Year |
Citation |
Score |
2023 |
Fernández-de-la-Pradilla A, Royo S, Schirmeister T, Barthels F, Świderek K, González FV, Moliner V. Impact of the Warhead of Dipeptidyl Keto Michael Acceptors on the Inhibition Mechanism of Cysteine Protease Cathepsin L. Acs Catalysis. 13: 13354-13368. PMID 37881790 DOI: 10.1021/acscatal.3c02748 |
0.684 |
|
2023 |
Arafet K, Royo S, Schirmeister T, Barthels F, González FV, Moliner V. Impact of the Recognition Part of Dipeptidyl Nitroalkene Compounds on the Inhibition Mechanism of Cysteine Proteases Cruzain and Cathepsin L. Acs Catalysis. 13: 6289-6300. PMID 37180968 DOI: 10.1021/acscatal.3c01035 |
0.653 |
|
2020 |
Macías-Villamizar VE, Cuca-Suárez L, Rodríguez S, González FV. Formal [3+2] Cycloaddition Reactions of Electron-Rich Aryl Epoxides with Alkenes under Lewis Acid Catalysis Affording Tetrasubstituted Tetrahydrofurans. Molecules (Basel, Switzerland). 25. PMID 32041165 DOI: 10.3390/molecules25030692 |
0.375 |
|
2019 |
Bou-Iserte L, Latorre A, Rodríguez S, González FV. Three-Step Telescoped Synthesis of Monosubstituted Vicinal Diamines from Aldehydes. Acs Omega. 4: 2261-2267. PMID 31459468 DOI: 10.1021/acsomega.8b03030 |
0.757 |
|
2018 |
Royo S, Schirmeister T, Kaiser M, Jung S, Rodríguez S, Bautista JM, González FV. Antiprotozoal and cysteine proteases inhibitory activity of dipeptidyl enoates. Bioorganic & Medicinal Chemistry. PMID 30037754 DOI: 10.1016/J.Bmc.2018.07.015 |
0.629 |
|
2016 |
Latorre A, Schirmeister T, Kesselring J, Jung S, Johé P, Hellmich UA, Heilos A, Engels B, Krauth-Siegel RL, Dirdjaja N, Bou-Iserte L, Rodríguez S, González FV. Dipeptidyl Nitroalkenes as Potent Reversible Inhibitors of Cysteine Proteases Rhodesain and Cruzain. Acs Medicinal Chemistry Letters. 7: 1073-1076. PMID 27994740 DOI: 10.1021/Acsmedchemlett.6B00276 |
0.72 |
|
2015 |
Royo S, Rodríguez S, Schirmeister T, Kesselring J, Kaiser M, González FV. Dipeptidyl Enoates As Potent Rhodesain Inhibitors That Display a Dual Mode of Action. Chemmedchem. 10: 1484-7. PMID 26179752 DOI: 10.1002/Cmdc.201500204 |
0.647 |
|
2015 |
Latorre A, Rodríguez S, González FV, Florea BI, Overkleeft HS. Synthetic Studies on the Preparation of Alanyl Epoxysulfones as Cathepsin Cysteine Protease Electrophilic Traps. The Journal of Organic Chemistry. 80: 7752-6. PMID 26147718 DOI: 10.1021/acs.joc.5b01013 |
0.768 |
|
2014 |
Willemen HL, Campos PM, Lucas E, Morreale A, Gil-Redondo R, Agut J, González FV, Ramos P, Heijnen C, Mayor F, Kavelaars A, Murga C. A novel p38 MAPK docking-groove-targeted compound is a potent inhibitor of inflammatory hyperalgesia. The Biochemical Journal. 459: 427-39. PMID 24517375 DOI: 10.1042/Bj20130172 |
0.666 |
|
2014 |
Fabregat-Cabello N, Sancho JV, Vidal A, González FV, Roig-Navarro AF. Development and validation of a liquid chromatography isotope dilution mass spectrometry method for the reliable quantification of alkylphenols in environmental water samples by isotope pattern deconvolution. Journal of Chromatography. A. 1328: 43-51. PMID 24423386 DOI: 10.1016/j.chroma.2013.12.077 |
0.559 |
|
2013 |
Agut J, Vidal A, RodrÃguez S, González FV. Dynamic kinetic asymmetric ring-opening/reductive amination sequence of racemic nitroepoxides with chiral amines: enantioselective synthesis of chiral vicinal diamines. The Journal of Organic Chemistry. 78: 5717-22. PMID 23641667 DOI: 10.1021/jo400501k |
0.726 |
|
2012 |
Latorre A, López I, Ramírez V, Rodríguez S, Izquierdo J, González FV, Vicent C. Radical mechanism in the elimination of 2-arylsulfinyl esters. The Journal of Organic Chemistry. 77: 5191-7. PMID 22582746 DOI: 10.1021/jo300699w |
0.509 |
|
2011 |
Izquierdo J, Rodríguez S, González FV. Regioselective ring opening and isomerization reactions of 3,4-epoxyesters catalyzed by boron trifluoride. Organic Letters. 13: 3856-9. PMID 21732641 DOI: 10.1021/ol201378w |
0.535 |
|
2007 |
González FV, Izquierdo J, Rodríguez S, McKerrow JH, Hansell E. Dipeptidyl-alpha,beta-epoxyesters as potent irreversible inhibitors of the cysteine proteases cruzain and rhodesain. Bioorganic & Medicinal Chemistry Letters. 17: 6697-700. PMID 17977725 DOI: 10.1016/J.Bmcl.2007.10.056 |
0.475 |
|
2007 |
López I, RodrÃguez S, Izquierdo J, González FV. Highly stereoselective epoxidation of alpha-methyl-gamma-hydroxy-alpha,beta-unsaturated esters: rationalization and synthetic applications. The Journal of Organic Chemistry. 72: 6614-7. PMID 17655257 DOI: 10.1021/jo0709955 |
0.464 |
|
1998 |
Marco JA, Carda M, González F, Rodríguez S, Castillo E, Murga J. Diastereoselectivity in Organometallic Additions to the Carbonyl Group of Protected Erythrulose Derivatives. The Journal of Organic Chemistry. 63: 698-707. PMID 11672063 DOI: 10.1021/jo9716744 |
0.597 |
|
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