Phillip Robinson - Publications

Affiliations: 
Cell Signalling Children's Medical Research Institute, New South Wales, Australia, Westmead, New South Wales, Australia 

30 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2024 McCluskey A, Prichard K, Chau N, Xue J, Krauss M, Sakoff JA, Gilbert J, Bahnik C, Muehlbauer M, Radetzki S, Robinson PJ, Haucke V. Inhibition clathrin mediated endocytosis: Pitstop 1 and Pitstop 2 chimeras. Chemmedchem. e202400253. PMID 38894585 DOI: 10.1002/cmdc.202400253  0.439
2023 Odell LR, Jones NC, Chau N, Robertson MJ, Ambrus JI, Deane FM, Young KA, Whiting A, Xue J, Prichard K, Daniel JA, Gorgani NN, O'Brien TJ, Robinson PJ, McCluskey A. The sulfonadyns: a class of aryl sulfonamides inhibiting dynamin I GTPase and clathrin mediated endocytosis are anti-seizure in animal models. Rsc Medicinal Chemistry. 14: 1492-1511. PMID 37593570 DOI: 10.1039/d2md00371f  0.603
2022 Cossar PJ, Cardoso D, Mathwin D, Russell CC, Chiew B, Hamilton MP, Baker JR, Young KA, Chau N, Robinson PJ, McCluskey A. Wiskostatin and other carbazole scaffolds as off target inhibitors of dynamin I GTPase activity and endocytosis. European Journal of Medicinal Chemistry. 247: 115001. PMID 36577213 DOI: 10.1016/j.ejmech.2022.115001  0.455
2022 Odell LR, Robertson MJ, Young KA, McGeachie AB, Quan A, Robinson PJ, McCluskey A. Prodrugs of the Archetypal Dynamin Inhibitor Bis-T-22. Chemmedchem. e202200400. PMID 36351775 DOI: 10.1002/cmdc.202200400  0.317
2022 Russell CC, Prichard KL, O'Brien NS, McCluskey A, Robinson PJ, Baker JR. Synthesis of Phthaladyn-29 and Naphthalimide-10, GTP Site Directed Dynamin GTPase Inhibitors. Methods in Molecular Biology (Clifton, N.J.). 2417: 239-258. PMID 35099804 DOI: 10.1007/978-1-0716-1916-2_18  0.362
2022 Baker JR, O'Brien NS, Prichard KL, Robinson PJ, McCluskey A, Russell CC. Dynole 34-2 and Acrylo-Dyn 2-30, Novel Dynamin GTPase Chemical Biology Probes. Methods in Molecular Biology (Clifton, N.J.). 2417: 221-238. PMID 35099803 DOI: 10.1007/978-1-0716-1916-2_17  0.35
2021 Odell LR, Chau N, Russell CC, Young KA, Gilbert J, Robinson PJ, Sakoff JA, McCluskey A. Pyrimidyn based dynamin inhibitors as novel cytotoxic agents. Chemmedchem. PMID 34590434 DOI: 10.1002/cmdc.202100560  0.35
2016 Odell LR, Abdel-Hamid MK, Hill TA, Chau N, Young KA, Deane FM, Sakoff JA, Andersson S, Daniel JA, Robinson PJ, McCluskey A. Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain. Journal of Medicinal Chemistry. PMID 27997171 DOI: 10.1021/acs.jmedchem.6b01422  0.609
2016 Robertson MJ, Horatscheck A, Sauer S, von Kleist L, Baker JR, Stahlschmidt W, Nazaré M, Whiting A, Chau N, Robinson PJ, Haucke V, McCluskey A. 5-Aryl-2-(naphtha-1-yl)sulfonamido-thiazol-4(5H)-ones as clathrin inhibitors. Organic & Biomolecular Chemistry. PMID 27853797 DOI: 10.1039/c6ob02308h  0.401
2015 Abdel-Hamid MK, Macgregor KA, Odell LR, Chau N, Mariana A, Whiting A, Robinson PJ, McCluskey A. 1,8-Naphthalimide derivatives: new leads against dynamin I GTPase activity. Organic & Biomolecular Chemistry. 13: 8016-28. PMID 26118967 DOI: 10.1039/c5ob00751h  0.455
2015 Daniel JA, Chau N, Abdel-Hamid MK, Hu L, von Kleist L, Whiting A, Krishnan S, Maamary P, Joseph SR, Simpson F, Haucke V, McCluskey A, Robinson PJ. Phenothiazine-derived antipsychotic drugs inhibit dynamin and clathrin-mediated endocytosis. Traffic (Copenhagen, Denmark). 16: 635-54. PMID 25693808 DOI: 10.1111/tra.12272  0.627
2014 Kockx M, Karunakaran D, Traini M, Xue J, Huang KY, Nawara D, Gaus K, Jessup W, Robinson PJ, Kritharides L. Pharmacological inhibition of dynamin II reduces constitutive protein secretion from primary human macrophages. Plos One. 9: e111186. PMID 25347775 DOI: 10.1371/journal.pone.0111186  0.311
2014 MacGregor KA, Abdel-Hamid MK, Odell LR, Chau N, Whiting A, Robinson PJ, McCluskey A. Development of quinone analogues as dynamin GTPase inhibitors. European Journal of Medicinal Chemistry. 85: 191-206. PMID 25084145 DOI: 10.1016/j.ejmech.2014.06.070  0.427
2014 Robertson MJ, Deane FM, Stahlschmidt W, von Kleist L, Haucke V, Robinson PJ, McCluskey A. Synthesis of the Pitstop family of clathrin inhibitors. Nature Protocols. 9: 1592-606. PMID 24922269 DOI: 10.1038/nprot.2014.106  0.306
2014 MacGregor KA, Robertson MJ, Young KA, von Kleist L, Stahlschmidt W, Whiting A, Chau N, Robinson PJ, Haucke V, McCluskey A. Development of 1,8-naphthalimides as clathrin inhibitors. Journal of Medicinal Chemistry. 57: 131-43. PMID 24299503 DOI: 10.1021/jm4015263  0.414
2013 McCluskey A, Daniel JA, Hadzic G, Chau N, Clayton EL, Mariana A, Whiting A, Gorgani NN, Lloyd J, Quan A, Moshkanbaryans L, Krishnan S, Perera S, Chircop M, von Kleist L, ... ... Robinson PJ, et al. Building a better dynasore: the dyngo compounds potently inhibit dynamin and endocytosis. Traffic (Copenhagen, Denmark). 14: 1272-89. PMID 24025110 DOI: 10.1111/Tra.12119  0.597
2013 McGeachie AB, Odell LR, Quan A, Daniel JA, Chau N, Hill TA, Gorgani NN, Keating DJ, Cousin MA, van Dam EM, Mariana A, Whiting A, Perera S, Novelle A, Young KA, ... ... Robinson PJ, et al. Pyrimidyn compounds: dual-action small molecule pyrimidine-based dynamin inhibitors. Acs Chemical Biology. 8: 1507-18. PMID 23642287 DOI: 10.1021/Cb400137P  0.657
2013 Smith CM, Haucke V, McCluskey A, Robinson PJ, Chircop M. Inhibition of clathrin by pitstop 2 activates the spindle assembly checkpoint and induces cell death in dividing HeLa cancer cells. Molecular Cancer. 12: 4. PMID 23327284 DOI: 10.1186/1476-4598-12-4  0.305
2013 Gordon CP, Venn-Brown B, Robertson MJ, Young KA, Chau N, Mariana A, Whiting A, Chircop M, Robinson PJ, McCluskey A. Development of second-generation indole-based dynamin GTPase inhibitors. Journal of Medicinal Chemistry. 56: 46-59. PMID 23167654 DOI: 10.1021/jm300844m  0.404
2012 Robertson MJ, Hadzic G, Ambrus J, Pomè DY, Hyde E, Whiting A, Mariana A, von Kleist L, Chau N, Haucke V, Robinson PJ, McCluskey A. The Rhodadyns, a New Class of Small Molecule Inhibitors of Dynamin GTPase Activity. Acs Medicinal Chemistry Letters. 3: 352-6. PMID 24900478 DOI: 10.1021/ml200284s  0.459
2012 Daniel JA, Malladi CS, Kettle E, McCluskey A, Robinson PJ. Analysis of synaptic vesicle endocytosis in synaptosomes by high-content screening. Nature Protocols. 7: 1439-55. PMID 22767087 DOI: 10.1038/nprot.2012.070  0.51
2011 Chircop M, Perera S, Mariana A, Lau H, Ma MP, Gilbert J, Jones NC, Gordon CP, Young KA, Morokoff A, Sakoff J, O'Brien TJ, McCluskey A, Robinson PJ. Inhibition of dynamin by dynole 34-2 induces cell death following cytokinesis failure in cancer cells. Molecular Cancer Therapeutics. 10: 1553-62. PMID 21750222 DOI: 10.1158/1535-7163.MCT-11-0067  0.314
2010 Odell LR, Howan D, Gordon CP, Robertson MJ, Chau N, Mariana A, Whiting AE, Abagyan R, Daniel JA, Gorgani NN, Robinson PJ, McCluskey A. The pthaladyns: GTP competitive inhibitors of dynamin I and II GTPase derived from virtual screening. Journal of Medicinal Chemistry. 53: 5267-80. PMID 20575553 DOI: 10.1021/Jm100442U  0.64
2010 Joshi S, Perera S, Gilbert J, Smith CM, Mariana A, Gordon CP, Sakoff JA, McCluskey A, Robinson PJ, Braithwaite AW, Chircop M. The dynamin inhibitors MiTMAB and OcTMAB induce cytokinesis failure and inhibit cell proliferation in human cancer cells. Molecular Cancer Therapeutics. 9: 1995-2006. PMID 20571068 DOI: 10.1158/1535-7163.MCT-10-0161  0.303
2010 Hill TA, Mariana A, Gordon CP, Odell LR, Robertson MJ, McGeachie AB, Chau N, Daniel JA, Gorgani NN, Robinson PJ, McCluskey A. Iminochromene inhibitors of dynamins I and II GTPase activity and endocytosis. Journal of Medicinal Chemistry. 53: 4094-102. PMID 20426422 DOI: 10.1021/jm100119c  0.613
2009 Hill TA, Gordon CP, McGeachie AB, Venn-Brown B, Odell LR, Chau N, Quan A, Mariana A, Sakoff JA, Chircop M, Robinson PJ, McCluskey A. Inhibition of dynamin mediated endocytosis by the dynoles--synthesis and functional activity of a family of indoles. Journal of Medicinal Chemistry. 52: 3762-73. PMID 19459681 DOI: 10.1021/jm900036m  0.492
2009 Odell LR, Chau N, Mariana A, Graham ME, Robinson PJ, McCluskey A. Azido and diazarinyl analogues of bis-tyrphostin as asymmetrical inhibitors of dynamin GTPase. Chemmedchem. 4: 1182-8. PMID 19437476 DOI: 10.1002/cmdc.200900054  0.383
2007 Quan A, McGeachie AB, Keating DJ, van Dam EM, Rusak J, Chau N, Malladi CS, Chen C, McCluskey A, Cousin MA, Robinson PJ. Myristyl trimethyl ammonium bromide and octadecyl trimethyl ammonium bromide are surface-active small molecule dynamin inhibitors that block endocytosis mediated by dynamin I or dynamin II. Molecular Pharmacology. 72: 1425-39. PMID 17702890 DOI: 10.1124/Mol.107.034207  0.434
2005 Hill T, Odell LR, Edwards JK, Graham ME, McGeachie AB, Rusak J, Quan A, Abagyan R, Scott JL, Robinson PJ, McCluskey A. Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins. Journal of Medicinal Chemistry. 48: 7781-8. PMID 16302817 DOI: 10.1021/Jm040208L  0.442
2004 Hill TA, Odell LR, Quan A, Abagyan R, Ferguson G, Robinson PJ, McCluskey A. Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity. Bioorganic & Medicinal Chemistry Letters. 14: 3275-8. PMID 15149689 DOI: 10.1016/J.Bmcl.2004.03.096  0.41
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