Doug Pettibone

Affiliations: 
Merck, Semoy, Centre-Val de Loire, France 
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"Doug Pettibone"
Mean distance: 14.57 (cluster 11)
 
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Publications

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Bodmer-Narkevitch V, Anthony NJ, Cofre V, et al. (2010) Indazole derivatives as novel bradykinin B1 receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 20: 7011-4
Wolkenberg SE, Zhao Z, Wisnoski DD, et al. (2009) Discovery of GlyT1 inhibitors with improved pharmacokinetic properties. Bioorganic & Medicinal Chemistry Letters. 19: 1492-5
Zhao Z, Leister WH, O'Brien JA, et al. (2009) Discovery of N-{[1-(propylsulfonyl)-4-pyridin-2-ylpiperidin-4-yl]methyl}benzamides as novel, selective and potent GlyT1 inhibitors. Bioorganic & Medicinal Chemistry Letters. 19: 1488-91
Kuduk SD, Chang RK, Dipardo RM, et al. (2008) Bradykinin B1 receptor antagonists: an alpha-hydroxy amide with an improved metabolism profile. Bioorganic & Medicinal Chemistry Letters. 18: 5107-10
Su DS, Lim JL, Tinney E, et al. (2008) 2-Aminobenzophenones as a novel class of bradykinin B1 receptor antagonists. Journal of Medicinal Chemistry. 51: 3946-52
Feng DM, DiPardo RM, Wai JM, et al. (2008) A new class of bradykinin B1 receptor antagonists with high oral bioavailability and minimal PXR activity. Bioorganic & Medicinal Chemistry Letters. 18: 682-7
Bergman JM, Roecker AJ, Mercer SP, et al. (2008) Proline bis-amides as potent dual orexin receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 18: 1425-30
Wood MR, Schirripa KM, Kim JJ, et al. (2008) Alpha-hydroxy amides as a novel class of bradykinin B1 selective antagonists. Bioorganic & Medicinal Chemistry Letters. 18: 716-20
Kuduk SD, DiPardo RM, Chang RK, et al. (2007) Bradykinin B1 antagonists: biphenyl SAR studies in the cyclopropanecarboxamide series. Bioorganic & Medicinal Chemistry Letters. 17: 3608-12
Su DS, Lim JL, Markowitz MK, et al. (2007) Potent bradykinin B1 receptor antagonists: 4-substituted phenyl cyclohexanes. Bioorganic & Medicinal Chemistry Letters. 17: 3006-9
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