemie (International Ed. in English). 51: 12285-8. PMID 23109259 DOI: 10.1002/Anie.201206880  0.45
2012 Heuckendorff M, Pedersen CM, Bols M. Rhamnosylation: diastereoselectivity of conformationally armed donors. The Journal of Organic Chemistry. 77: 5559-68. PMID 22639871 DOI: 10.1021/Jo300591K  0.531
2012 Pedersen CM, Bols M, Qiao Y. Total synthesis of biologically active lipoteichoic acids Arkivoc. 2013. DOI: 10.3998/Ark.5550190.0014.220  0.504
2012 Lindbäck E, Zhou Y, Pedersen CM, Bols M. Artificial enzymes based on cyclodextrin with phenol as the catalytic group Tetrahedron Letters. 53: 5023-5026. DOI: 10.1016/J.Tetlet.2012.07.050  0.499
2012 Lindbäck E, Zhou Y, López Ó, Fernández-Bolaños JG, Pedersen CM, Bols M. A uronic acid analogue of isofagomine lactam as a nanomolar glucuronidase inhibitor Tetrahedron Letters. 53: 2045-2047. DOI: 10.1016/J.Tetlet.2012.02.009  0.52
2012 Jadhav H, Taarning E, Pedersen CM, Bols M. Conversion of d-glucose into 5-hydroxymethylfurfural (HMF) using zeolite in [Bmim]Cl or tetrabutylammonium chloride (TBAC)/CrCl2 Tetrahedron Letters. 53: 983-985. DOI: 10.1016/J.Tetlet.2011.12.059  0.49
2012 Zhou Y, Marinescu L, Pedersen CM, Bols M. Synthesis of Tin-Containing Cyclodextrins as Potential Enzyme Models European Journal of Organic Chemistry. 2012: 6383-6389. DOI: 10.1002/Ejoc.201200756  0.543
2012 Lindbäck E, Zhou Y, Pedersen CM, Bols M. Two Diastereomeric Artificial Enzymes with Different Catalytic Activity European Journal of Organic Chemistry. 2012: 5366-5372. DOI: 10.1002/Ejoc.201200699  0.55
2012 Zhou Y, Lindbäck E, Marinescu LG, Pedersen CM, Bols M. Synthesis of Cyclodextrins with Carboxylic Acids at the Secondary Rim and an Evaluation of Their Properties as Chemzymes for Glycoside Hydrolysis European Journal of Organic Chemistry. 2012: 4063-4070. DOI: 10.1002/Ejoc.201200404  0.532
2011 Heuckendorff M, Pedersen CM, Bols M. The influence of neighboring group participation on the hydrolysis of 2-O-substituted methyl glucopyranosides. Organic Letters. 13: 5956-9. PMID 22007683 DOI: 10.1021/Ol202308Y  0.504
2011 Jadhav V, Pedersen CM, Bols M. A study of anhydrocelluloses--is a cellulose structure with residues in a 1C4-conformation more prone to hydrolysis? Organic & Biomolecular Chemistry. 9: 7525-34. PMID 21931923 DOI: 10.1039/C1Ob06085F  0.531
2011 Jadhav H, Pedersen CM, Sølling T, Bols M. 3-Deoxy-glucosone is an intermediate in the formation of furfurals from D-glucose. Chemsuschem. 4: 1049-51. PMID 21717583 DOI: 10.1002/Cssc.201100249  0.464
2011 Amorim L, Marcelo F, Rousseau C, Nieto L, Jiménez-Barbero J, Marrot J, Rauter AP, Sollogoub M, Bols M, Blériot Y. Direct experimental evidence for the high chemical reactivity of α- and β-xylopyranosides adopting a (2,5)B conformation in glycosyl transfer. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 7345-56. PMID 21567492 DOI: 10.1002/Chem.201003251  0.33
2011 Lindbäck E, López O, Fernández-Bolaños JG, Sauer SP, Bols M. An isofagomine analogue with an amidine at the pseudoanomeric position. Organic Letters. 13: 2908-11. PMID 21548609 DOI: 10.1021/Ol200942G  0.358
2011 Pedersen CM, Olsen J, Brka AB, Bols M. Quantifying the electronic effects of carbohydrate hydroxy groups by using aminosugar models. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 7080-6. PMID 21542038 DOI: 10.1002/Chem.201100020  0.547
2011 Yang Y, Zheng F, Bols M, Marinescu LG, Qing FL. Synthesis of monofluorinated isofagomine analogues and evaluation as glycosidase inhibitors Journal of Fluorine Chemistry. 132: 838-845. DOI: 10.1016/J.Jfluchem.2011.05.031  0.337
2011 Pedersen CM, Marinescu LG, Bols M. Glycosyl donors in “unusual” conformations – influence on reactivity and selectivity Comptes Rendus Chimie. 14: 17-43. DOI: 10.1016/J.Crci.2010.03.030  0.519
2011 Christensen HS, Sigurskjold BW, Frihed TG, Marinescu LG, Pedersen CM, Bols M. Recognition of Peptides by Cyclodextrin Trimers European Journal of Organic Chemistry. 2011: 5279-5290. DOI: 10.1002/Ejoc.201100671  0.456
2011 Fenger TH, Marinescu LG, Bols M. Cyclodextrin Ketones with the Catalytic Group at the Secondary Rim and Their Effectiveness in Enzyme-Like Epoxidation of Stilbenes European Journal of Organic Chemistry. 2011: 2339-2345. DOI: 10.1002/Ejoc.201001696  0.372
2011 Kumari N, Olesen JK, Pedersen CM, Bols M. Synthesis of 5-Bromomethylfurfural from Cellulose as a Potential Intermediate for Biofuel European Journal of Organic Chemistry. 2011: 1266-1270. DOI: 10.1002/Ejoc.201001539  0.507
2011 Pedersen CM, Marinescu LG, Bols M. ChemInform Abstract: Glycosyl Donors in “Unusual” Conformations - Influence on Reactivity and Selectivity Cheminform. 42: no-no. DOI: 10.1002/CHIN.201134241  0.43
2010 Heuckendorff M, Pedersen CM, Bols M. Quantifying electronic effects of common carbohydrate protecting groups in a piperidine model system. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 13982-94. PMID 21132699 DOI: 10.1002/Chem.201002313  0.523
2010 Fenger TH, Bols M. Substrate control through per-O-methylation of cyclodextrin acids. Chemical Communications (Cambridge, England). 46: 7769-71. PMID 20871875 DOI: 10.1039/C0Cc02071K  0.312
2010 Petrillo M, Marinescu L, Bols M. Regioselective difunctionalization of cyclodextrins Journal of Inclusion Phenomena and Macrocyclic Chemistry. 69: 425-431. DOI: 10.1007/S10847-010-9775-7  0.377
2010 Fenger TH, Bols M. Simple cyclodextrin aldehydes as excellent artificial oxidases Journal of Inclusion Phenomena and Macrocyclic Chemistry. 69: 397-402. DOI: 10.1007/S10847-010-9771-Y  0.304
2010 Bjerre J, Bols M. Substantial Spatial Flexibility and Hydrogen Bonding within the Catalysis Exerted by Cyclodextrin Artificial Glycosidases European Journal of Organic Chemistry. 2010: 3487-3500. DOI: 10.1002/Ejoc.201000380  0.329
2010 Lindbäck E, Zhou Y, Marinescu L, Pedersen CM, Bols M. The Grignard Reaction of Cyclodextrin-6-aldehydes Revisited: A Study of the Stereoselectivity Upon Addition of Organometallic Reagents to Aldehydes and Ketones European Journal of Organic Chemistry. 2010: 3883-3896. DOI: 10.1002/Ejoc.201000295  0.515
2009 Wang RW, Xu J, Lopez O, Bols M, Qing FL. Difluoromethylenated polyhydroxylated pyrrolidines: facile synthesis, crystal structure and biological evaluation. Future Medicinal Chemistry. 1: 991-7. PMID 21426093 DOI: 10.4155/Fmc.09.82  0.304
2009 Nielsen S, Pedersen CM, Hansen SG, Petersen MD, Sinning S, Wiborg O, Jensen HH, Bols M. An extended study of dimeric phenyl tropanes. Bioorganic & Medicinal Chemistry. 17: 4900-9. PMID 19560930 DOI: 10.1016/J.Bmc.2009.06.007  0.516
2009 Fenger TH, Marinescu LG, Bols M. Cyclodextrin ketones as oxidation catalysts: investigation of bridged derivatives. Organic & Biomolecular Chemistry. 7: 933-43. PMID 19225677 DOI: 10.1039/B814245A  0.321
2009 Li R, Bols M, Rousseau C, Zhang X, Wang R, Qing F. Synthesis and biological evaluation of potent glycosidase inhibitors: 4-deoxy-4,4-difluoroisofagomine and analogues Tetrahedron. 65: 3717-3727. DOI: 10.1016/J.Tet.2009.02.079  0.326
2009 Marinescu LG, Doyagüez EG, Petrillo M, Fernández-Mayoralas A, Bols M. Amino-Acetone-Bridged Cyclodextrins ― Artificial Alcohol Oxidases European Journal of Organic Chemistry. 2010: 157-167. DOI: 10.1002/Ejoc.200901099  0.362
2008 Pedersen CM, Marinescu LG, Bols M. Conformationally armed glycosyl donors: reactivity quantification, new donors and one pot reactions. Chemical Communications (Cambridge, England). 2465-7. PMID 18491016 DOI: 10.1039/B801305E  0.498
2008 López Ó, Bols M. Effective synthesis of negatively charged cyclodextrins. Selective access to phosphate cyclodextrins Tetrahedron. 64: 7587-7593. DOI: 10.1016/J.Tet.2008.05.094  0.376
2008 Bjerre J, Nielsen EH, Bols M. Hydrolysis of Toxic Natural Glucosides Catalyzed by Cyclodextrin Dicyanohydrins European Journal of Organic Chemistry. 2008: 745-752. DOI: 10.1002/Ejoc.200700954  0.373
2007 Boye SV, Ortega-Caballero F, Sinning S, Wiborg O, Jensen HH, Bols M. High dopamine transporter selectivity can be displayed by remarkably simple non-nitrogen containing inhibitors. Bioorganic & Medicinal Chemistry Letters. 17: 6019-25. PMID 17869101 DOI: 10.1016/J.Bmcl.2007.07.076  0.302
2007 Jensen HH, Pedersen CM, Bols M. Going to extremes: "super" armed glycosyl donors in glycosylation chemistry. Chemistry (Weinheim An Der Bergstrasse, Germany). 13: 7576-82. PMID 17705330 DOI: 10.1002/Chem.200700947  0.504
2007 Pedersen CM, Nordstrøm LU, Bols M. "Super armed" glycosyl donors: conformational arming of thioglycosides by silylation. Journal of the American Chemical Society. 129: 9222-35. PMID 17602482 DOI: 10.1021/Ja071955L  0.53
2007 Petersen MD, Boye SV, Nielsen EH, Willumsen J, Sinning S, Wiborg O, Bols M. Synthesis, inhibition and binding of simple non-nitrogen inhibitors of monoamine transporters. Bioorganic & Medicinal Chemistry. 15: 4159-74. PMID 17446076 DOI: 10.1016/J.Bmc.2007.03.069  0.314
2007 Lopez OL, Bols M. Anomer-selective glycosidase inhibition by 2-N-alkylated 1-azafagomines Chembiochem. 8: 657-661. PMID 17352429 DOI: 10.1002/Cbic.200700012  0.36
2007 Lopez OL, Marinescu L, Bols M. New cup-shaped α-cyclodextrin derivatives and a study of their catalytic properties in oxidation reactions Tetrahedron. 63: 8872-8880. DOI: 10.1016/J.Tet.2007.06.018  0.332
2007 Sivertsen AC, Gasior M, Bjerring M, Hansen SU, Lopez OL, Nielsen NC, Bols M. Active site protonation of 1-azafagomine in glucosidases studied by solid-state NMR spectroscopy European Journal of Organic Chemistry. 1735-1742. DOI: 10.1002/Ejoc.200600816  0.326
2007 Bjerre J, Hauch Fenger T, Marinescu LG, Bols M. Synthesis of Some Trifluoromethylated Cyclodextrin Derivatives and Analysis of Their Properties as Artificial Glycosidases and Oxidases European Journal of Organic Chemistry. 2007: 704-710. DOI: 10.1002/Ejoc.200600762  0.367
2007 Jensen HH, Pedersen CM, Bols M. Going to Extremes: “Super” Armed Glycosyl Donors in Glycosylation Chemistry Cheminform. 38. DOI: 10.1002/CHIN.200750238  0.412
2007 Pedersen CM, Nordstroem LU, Bols M. “Super Armed” Glycosyl Donors: Conformational Arming of Thioglycosides by Silylation. Cheminform. 38. DOI: 10.1002/CHIN.200750201  0.413
2006 Wang RW, Qiu XL, Bols M, Ortega-Caballero F, Qing FL. Synthesis and biological evaluation of glycosidase inhibitors: gem-difluoromethylenated nojirimycin analogues. Journal of Medicinal Chemistry. 49: 2989-97. PMID 16686540 DOI: 10.1021/Jm060066Q  0.312
2006 Jensen HH, Bols M. Stereoelectronic substituent effects. Accounts of Chemical Research. 39: 259-65. PMID 16618093 DOI: 10.1021/Ar050189P  0.305
2006 Ortega-Caballero F, Bols M. Cyclodextrin derivatives with cyanohydrin and carboxylate groups as artificial glycosidases Canadian Journal of Chemistry. 84: 650-658. DOI: 10.1139/V06-039  0.364
2006 Kuntz DA, Liu H, Bols M, Rose DR. The role of the active site Zn in the catalytic mechanism of the GH38 Golgi α-mannosidase II: Implications from noeuromycin inhibition Biocatalysis and Biotransformation. 24: 55-61. DOI: 10.1080/10242420500533242  0.315
2006 Tagmose TM, Bols M. Synthesis of the 2-Deoxyisomaltose Analogue of Acarbose by an Improved Route to Chiral Valieneamines Chemistry - a European Journal. 3: 453-462. DOI: 10.1002/Chem.19970030318  0.353
2005 Ortega-Caballero F, Bjerre J, Laustsen LS, Bols M. Four orders of magnitude rate increase in artificial enzyme-catalyzed aryl glycoside hydrolysis. The Journal of Organic Chemistry. 70: 7217-26. PMID 16122240 DOI: 10.1021/Jo050861W  0.35
2005 Rousseau C, Ortega-Caballero F, Nordstrøm LU, Christensen B, Petersen TE, Bols M. Artificial glycosyl phosphorylases. Chemistry (Weinheim An Der Bergstrasse, Germany). 11: 5094-101. PMID 15981287 DOI: 10.1002/Chem.200500364  0.306
2005 Gregersen A, Pedersen CM, Jensen HH, Bols M. On the electronic effects of OH groups. Synthesis and investigation of tetrahydroxylated azabicycloheptanes. Organic & Biomolecular Chemistry. 3: 1514-9. PMID 15827650 DOI: 10.1039/B419154D  0.548
2005 Pedersen CM, Marinescu LG, Bols M. Radical substitution with azide: TMSN3-PhI(OAc)2 as a substitute of IN3. Organic & Biomolecular Chemistry. 3: 816-22. PMID 15731868 DOI: 10.1039/B500037H  0.518
2005 Marinescu LG, Pedersen CM, Bols M. Safe Radical Azidonation Using Polystyrene Supported Diazidoiodate(I). Cheminform. 36. DOI: 10.1016/J.Tet.2004.10.040  0.489
2005 Marinescu LG, Pedersen CM, Bols M. Safe radical azidonation using polystyrene supported diazidoiodate(I) Tetrahedron. 61: 123-127. DOI: 10.1016/J.TET.2004.10.040  0.357
2005 Pedersen CM, Bols M. Stereochemical substituent effects: investigation of the cyano, amide and carboxylate group Tetrahedron. 61: 115-122. DOI: 10.1016/J.Tet.2004.10.039  0.471
2005 Rousseau C, Christensen B, Bols M. Artificial Epoxidase II. Synthesis of Cyclodextrin Ketoesters and Epoxidation of Alkenes European Journal of Organic Chemistry. 2005: 2734-2739. DOI: 10.1002/Ejoc.200500034  0.319
2005 Pedersen CM, Marinescu LG, Bols M. Radical Substitution with Azide: TMSN3—PhI(OAc)2 as a Substitute of IN3. Cheminform. 36. DOI: 10.1002/CHIN.200532062  0.437
2004 Rousseau C, Christensen B, Petersen TE, Bols M. Cyclodextrins containing an acetone bridge. Synthesis and study as epoxidation catalysts. Organic & Biomolecular Chemistry. 2: 3476-82. PMID 15565240 DOI: 10.1039/B410098K  0.357
2004 Pedersen H, Sinning S, Bulow A, Wiborg O, Falborg L, Bols M. Combinatorial synthesis of benztropine libraries and their evaluation as monoamine transporter inhibitors. Organic & Biomolecular Chemistry. 2: 2861-9. PMID 15455161 DOI: 10.1039/B405768F  0.364
2004 McDonnell C, López O, Murphy P, Fernández Bolaños JG, Hazell R, Bols M. Conformational effects on glycoside reactivity: study of the high reactive conformer of glucose. Journal of the American Chemical Society. 126: 12374-85. PMID 15453771 DOI: 10.1021/Ja047476T  0.3
2004 Jensen HH, Nordstrøm LU, Bols M. The disarming effect of the 4,6-acetal group on glycoside reactivity: torsional or electronic? Journal of the American Chemical Society. 126: 9205-13. PMID 15281809 DOI: 10.1021/Ja047578J  0.343
2004 Bülow A, Sinning S, Wiborg O, Bols M. Two- and three dimensional combinatorial chemistry from multicomponent Grignard reagents. Journal of Combinatorial Chemistry. 6: 509-19. PMID 15244412 DOI: 10.1021/Cc049947D  0.328
2004 Andersch J, Bols M, Hazell A. Benzyl 4-C-nitrosomethyl-β-D-arabinopyranoside Acta Crystallographica Section E Structure Reports Online. 60: o660-o661. DOI: 10.1107/S1600536804006488  0.308
2004 Rousseau C, Nielsen N, Bols M. An artificial enzyme that catalyzes hydrolysis of aryl glycosides Tetrahedron Letters. 45: 8709-8711. DOI: 10.1016/J.Tetlet.2004.09.134  0.315
2004 Bülow A, Meyer T, Olszewski T, Bols M. The C-4 Configuration as a Probe for the Study of Glycosidation Reactions European Journal of Organic Chemistry. 2004: 323-329. DOI: 10.1002/Ejoc.200300540  0.33
2003 Marinescu L, Thinggaard J, Thomsen IB, Bols M. Radical azidonation of aldehydes. The Journal of Organic Chemistry. 68: 9453-5. PMID 14629171 DOI: 10.1021/Jo035163V  0.326
2003 Lillelund VH, Liu H, Liang X, Søhoel H, Bols M. Isofagomine lactams, synthesis and enzyme inhibition. Organic & Biomolecular Chemistry. 1: 282-7. PMID 12929423 DOI: 10.1039/B208784G  0.311
2003 Lopez OL, Fernández-Bolaños JG, Lillelund VH, Bols M. Aziridines as a structural motif to conformational restriction of azasugars Organic and Biomolecular Chemistry. 1: 478-482. PMID 12926248 DOI: 10.1039/B210038J  0.335
2003 Ulgar V, López Ó, Maya I, Fernández-Bolaños JG, Bols M. Synthesis of furan 4′-thio-C-nucleosides, their methylsulfonium and sulfoxide derivatives. Evaluation as glycosidase inhibitors Tetrahedron. 59: 2801-2809. DOI: 10.1016/S0040-4020(03)00339-9  0.39
2002 Bols M, Liang X, Jensen HH. Equatorial contra axial polar substituents. The relation of a chemical reaction to stereochemical substituent constants. The Journal of Organic Chemistry. 67: 8970-4. PMID 12467416 DOI: 10.1021/Jo0205356  0.314
2002 Jensen HH, Lyngbye L, Jensen A, Bols M. Stereoelectronic substituent effects in polyhydroxylated piperidines and hexahydropyridazines. Chemistry (Weinheim An Der Bergstrasse, Germany). 8: 1218-26. PMID 11891910 DOI: 10.1002/1521-3765(20020301)8:5<1218::Aid-Chem1218>3.0.Co;2-X  0.334
2002 Andersch J, Bols M. Efficient synthesis of isofagomine and noeuromycin. Chemistry (Weinheim An Der Bergstrasse, Germany). 7: 3744-7. PMID 11575775 DOI: 10.1002/1521-3765(20010903)7:17<3744::Aid-Chem3744>3.0.Co;2-3  0.356
2002 Hardlei T, Bols M. Unusual hydrogen-bonding differences in stereoisomeric 6-C-alkylated cyclodextrins Journal of the Chemical Society-Perkin Transactions 1. 2880-2885. DOI: 10.1039/B207033M  0.355
2002 Ulgar V, Fernández-Bolaños JG, Bols M. Synthesis and evaluation of sulfonium analogues of isofucofagomine as glycosidase inhibitors Journal of the Chemical Society-Perkin Transactions 1. 1242-1246. DOI: 10.1039/B202021C  0.333
2002 Jensen HH, Jensen A, Hazell RG, Bols M. Synthesis and investigation of L-fuco- and D-glucurono-azafagomine Journal of the Chemical Society-Perkin Transactions 1. 1190-1198. DOI: 10.1039/B200884J  0.36
2002 Muldgaard L, Thomsen IB, Hazell RG, Bols M. Investigation of the base promoted tandem syn-elimination–Favorskii rearrangement of levoglucosan sulfonates Journal of the Chemical Society-Perkin Transactions 1. 1297-1301. DOI: 10.1039/B200064B  0.37
2002 Baruah M, Bols M. Substitution of α-azido ethers with Grignard reagents and its use in combinatorial chemistry Journal of the Chemical Society-Perkin Transactions 1. 509-512. DOI: 10.1039/B110428B  0.319
2002 Liang X, Bols M. Solution-phase combinatorial synthesis using multicomponent Grignard reagents Journal of the Chemical Society-Perkin Transactions 1. 503-508. DOI: 10.1039/B109952N  0.338
2001 Viuf C, Bols M. Radical Azidonation of Benzylic Positions with Iodonium Azide. Angewandte Chemie (International Ed. in English). 40: 623-625. PMID 29712008 DOI: 10.1002/1521-3773(20010202)40:3<623::Aid-Anie623>3.0.Co;2-G  0.306
2001 Søndergaard K, Liang X, Bols M. Synthesis of 5-azacastanospermine, a conformationally restricted azafagomine analogue. Chemistry (Weinheim An Der Bergstrasse, Germany). 7: 2324-31. PMID 11446635 DOI: 10.1002/1521-3765(20010601)7:11<2324::Aid-Chem23240>3.0.Co;2-Y  0.349
2001 Andreassen V, Svensson B, Bols M. Synthesis of an 1′-Azasugar Analogue of Maltose Synthesis. 2001: 0339-0342. DOI: 10.1055/S-2001-10799  0.345
2001 Søhoel H, Liang X, Bols M. Isogalactofagomine lactam. A neutral nanomolar galactosidase inhibitor Journal of the Chemical Society-Perkin Transactions 1. 1584-1585. DOI: 10.1039/B103831C  0.312
2001 Liang X, Petersen BO, Duus JØ, Bols M. A bioisosteric oligosaccharide mimetic based on isofagomine-type monomers Journal of the Chemical Society-Perkin Transactions 1. 2764-2773. DOI: 10.1039/B103756K  0.313
2001 Jensen HH, Bols M. Synthesis of 1-azagalactofagomine, a potent galactosidase inhibitor Journal of the Chemical Society-Perkin Transactions 1. 905-909. DOI: 10.1039/B007973L  0.317
2000 Ernholt BV, Thomsen Ib B, Lohse A, Plesner IW, Jensen KB, Hazell RG, Liang X, Jakobsen A, Bols M. Enantiospecific synthesis of 1-azafagomine. Chemistry (Weinheim An Der Bergstrasse, Germany). 6: 278-87. PMID 11931107 DOI: 10.1002/(Sici)1521-3765(20000117)6:2<278::Aid-Chem278>3.0.Co;2-6  0.383
2000 Liang X, Lohse A, Bols M. Chemoenzymatic synthesis of isogalactofagomine. The Journal of Organic Chemistry. 65: 7432-7. PMID 11076600 DOI: 10.1021/Jo000699R  0.377
2000 Jensen HH, Lohse A, Petersen BO, Duus JØ, Bols M. Synthesis of 3-C-hydroxymethyl- and 3-deoxyisofagomine and investigation of their binding to β-glucosidase Journal of the Chemical Society-Perkin Transactions 1. 667-670. DOI: 10.1039/A909869K  0.318
2000 Lohse A, Jensen HH, Bach P, Bols M. Synthesis of 3-substituted isofagomine analogues using an unusual syn hydrogenation reaction Journal of the Chemical Society, Perkin Transactions 1. 659-665. DOI: 10.1039/A908340E  0.37
1999 Lohse A, Jensen KB, Lundgren K, Bols M. Synthesis and deconvolution of the first combinatorial library of glycosidase inhibitors. Bioorganic & Medicinal Chemistry. 7: 1965-71. PMID 10530945 DOI: 10.1016/S0968-0896(99)00116-9  0.314
1999 Hansen SU, Bols M. Synthesis of labelled 1-azafagomine Journal of the Chemical Society-Perkin Transactions 1. 3323-3325. DOI: 10.1039/A907365E  0.315
1999 Liang X, Bols M. Chemoenzymatic Synthesis of Enantiopure 1-Azafagomine The Journal of Organic Chemistry. 64: 8485-8488. DOI: 10.1021/Jo9907989  0.366
1999 Bach P, Bols M. Synthesis of an 1-azaglucose analogue with ring-oxygen retained Tetrahedron Letters. 40: 3461-3464. DOI: 10.1016/S0040-4039(99)00423-2  0.31
1999 Bach P, Lohse A, Bols M. Short synthesis of piperidine based hexopyranose minics. A remarkable example of syn hydrogenation Tetrahedron Letters. 40: 367-370. DOI: 10.1016/S0040-4039(98)02313-2  0.351
1998 Madsen J, Bols M. A New Intramolecular Reaction for the Regioselective Debenzylation or Protection of Alcohols. Angewandte Chemie (International Ed. in English). 37: 3177-3178. PMID 29711310 DOI: 10.1002/(Sici)1521-3773(19981204)37:22<3177::Aid-Anie3177>3.0.Co;2-A  0.346
1998 Bols M. New branched carbohydrate building block from a tandem elimination-Farvorski rearrangement Chemical Communications. 1869-1870. DOI: 10.1039/A803397H  0.324
1997 Byrgesen E, Nielsen J, Willert M, Bols M. Combinatorial chemistry of piperidine based carbohydrate mimics Tetrahedron Letters. 38: 5697-5700. DOI: 10.1016/S0040-4039(97)01249-5  0.317
1997 Thomsen I, Ernholt BV, Bols M. Synthetic studies of fluorinated analogues of 1-azafagomine: Remarkable nucleophilic substitution of fluorine by hydrazine Tetrahedron. 53: 9357-9364. DOI: 10.1016/S0040-4020(97)00588-7  0.349
1997 Lohse A, Bols M. Synthesis of 6-deoxy-6-phenylisofagomine derivatives Tetrahedron. 53: 6917-6924. DOI: 10.1016/S0040-4020(97)00392-X  0.333
1997 Bols M, Hazell RG, Thomsen IB. 1-Azafagomine: A Hydroxyhexahydropyridazine That Potently Inhibits Enzymatic Glycoside Cleavage Chemistry - a European Journal. 3: 940-947. DOI: 10.1002/Chem.19970030616  0.405
1996 Dong W, Jespersen T, Bols M, Skrydstrup T, Sierks MR. Evaluation of isofagomine and its derivatives as potent glycosidase inhibitors Biochemistry. 35: 2788-2795. PMID 8611585 DOI: 10.1021/Bi9522514  0.363
1996 Hansen A, Tagmose TM, Bols M. Synthesis of a new potent α-fucosidase inhibitor Chemical Communications. 2649-2650. DOI: 10.1039/Cc9960002649  0.324
1996 Skrydstrup T, Jespersen T, Beau J, Bols M. A new and convenient benzyloxyalkylating agent induced by samarium diiodide Chemical Communications. 515-516. DOI: 10.1039/Cc9960000515  0.319
1996 Hansen HC, Hindsgaul O, Bols M. Synthesis of tributyltinmethylated sugars, building blocks for tethered reactions Tetrahedron Letters. 37: 4211-4212. DOI: 10.1016/0040-4039(96)00798-8  0.351
1996 Bols M, Persson MP, Butt WM, Jørgensen M, Christensen P, Hansen LT. Synthesis of a ribofuranosyl cation mimic Tetrahedron Letters. 37: 2097-2100. DOI: 10.1016/0040-4039(96)00202-X  0.353
1995 Thomas SS, Plenkiewicz J, Ison ER, Bols M, Zou W, Szarek WA, Kisilevsky R. Influence of monosaccharide derivatives on liver cell glycosaminoglycan synthesis: 3-deoxy-D-xylo-hexose (3-deoxy-D-galactose) and methyl (methyl 4-chloro-4-deoxy-beta-D-galactopyranosid) uronate. Biochimica Et Biophysica Acta. 1272: 37-48. PMID 7662718 DOI: 10.1016/0925-4439(95)00065-C  0.35
1995 Mikkelsen G, Christensen TV, Bols M, Lundt I, Sierks MR. Aglycon mimicking: Glycoside bond cleavage transition state mimics based on hydroxypyrrolidine inhibitors Tetrahedron Letters. 36: 6541-6544. DOI: 10.1016/0040-4039(95)01281-L  0.309
1995 Barbaud C, Bols M, Lundt I, Sierks MR. Synthesis of the first pseudosugar-C-disaccharide. A potential antigen for eliciting glycoside-bond forming antibodies with catalytic groups Tetrahedron. 51: 9063-9078. DOI: 10.1016/0040-4020(95)00505-3  0.361
1994 Bols M, Hansen HC. Long Range Intramolecular Glycosidation Chemistry Letters. 23: 1049-1052. DOI: 10.1246/Cl.1994.1049  0.346
1994 M. Jespersen T, Bols M, R. Sierks M, Skrydstrup T. Synthesis of isofagomine, a novel glycosidase inhibitor Tetrahedron. 50: 13449-13460. DOI: 10.1016/S0040-4020(01)89351-0  0.411
1993 Bols M. Application of intramolecular glycosidation to the stereocontrolled synthesis of disaccharides containing α-gluco and α-galacto linkages Journal of the Chemical Society, Chemical Communications. 791-792. DOI: 10.1039/C39930000791  0.332
1993 Bols M. Efficient stereocontrolled glycosidation of secondary sugar hydroxyls by silicon tethered intramolecular glycosidation Tetrahedron. 49: 10049-10060. DOI: 10.1016/S0040-4020(01)80200-3  0.307
1992 Bols M, Lundt I, Ottosen ER. Preparation of 2-, 3-, and 4-deoxy derivatives of L-rhamnose, and derivatives of 2-azido-2-deoxy-L-rhamnose and 2,6-dideoxy-2-fluoro-L-glucose, for use in glycosylation reactions. Carbohydrate Research. 222: 141-9. PMID 1813104 DOI: 10.1016/0008-6215(91)89013-6  0.324
1992 Bols M, Binderup L, Hansen J, Rasmussen P. Inhibition of collagenase by aranciamycin and aranciamycin derivatives. Journal of Medicinal Chemistry. 35: 2768-71. PMID 1322986 DOI: 10.1021/Jm00093A008  0.302
1992 Bols M. Stereocontrolled synthesis of α-glucosides by intramolecular glycosidation Journal of the Chemical Society, Chemical Communications. 913-914. DOI: 10.1039/C39920000913  0.341
1992 Bols M, Lundt I, Pedersen C. Simple synthesis of (R)-Carnitine from d-Galactono-1,4-lactone Tetrahedron. 48: 319-324. DOI: 10.1016/S0040-4020(01)88143-6  0.301
1991 Bols M. Stereoselective synthesis of 1-O-pivaloyl .beta.-D-glucopyranuronic acid The Journal of Organic Chemistry. 56: 5943-5945. DOI: 10.1021/Jo00020A044  0.307
1990 Bols M, Lundt I, Aksnes DW, Brekke T, Maartmann-Moe K, Tønnesen HH, Tokii T. Preparation of 2,3-Epoxyaldonolactones and their Conversion into 2-Fluoro-2-deoxy-aldonolactones and -sugars. Acta Chemica Scandinavica. 44: 252-256. DOI: 10.3891/Acta.Chem.Scand.44-0252  0.331
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