| Year |
Citation |
Score |
| 2011 |
Overman LE, Humphreys PG, Welmaker GS. The aza-cope/mannich reaction Organic Reactions. 75: 747-820. DOI: 10.1002/0471264180.Or075.04 |
0.351 |
|
| 1996 |
Marshall JA, Jablonowski JA, Welmaker GS. On the Relative Reactivities of Allyl, Crotyl, alpha-Oxygenated Crotyl, gamma-Oxygenated alpha-Methylallyl, and Allenyl Tri-n-butylstannane Reagents in Lewis Acid Promoted Additions to Aldehydes. The Journal of Organic Chemistry. 61: 2904-2907. PMID 11667135 DOI: 10.1021/Jo9519975 |
0.477 |
|
| 1996 |
Marshall JA, Jablonowski JA, Welmaker GS. On the relative reactivities of allyl, crotyl, α-oxygenated crotyl, γ-oxygenated α-methylallyl, and allenyl tri-n-butylstannane reagents in Lewis acid promoted additions to aldehydes Journal of Organic Chemistry. 61: 2904-2907. |
0.479 |
|
| 1995 |
Lögers M, Overman LE, Welmaker GS. Mannich biscyclizations. Total synthesis of (-)-ajmalicine Journal of the American Chemical Society. 117: 9139-9150. DOI: 10.1021/Ja00141A004 |
0.308 |
|
| 1991 |
Marshall JA, Welmaker GS, Gung BW. On the 1,3-isomerization of nonracemic α-(alkoxy)allyl stannanes Journal of the American Chemical Society. 113: 647-656. |
0.319 |
|
| Low-probability matches (unlikely to be authored by this person) |
| 1994 |
Marshall JA, Welmaker GS. Enantioselective synthesis of (+)- and (-)-muricatacin through SE2′ addition of nonracemic γ-silyloxy allylic stannanes to aldehydes Journal of Organic Chemistry. 59: 4122-4125. |
0.268 |
|
| 2009 |
Wilson MA, Filzen G, Welmaker GS. A microwave-assisted, green procedure for the synthesis of N-aryl sulfonyl and N-aryl pyrroles Tetrahedron Letters. 50: 4807-4809. DOI: 10.1016/j.tetlet.2009.06.079 |
0.257 |
|
| 1991 |
Marshall JA, Welmaker GS. Chiral γ-silyloxy allylstannanes as synthetic reagents. Proof of absolute configuration Tetrahedron Letters. 32: 2101-2104. DOI: 10.1016/S0040-4039(00)71247-0 |
0.202 |
|
| 1992 |
Marshall JA, Welmaker GS. (Z)- and (E)-γ-silyloxy allylic stannanes. Highly syn selective reagents for SE′ additions to aldehydes Journal of Organic Chemistry. 57: 7158-7163. |
0.182 |
|
| 1994 |
Leotta GJ, Overman LE, Welmaker GS. A convenient method for the preparation of 3-substituted glutarate diesters Journal of Organic Chemistry. 59: 1946. |
0.14 |
|
| 1993 |
Welmaker GS. A simple, efficient preparation of 1,1-bis(Trimethylsiloxy)-1,3-butadiene Organic Preparations and Procedures International. 25: 595-597. DOI: 10.1080/00304949309458009 |
0.136 |
|
| 2017 |
Wu J, Cippitelli A, Zhang Y, Debevec G, Schoch J, Ozawa A, Yu Y, Liu H, Chen W, Houghten RA, Welmaker GS, Giulianotti MA, Toll L. Highly Selective and Potent α4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats. Journal of Medicinal Chemistry. PMID 29178785 DOI: 10.1021/Acs.Jmedchem.7B01250 |
0.076 |
|
| 2018 |
Cippitelli A, Brunori G, Schoch J, Armishaw CJ, Wu J, Zaveri NT, Giulianotti MA, Welmaker GS, Toll L. Differential regulation of alcohol taking and seeking by antagonism at α4β2 and α3β4 nAChRs. Psychopharmacology. PMID 29572652 DOI: 10.1007/S00213-018-4883-Y |
0.071 |
|
| 2013 |
Wu J, Zhang Y, Maida LE, Santos RG, Welmaker GS, LaVoi TM, Nefzi A, Yu Y, Houghten RA, Toll L, Giulianotti MA. Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies. Journal of Medicinal Chemistry. 56: 10103-17. PMID 24274400 DOI: 10.1021/Jm401543H |
0.065 |
|
| 2009 |
Moore WJ, Kern JC, Bhat R, Commons TJ, Fukayama S, Goljer I, Krishnamurthy G, Magolda RL, Nogle L, Pitts K, Stauffer B, Trybulski EJ, Welmaker GS, Wilson M, Bodine PV. Modulation of Wnt signaling through inhibition of secreted frizzled-related protein I (sFRP-1) with N-substituted piperidinyl diphenylsulfonyl sulfonamides. Journal of Medicinal Chemistry. 52: 105-16. PMID 19072540 DOI: 10.1021/Jm801144H |
0.063 |
|
| 2015 |
Fleeman R, LaVoi TM, Santos RG, Morales A, Nefzi A, Welmaker GS, Medina-Franco JL, Giulianotti MA, Houghten RA, Shaw LN. Combinatorial Libraries As a Tool for the Discovery of Novel, Broad-Spectrum Antibacterial Agents Targeting the ESKAPE Pathogens. Journal of Medicinal Chemistry. 58: 3340-55. PMID 25780985 DOI: 10.1021/jm501628s |
0.043 |
|
| 2015 |
Houghten RA, Ganno ML, McLaughlin JP, Dooley CT, Eans SO, Santos RG, LaVoi T, Nefzi A, Welmaker G, Giulianotti MA, Toll L. Direct High Throughput In Vivo Screening: Identification of Individual, Novel Antinociceptive Compounds from a Library of 734,821 Pyrrolidine bis-Piperazines. Acs Combinatorial Science. PMID 26651386 DOI: 10.1021/Acscombsci.5B00126 |
0.035 |
|
| 2018 |
Fleeman RM, Debevec G, Antonen K, Adams JL, Santos RG, Welmaker GS, Houghten RA, Giulianotti MA, Shaw LN. Identification of a Novel Polyamine Scaffold With Potent Efflux Pump Inhibition Activity Toward Multi-Drug Resistant Bacterial Pathogens. Frontiers in Microbiology. 9: 1301. PMID 29963035 DOI: 10.3389/fmicb.2018.01301 |
0.034 |
|
| 2016 |
Sandhaus S, Annamalai T, Welmaker G, Houghten RA, Paz C, Garcia PK, Andres A, Narula G, Rodrigues Felix C, Geden S, Netherton M, Gupta R, Rohde KH, Giulianotti MA, Tse-Dinh YC. Small Molecule Inhibitors Targeting Topoisomerase I as Novel Antituberculosis Agents. Antimicrobial Agents and Chemotherapy. PMID 27114277 DOI: 10.1128/Aac.00288-16 |
0.024 |
|
| 2004 |
Welmaker GS, Sabalski JE. A process for the preparation of 1,2,3,4,8,9,10,10a-octahydro-7bH- cyclopenta[b][1,4]diazepino[6,7,1-hi]indole Tetrahedron Letters. 45: 4851-4854. DOI: 10.1016/j.tetlet.2004.04.157 |
0.019 |
|
| 2009 |
Bodine PV, Stauffer B, Ponce-de-Leon H, Bhat RA, Mangine A, Seestaller-Wehr LM, Moran RA, Billiard J, Fukayama S, Komm BS, Pitts K, Krishnamurthy G, Gopalsamy A, Shi M, Kern JC, ... ... Welmaker GS, et al. A small molecule inhibitor of the Wnt antagonist secreted frizzled-related protein-1 stimulates bone formation. Bone. 44: 1063-8. PMID 19254787 DOI: 10.1016/j.bone.2009.02.013 |
0.018 |
|
| 2013 |
Medina-Franco JL, Giulianotti MA, Welmaker GS, Houghten RA. Shifting from the single to the multitarget paradigm in drug discovery. Drug Discovery Today. 18: 495-501. PMID 23340113 DOI: 10.1016/j.drudis.2013.01.008 |
0.01 |
|
| 2006 |
Rosenzweig-Lipson S, Zhang J, Mazandarani H, Harrison BL, Sabb A, Sabalski J, Stack G, Welmaker G, Barrett JE, Dunlop J. Antiobesity-like effects of the 5-HT2C receptor agonist WAY-161503. Brain Research. 1073: 240-51. PMID 16430874 DOI: 10.1016/j.brainres.2005.12.052 |
0.01 |
|
| 2004 |
Sabb AL, Vogel RL, Welmaker GS, Sabalski JE, Coupet J, Dunlop J, Rosenzweig-Lipson S, Harrison B. Cycloalkyl[b][1,4]benzodiazepinoindoles are agonists at the human 5-HT2C receptor. Bioorganic & Medicinal Chemistry Letters. 14: 2603-7. PMID 15109661 DOI: 10.1016/j.bmcl.2004.02.100 |
0.01 |
|
| 2000 |
Welmaker GS, Nelson JA, Sabalski JE, Sabb AL, Potoski JR, Graziano D, Kagan M, Coupet J, Dunlop J, Mazandarani H, Rosenzweig-Lipson S, Sukoff S, Zhang Y. Synthesis and 5-hydroxytryptamine (5-HT) activity of 2,3,4,4a-tetrahydro-1H-pyrazino[1,2-a]quinoxalin-5-(6H)ones and 2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxalines. Bioorganic & Medicinal Chemistry Letters. 10: 1991-4. PMID 10987434 DOI: 10.1016/S0960-894X(00)00400-5 |
0.01 |
|
| Hide low-probability matches. |