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Raphael T Labruere - Publications

Affiliations: 
Université Paris-Saclay, Gif-sur-Yvette, Île-de-France, France 
Area:
bioorganic chemistry; chemical biology; bioorthogonal reactions; prodrug
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26 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Espinosa A, Rascol E, Abellán Flos M, Skarbek C, Lieben P, Bannerman E, Martinez AD, Pethe S, Benoit P, Nélieu S, Labruère R. Re-designing environmentally persistent pharmaceutical pollutant through programmed inactivation: The case of methotrexate. Chemosphere. 306: 135616. PMID 35810859 DOI: 10.1016/j.chemosphere.2022.135616  0.733
2021 Maslah H, Skarbek C, Gourson C, Plamont MA, Pethe S, Jullien L, Le Saux T, Labruere RT. In-cell generation of anticancer phenanthridine through bioorthogonal cyclization: a paradigm in antitumor prodrug development. Angewandte Chemie (International Ed. in English). PMID 34487611 DOI: 10.1002/anie.202110041  0.783
2021 Espinosa A, Nélieu S, Lieben P, Skarbek C, Labruère R, Benoit P. Photodegradation of methotrexate in aqueous solution: degradation kinetics and identification of transformation products. Environmental Science and Pollution Research International. PMID 34431057 DOI: 10.1007/s11356-021-15820-3  0.729
2020 Maslah H, Skarbek C, Pethe S, Labruère R. Anticancer boron-containing prodrugs responsive to oxidative stress from the tumor microenvironment. European Journal of Medicinal Chemistry. 207: 112670. PMID 32858470 DOI: 10.1016/J.Ejmech.2020.112670  0.753
2019 Labruère R, Sona AJ, Turos E. Anti-Methicillin-Resistant Nanoantibiotics. Frontiers in Pharmacology. 10: 1121. PMID 31636560 DOI: 10.3389/Fphar.2019.01121  0.566
2019 Skarbek C, Serra S, Maslah H, Rascol E, Labruère R. Arylboronate prodrugs of doxorubicin as promising chemotherapy for pancreatic cancer. Bioorganic Chemistry. 91: 103158. PMID 31376782 DOI: 10.1016/J.Bioorg.2019.103158  0.718
2019 Jagu E, Pomel S, Pethe S, Cintrat JC, Loiseau PM, Labruère R. Spermine-NBD as fluorescent probe for studies of the polyamine transport system in Leishmania donovani. Bioorganic & Medicinal Chemistry Letters. 29: 1710-1713. PMID 31122868 DOI: 10.1016/J.Bmcl.2019.05.030  0.747
2018 Serra S, Alouane A, Le Saux T, Huvelle S, Plasson R, Schmidt F, Jullien L, Labruère R. A chemically encoded timer for dual molecular delivery at tailored ranges and concentrations. Chemical Communications (Cambridge, England). PMID 29872786 DOI: 10.1039/C8Cc03253J  0.739
2018 Jagu E, Pomel S, Diez-Martinez A, Rascol E, Pethe S, Loiseau PM, Labruère R. Synthesis and antikinetoplastid evaluation of bis(benzyl)spermidine derivatives. European Journal of Medicinal Chemistry. 150: 655-666. PMID 29567458 DOI: 10.1016/J.Ejmech.2018.02.087  0.712
2017 Jagu E, Pomel S, Pethe S, Loiseau PM, Labruère R. Polyamine-based analogs and conjugates as antikinetoplastid agents. European Journal of Medicinal Chemistry. 139: 982-1015. PMID 28886510 DOI: 10.1016/J.Ejmech.2017.08.014  0.776
2017 Jagu E, Pomel S, Diez-Martinez A, Ramiandrasoa F, Krauth-Siegel RL, Pethe S, Blonski C, Labruère R, Loiseau PM. Synthesis and in vitro antikinetoplastid activity of polyamine-hydroxybenzotriazole conjugates. Bioorganic & Medicinal Chemistry. 25: 84-90. PMID 27793448 DOI: 10.1016/J.Bmc.2016.10.013  0.745
2015 Alouane A, Labruère R, Le Saux T, Schmidt F, Jullien L. Self-Immolative Spacers: Kinetic Aspects, Structure-Property Relationships, and Applications. Angewandte Chemie (International Ed. in English). 54: 7492-509. PMID 26053475 DOI: 10.1002/Anie.201500088  0.725
2015 Jagu E, Djilali R, Pomel S, Ramiandrasoa F, Pethe S, Labruère R, Loiseau PM, Blonski C. Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives. Bioorganic & Medicinal Chemistry Letters. 25: 207-9. PMID 25499437 DOI: 10.1016/J.Bmcl.2014.11.073  0.778
2015 Alouane A, Labruère R, Le Saux T, Schmidt F, Jullien L. Selbstzerlegende Spacer: kinetische Aspekte, Struktur-Eigenschafts-Beziehungen und Anwendungen Angewandte Chemie. 127: 7600-7619. DOI: 10.1002/Ange.201500088  0.684
2014 Alouane A, Labruère R, Silvestre KJ, Le Saux T, Schmidt F, Jullien L. Disassembly kinetics of quinone-methide-based self-immolative spacers that contain aromatic nitrogen heterocycles. Chemistry, An Asian Journal. 9: 1334-40. PMID 24652669 DOI: 10.1002/Asia.201400051  0.736
2013 Alouane A, Labruère R, Le Saux T, Aujard I, Dubruille S, Schmidt F, Jullien L. Light activation for the versatile and accurate kinetic analysis of disassembly of self-immolative spacers. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 11717-24. PMID 23861286 DOI: 10.1002/Chem.201301298  0.722
2013 Reille-Seroussi M, Labruère R, Inguimbert N, Broussy S, Gagey-Eilstein N, Liu W, Vidal M, Huguenot F. Thienopyrimidinedione Formation Versus Ester Hydrolysis from Ureido Carboxylic Acid Methyl Ester Synthesis. 45: 479-490. DOI: 10.1055/S-0032-1318100  0.302
2013 Labruère R, Helissey P, Desbène‐Finck S, Giorgi‐Renault S. Synthesis of New Furo[3,4‐b]quinolin‐1(3H)‐one Scaffolds Derived from γ‐Lactone‐Fused Quinolin‐4(1H)‐ones Helvetica Chimica Acta. 96: 919-923. DOI: 10.1002/Hlca.201200313  0.308
2012 Labruère R, Alouane A, Le Saux T, Aujard I, Pelupessy P, Gautier A, Dubruille S, Schmidt F, Jullien L. "Self-immolative" spacer for uncaging with fluorescence reporting. Angewandte Chemie (International Ed. in English). 51: 9344-7. PMID 22930567 DOI: 10.1002/Anie.201204032  0.706
2012 Labruère R, Turos E. Attenuating the size and molecular carrier capabilities of polyacrylate nanoparticles by a hydrophobic fluorine effect. Bioorganic & Medicinal Chemistry. 20: 5042-5. PMID 22789705 DOI: 10.1016/J.Bmc.2012.06.010  0.566
2012 Labruere R, Helissey P, Desbene-Finck S, Giorgi-Renault S. Synthesis of the 3,4,5-Trimethoxy-2-(3,4-methylenedioxy-6-nitrophenyl) benzaldehyde for Divergent Preparation of Cytotoxic Biaryls Letters in Organic Chemistry. 9: 568-571. DOI: 10.2174/157017812802850276  0.679
2010 Labruère R, Gautier B, Testud M, Seguin J, Lenoir C, Desbène-Finck S, Helissey P, Garbay C, Chabot GG, Vidal M, Giorgi-Renault S. Design, synthesis, and biological evaluation of the first podophyllotoxin analogues as potential vascular-disrupting agents. Chemmedchem. 5: 2016-25. PMID 20979080 DOI: 10.1002/Cmdc.201000305  0.704
2010 Labruère R, Sicard R, Cormier R, Turos E, West L. Poly(vinyl benzoate) nanoparticles for molecular delivery: Studies on their preparation and in vitro properties. Journal of Controlled Release : Official Journal of the Controlled Release Society. 148: 234-40. PMID 20728487 DOI: 10.1016/J.Jconrel.2010.08.016  0.689
2010 Labruère R, Gautier B, Testud M, Seguin J, Lenoir C, Desbène‐Finck S, Helissey P, Garbay C, Chabot GG, Vidal M, Giorgi‐Renault S. Inside Cover: Design, Synthesis, and Biological Evaluation of the First Podophyllotoxin Analogues as Potential Vascular-Disrupting Agents (ChemMedChem 12/2010) Chemmedchem. 5: 1958-1958. DOI: 10.1002/Cmdc.201090055  0.328
2008 Labruère R, Helissey P, Desbène-Finck S, Giorgi-Renault S. Design and effective synthesis of the first 4-aza-2,3-didehydropodophyllotoxin rigid aminologue: a N-methyl-4-[(3,4,5-trimethoxyphenyl)amino)]-1,2-dihydroquinoline-lactone. The Journal of Organic Chemistry. 73: 3642-5. PMID 18380479 DOI: 10.1021/Jo800166B  0.665
2006 Labruère R, Desbène-Finck S, Helissey P, Giorgi-Renault S. Efficient Syntheses of Thiono and Dithio Analogues of Tetronic Acid Synthesis. 2006: 4163-4166. DOI: 10.1055/S-2006-950351  0.64
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