Year |
Citation |
Score |
2021 |
Porcu A, Mostallino R, Serra V, Melis M, Sogos V, Beggiato S, Ferraro L, Manetti F, Gianibbi B, Bettler B, Corelli F, Mugnaini C, Castelli MP. COR758, a negative allosteric modulator of GABA receptors. Neuropharmacology. 189: 108537. PMID 33798546 DOI: 10.1016/j.neuropharm.2021.108537 |
0.585 |
|
2020 |
Porcu A, Vaughan M, Nilsson A, Arimoto N, Lamia K, Welsh DK. Vulnerability to helpless behavior is regulated by the circadian clock component CRYPTOCHROME in the mouse nucleus accumbens. Proceedings of the National Academy of Sciences of the United States of America. PMID 32487727 DOI: 10.1073/Pnas.2000258117 |
0.367 |
|
2018 |
Porcu A, Melis M, Turecek R, Ullrich C, Mocci I, Bettler B, Gessa GL, Castelli MP. Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a Gαi/o protein inhibitor. Neuropharmacology. 133: 107-120. PMID 29407764 DOI: 10.1016/J.Neuropharm.2018.01.024 |
0.407 |
|
2016 |
Porcu A, Lobina C, Giunta D, Solinas M, Mugnaini C, Castelli MP. In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator. European Journal of Pharmacology. 791: 115-123. PMID 27578262 DOI: 10.1016/J.Ejphar.2016.08.032 |
0.421 |
|
2015 |
De Luca MA, Castelli MP, Loi B, Porcu A, Martorelli M, Miliano C, Kellett K, Davidson C, Stair JL, Schifano F, Di Chiara G. Native CB1 receptor affinity, intrinsic activity and accumbens shell dopamine stimulant properties of third generation SPICE/K2 cannabinoids: BB-22, 5F-PB-22, 5F-AKB-48 and STS-135. Neuropharmacology. 105: 630-638. PMID 26686391 DOI: 10.1016/J.Neuropharm.2015.11.017 |
0.457 |
|
2013 |
Ferraro L, Loche A, Beggiato S, Tomasini MC, Antonelli T, Colombo G, Lobina C, Carai MA, Porcu A, Castelli MP, Clerici F, Borelli AC, Cacciaglia R, Tanganelli S. The new compound GET73, N-[(4-trifluoromethyl)benzyl]4-methoxybutyramide, Regulates hippocampal Aminoacidergic transmission possibly via an allosteric modulation of mGlu5 receptor. Behavioural evidence of its "anti-alcohol" and anxiolytic properties. Current Medicinal Chemistry. 20: 3339-57. PMID 23862615 DOI: 10.2174/09298673113209990167 |
0.481 |
|
2013 |
Mugnaini C, Pedani V, Casu A, Lobina C, Casti A, Maccioni P, Porcu A, Giunta D, Lamponi S, Solinas M, Dragoni S, Valoti M, Colombo G, Castelli MP, Gessa GL, et al. Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor. Journal of Medicinal Chemistry. 56: 3620-35. PMID 23544432 DOI: 10.1021/Jm400144W |
0.39 |
|
2013 |
Madeddu C, Casti A, Porcu A, Castelli MP, Ennas MG. Δ9-tetrahydrocannabinol attenuated methamphetamine-induced increase of neuronal nitric oxide synthase expression and Glial Fibrillary Acidic Protein immunoreactivity Italian Journal of Anatomy and Embryology. 118: 122. DOI: 10.13128/Ijae-14875 |
0.406 |
|
Show low-probability matches. |