| Year |
Citation |
Score |
| 2010 |
WANG B, MERTES MP, BOWMAN MERTES K, TAKUSAGAWA F. ChemInform Abstract: A Novel Intramolecular 1,3-Dipolar Cycloaddition Reaction of a C-6 Substituted Uridine Analog. Cheminform. 22: no-no. DOI: 10.1002/chin.199140242 |
0.48 |
|
| 1994 |
Wang BH, Kagel JR, Mertes MP, Bowmanjames K. Insight into the Chemical Mechanism of Thymidylate Synthase-Catalyzed Reaction Through the Evaluation of Chemical Models: The Role of C6 Sulfhydryl Addition During the Reductive Elimination Step of the Reaction1 Bioorganic Chemistry. 22: 405-420. DOI: 10.1006/Bioo.1994.1034 |
0.539 |
|
| 1993 |
Wang B, Takusagawa F, Mertes MP, Bowman-James K. Structure of the product from a novel cyclization reaction involving a C(6)-substituted uridine analog. Acta Crystallographica. Section C, Crystal Structure Communications. 49: 1568-71. PMID 8217019 DOI: 10.1107/S0108270193004123 |
0.657 |
|
| 1993 |
Kagel JR, Wang B, Mertes MP. A chemical model for the fragmentation reaction in thymidylate synthase catalysis. Synthesis and evaluation of a 5-methylene-1-(1,2,3,4-tetrahydroquinolyl)-6-allyluridine Journal of Organic Chemistry. 58: 2738-2746. DOI: 10.1021/Jo00062A014 |
0.514 |
|
| 1992 |
Bencini A, Bianchi A, Garcia-Espana E, Scott EC, Morales L, Wang B, Deffo T, Takusagawa F, Mertes MP, Mertes KB, Paoletti P. Potential ATPase mimics by polyammonium macrocycles: Criteria for catalytic activity Bioorganic Chemistry. 20: 8-29. DOI: 10.1016/0045-2068(92)90022-U |
0.48 |
|
| 1990 |
WANG B, KAGEL JR, RAO TS, MERTES MP. ChemInform Abstract: A Novel Cyclization Reaction of a C-6 Substituted Uridine Analog: An Entry to 5,6-Dialkylated Uridine Derivatives. Cheminform. 21. DOI: 10.1002/chin.199030298 |
0.491 |
|
| 1989 |
Wang B, Kagel JR, Rao TS, Mertes MP. A novel cyclization reaction of a C-6 substituted uridine analog: An entry to 5,6-dialkylated uridine derivatives Tetrahedron Letters. 30: 7005-7008. DOI: 10.1016/S0040-4039(01)93409-4 |
0.548 |
|
| 1989 |
Gu K, Mertes KB, Mertes MP. Strategy for the synthesis of unsymmetrical N-substituted polyazamacrocycles Tetrahedron Letters. 30: 1323-1326. DOI: 10.1016/S0040-4039(00)99455-3 |
0.36 |
|
| 1989 |
Jiang Z, Chalabi P, Mertes KB, Jahansouz H, Himes RH, Mertes MP. Reactions of formyl phosphate with linear and macrocyclic polyamines Bioorganic Chemistry. 17: 313-329. DOI: 10.1016/0045-2068(89)90034-5 |
0.339 |
|
| 1989 |
Jahansouz H, Mertes KB, Mertes MP, Himes RH. The mechanism of formyl phosphate hydrolysis Bioorganic Chemistry. 17: 207-216. DOI: 10.1016/0045-2068(89)90020-5 |
0.318 |
|
| 1987 |
Al-Razzak LA, Schwepler D, Decedue CJ, Balzarini J, De Clercq E, Mertes MP. 5-Quinone derivatives of 2'-deoxyuridine 5'-phosphate: inhibition and inactivation of thymidylate synthase, antitumor cell, and antiviral studies. Journal of Medicinal Chemistry. 30: 409-19. PMID 3027341 DOI: 10.1021/Jm00385A026 |
0.413 |
|
| 1986 |
Vadnere MK, Maggiora L, Mertes MP. Thiol addition to quinones: model reactions for the inactivation of thymidylate synthase by 5-p-benzoquinonyl-2'-deoxyuridine 5'-phosphate. Journal of Medicinal Chemistry. 29: 1714-20. PMID 3746818 DOI: 10.1021/Jm00159A025 |
0.368 |
|
| 1986 |
Maggiora L, Mertes MP. Diels-Alder reactions of aza dienes: A facile approach to the synthesis of pyridine- and pyridazine-substituted pyrimidine nucleosides Journal of Organic Chemistry. 51: 950-951. DOI: 10.1021/Jo00356A041 |
0.377 |
|
| 1984 |
Conway GA, Park JS, Maggiora L, Mertes MP, Galton N, Michaelis EK. Palladium (II)-catalyzed olefin-coupling reactions of kainic acid: effects of substitution on the isopropenyl group on receptor binding. Journal of Medicinal Chemistry. 27: 52-6. PMID 6317861 DOI: 10.1021/Jm00367A010 |
0.365 |
|
| 1984 |
Park JS, Bigge CF, Hassan ME, Maggiora L, Mertes MP. Conversion of uracil nucleotides into isotopically labelled 5-substituted uracil nucleotides: A convenient route to thymine nucleotides Journal of the Chemical Society, Chemical Communications. 553-554. DOI: 10.1039/C39840000553 |
0.335 |
|
| 1984 |
Chang G, Mertes MP. Palladium(O) catalyzed coupling reactions in the synthesis of 5-arylpyrimidine nucleosides Tetrahedron Letters. 25: 2431-2434. DOI: 10.1016/S0040-4039(01)81197-7 |
0.347 |
|
| 1983 |
Maggiora L, Chang CT, Hasson ME, Bigge CF, Mertes MP. 5-p-benzoquinonyl-2'-deoxyuridine 5'-phosphate: a possible mechanism-based inhibitor of thymidylate synthetase. Journal of Medicinal Chemistry. 26: 1028-36. PMID 6408258 DOI: 10.1002/Chin.198348325 |
0.342 |
|
| 1983 |
Al-Razzak L, Hassan ME, Mertes MP. Aromatic Photosubstitution Reactions for the Synthesis of 5-Aryl-2'-Deoxyuridines Nucleosides and Nucleotides. 2: 243-248. DOI: 10.1080/07328318308078858 |
0.36 |
|
| 1982 |
Balzarini J, De Clercq E, Mertes MP, Shugar D, Torrence PF. 5-Substituted 2'-deoxyuridines: correlation between inhibition of tumor cell growth and inhibition of thymidine kinase and thymidylate synthetase. Biochemical Pharmacology. 31: 3673-82. PMID 7181950 DOI: 10.1016/0006-2952(82)90594-9 |
0.328 |
|
| 1981 |
Bigge CF, Mertes MP. A palladium-catalyzed coupling reaction and a photolytic reaction for the direct synthesis of 5-arylpyrimidine nucleotides Journal of Organic Chemistry. 46: 1994-1997. DOI: 10.1021/Jo00323A005 |
0.335 |
|
| 1981 |
Maggiora L, Chang CCTC, Torrence PF, Mertes MP. 5-Nitro-2′-deoxyuridine 5′-phosphate: A mechanism-based inhibitor of thymidylate synthetase Journal of the American Chemical Society. 103: 3192-3198. DOI: 10.1021/Ja00401A042 |
0.335 |
|
| 1980 |
De Clercq E, Balzarini J, Chang CT, Bigge CF, Kalaritis P, Mertes MP. 5(E)-(3-azidostyryl)-2'-deoxyuridine 5'-phosphate is a photoactivated inhibitor of thymidylate synthetase. Biochemical and Biophysical Research Communications. 97: 1068-75. PMID 7470133 DOI: 10.1016/0006-291X(80)91484-9 |
0.31 |
|
| 1980 |
Park JS, Chang CT, Schmidt CL, Golander Y, De Clercq E, Descamps J, Mertes MP. Oxime and dithiolane derivatives of 5-formyl-2'-deoxyuridine and their 5'-phosphates: antiviral effects and thymidylate synthetase inhibition. Journal of Medicinal Chemistry. 23: 661-5. PMID 6248643 DOI: 10.1002/Chin.198042280 |
0.301 |
|
| 1980 |
Schmidt CL, Chang CT, De Clercq E, Descamps J, Mertes MP. Synthesis of 5-[(methylthio)methyl]-2'-deoxyuridine, the corresponding sulfoxide and sulfone, and their 5'-phosphates: antiviral effects and thymidylate synthetase inhibition. Journal of Medicinal Chemistry. 23: 252-6. PMID 6245212 DOI: 10.1021/Jm00177A008 |
0.37 |
|
| 1980 |
Bigge CF, Kalaritis P, Deck JR, Mertes MP. Palladium-catalyzed coupling reactions of uracil nucleosides and nucleotides Journal of the American Chemical Society. 102: 2033-2038. DOI: 10.1021/Ja00526A044 |
0.316 |
|
| 1980 |
SCHMIDT CL, CHANG CT, DE CLERCQ E, DESCAMPS J, MERTES MP. ChemInform Abstract: SYNTHESIS OF 5-((METHYLTHIO)METHYL)-2′-DEOXYURIDINE, THE CORRESPONDING SULFOXIDE AND SULFONE, AND THEIR 5′-PHOSPHATES: ANTIVIRAL EFFECTS AND THYMIDYLATE SYNTHETASE INHIBITION Chemischer Informationsdienst. 11. DOI: 10.1002/Chin.198034307 |
0.347 |
|
| 1980 |
Park JS, Chang CT-, Mertes MP. 5-((4-Methyl-1,2,3,4-Tetrahydroquinoxalyl)Methyl)-2′-Deoxyuridine 5′-Phosphate: An Analogue Of A Proposed Intermediate In Thymidylate Synthetase Catalysis Cheminform. 11. DOI: 10.1002/Chin.198005364 |
0.313 |
|
| 1980 |
Chang CT-, Edwards MW, Torrence PF, Mertes MP. 5-Cyano-2′-Deoxyuridine 5′-Phosphate: A Potent Competitive Inhibitor Of Thymidylate Synthetase Cheminform. 11. DOI: 10.1002/Chin.198004366 |
0.352 |
|
| 1979 |
De Clercq E, Descamps J, Schmidt CL, Mertes MP. Antiviral activity of 5-methylthiomethyl-2'-deoxyuridine and other 5-substituted 2'-deoxyuridines. Biochemical Pharmacology. 28: 3249-54. PMID 230848 DOI: 10.1016/0006-2952(79)90117-5 |
0.336 |
|
| 1979 |
Brouillette CB, Chang CT, Mertes MP. 5-(alpha-Bromoacetyl)-2'-deoxyuridine 5'-phosphate: an affinity label for thymidylate synthetase. Journal of Medicinal Chemistry. 22: 1541-4. PMID 119854 DOI: 10.1021/Jm00198A022 |
0.645 |
|
| 1979 |
Chang CT, Edwards MW, Torrence PF, Mertes MP. 5-Cyano-2'-deoxyuridine 5'-phosphate: a potent competitive inhibitor of thymidylate synthetase. Journal of Medicinal Chemistry. 22: 1137-9. PMID 114660 DOI: 10.1021/Jm00195A028 |
0.341 |
|
| 1979 |
Park JS, Chang CT, Mertes MP. 5-[(4-Methyl-1,2,3,4-tetrahydroquinoxalyl)methyl]-2'-deoxyuridine 5'-phosphate: an analogue of a proposed intermediate in thymidylate synthetase catalysis. Journal of Medicinal Chemistry. 22: 1134-7. PMID 114659 DOI: 10.1021/Jm00195A027 |
0.378 |
|
| 1979 |
Brouillette CB, Chang CT, Mertes MP. 5 (alpha-bromoacetyl)-2'=deoxyuridine 5'-phosphate: a mechanism based affinity label for thymidylate synthetase. Biochemical and Biophysical Research Communications. 87: 613-8. PMID 109088 DOI: 10.1016/0006-291X(79)91838-2 |
0.65 |
|
| 1979 |
Park JS, Chang CT, Mertes MP. Enzyme affinity of the 5,6-dihydro derivatives of the substrate and product of thymidylate synthetase catalysis. Journal of Medicinal Chemistry. 22: 319-21. PMID 106122 DOI: 10.1021/JM00189A021 |
0.32 |
|
| 1979 |
Bigge CF, Kalaritis P, Mertes MP. Synthesis of 5-styryl derivatives of uracil nucleosides and nucleotides. Tetrahedron Letters. 20: 1653-1656. DOI: 10.1016/S0040-4039(01)93615-9 |
0.396 |
|
| 1978 |
Mertes MP, Chang CT, De Clercq E, Huang GF, Torrence PF. 5-Nitro-2'-deoxyuridine 5'-monophosphate is a potent irreversible inhibitor of Lactobacillus caesi thymidylate synthetase. Biochemical and Biophysical Research Communications. 84: 1054-9. PMID 103545 DOI: 10.1016/0006-291X(78)91690-X |
0.32 |
|
| 1978 |
Partington CR, Mertes MP. The synthesis of 14C‐labeled N‐carbonylbenzyloxyphenylalanine methylorthoester Journal of Labelled Compounds and Radiopharmaceuticals. 14: 223-229. DOI: 10.1002/Jlcr.2580140210 |
0.304 |
|
| 1977 |
Edelman MS, Barfknecht RL, Huet-Rose R, Boguslawski S, Mertes MP. Thymidylate synthetase inhibitors. Synthesis of N-substituted 5-aminomethyl-2'-deoxyuridine 5'-phosphates. Journal of Medicinal Chemistry. 20: 669-73. PMID 323484 DOI: 10.1002/Chin.197739369 |
0.369 |
|
| 1976 |
Ressner EC, Fraher P, Edelman MS, Mertes MP. Synthesis of 5-substituted uracil derivatives. Journal of Medicinal Chemistry. 19: 194-6. PMID 1107549 DOI: 10.1002/Chin.197617248 |
0.347 |
|
| 1976 |
Kampf A, Pillar CJ, Woodford WJ, Mertes MP. Synthesis of 5-substituted 2'-deoxyuridines. Journal of Medicinal Chemistry. 19: 909-15. PMID 940110 DOI: 10.1021/Jm00229A010 |
0.376 |
|
| 1976 |
Kampf A, Barfknecht RL, Shaffer PJ, Osaki S, Mertes MP. Synthetic inhibitors of Escherichia coli, calf thymus, and Ehrlich ascites tumor thymidylate synthetase. Journal of Medicinal Chemistry. 19: 903-8. PMID 781246 DOI: 10.1002/Chin.197646335 |
0.355 |
|
| 1976 |
Kampf A, Pillar CJ, Woodford WJ, Mertes MP. Synthesis Of 5-Substituted 2′-Deoxyuridines Cheminform. 7. DOI: 10.1002/Chin.197646336 |
0.387 |
|
| 1976 |
BARFKNECHT RL, HUET-ROSE RA, KAMPF A, MERTES MP. ChemInform Abstract: 5-IODOACETAMIDOMETHYL-2′-DEOXYURIDINE 5′-PHOSPHATE. A SELECTIVE INHIBITOR OF MAMMALIAN THYMIDYLATE SYNTHETASES Chemischer Informationsdienst. 7: no-no. DOI: 10.1002/Chin.197644366 |
0.335 |
|
| 1971 |
Mertes MP, Powers LJ, Hava MM. Synthesis and pharmacological activity of dihydrobenzofurans. Journal of Medicinal Chemistry. 14: 361-5. PMID 5553752 DOI: 10.1021/Jm00286A022 |
0.33 |
|
| 1971 |
Mertes MP, Shipchandler MT. Synthesis of deoxyribosides of 5-formyl-, 5-hydroxymethyl- and 5-benzyloxymethyluracil Journal of Heterocyclic Chemistry. 8: 133-136. DOI: 10.1002/Jhet.5570080124 |
0.353 |
|
| 1970 |
Mertes MP, Hanna PE, Ramsey AA. Synthesis of gamma-dimethylamino-alpha-phenylcycloalkyl propionates as potential analgetics. Journal of Medicinal Chemistry. 13: 125-8. PMID 5460892 DOI: 10.1021/Jm00295A031 |
0.607 |
|
| 1970 |
Mertes MP, Ramsey AA, Hanna PE, Miller DD. Synthesis of gamma-dimethylaminomethyl-alpha-phenylcycloalkyl propionates as potential analgetics. Journal of Medicinal Chemistry. 13: 789-94. PMID 5458360 DOI: 10.1021/Jm00299A001 |
0.606 |
|
| 1970 |
Mertes MP, Lin AJ. Cofactor inhibitors of thymidylate synthetase. Piperidine and tetrahydroquinoline analogs of tetrahydrofolic acid. Journal of Medicinal Chemistry. 13: 276-9. PMID 5418501 DOI: 10.1021/Jm00296A026 |
0.31 |
|
| 1970 |
MERTES MP, HANNA PE, RAMSEY AA. ChemInform Abstract: SYNTH. VON GAMMA-DIMETHYLAMINO-ALPHA-PHENYLCYCLOALKYLPROPIONATEN ALS POTENTIELLE ANALGETICA Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197020219 |
0.581 |
|
| 1970 |
Mertes MP, Ramsey AA, Hanna PE, Miller DD. Synthesis of γ-dimethylaminomethyl-α-phenylcycloalkyl propionates as potential analgetics Journal of Medicinal Chemistry. 13: 789-794. |
0.543 |
|
| 1969 |
Mertes MP, Lin AJ. Synthesis and reactions ofN-(p-carbethoxy)phenyl-4-piperidone Journal of Heterocyclic Chemistry. 6: 941-943. DOI: 10.1002/Jhet.5570060628 |
0.333 |
|
| 1968 |
Mertes MP, Borne RF, Hare LE. Synthesis of furo[2,3-c]pyridine derivatives Journal of Organic Chemistry. 33: 133-137. DOI: 10.1021/Jo01265A024 |
0.347 |
|
| 1968 |
Mertes MP, Borne RF, Hare LE. Synthesis of 3‐pyridoxyalkanoic acids and their derivatives Journal of Heterocyclic Chemistry. 5: 281-283. DOI: 10.1002/Jhet.5570050224 |
0.327 |
|
| 1966 |
Mertes MP, Patel NR. Synthesis of methylenetetrahydrofolic acid analogs. Journal of Medicinal Chemistry. 9: 868-73. PMID 5972049 DOI: 10.1021/Jm00324A021 |
0.322 |
|
| 1966 |
Mertes MP, Saheb SE, Miller D. Synthesis of Fluorinated Pyrimidines and Triazines1,2 Journal of Medicinal Chemistry. 9: 876-881. DOI: 10.1021/Jm00324A023 |
0.355 |
|
| 1965 |
Mertes MP, Saheb SE, Miller D. The synthesis of 2-(2′-deoxy-D-ribofuranosyl)-6-trifluoromethyl-as-triazine-3,5-dione, (5-trifluoromethyl-6-aza-2′-deoxyuridine) Journal of Heterocyclic Chemistry. 2: 493-494. DOI: 10.1002/Jhet.5570020437 |
0.334 |
|
| 1965 |
Mertes MP, Saheb SE. 5-Trifluoromethyl-6-azauracil Journal of Heterocyclic Chemistry. 2: 491-491. DOI: 10.1002/Jhet.5570020435 |
0.326 |
|
| 1963 |
MERTES MP, SAHEB SE. THYMINE ANALOGS: THE SYNTHESIS OF 5-DIFLUOROMETHYLURACIL. Journal of Medicinal Chemistry. 6: 619. PMID 14173605 DOI: 10.1021/Jm00341A043 |
0.36 |
|
| 1961 |
MERTES MP, GISVOLD O. Ketals and hemithioketals of 1-methyl-4-piperidone and tropinone. Journal of Pharmaceutical Sciences. 50: 475-80. PMID 13769741 DOI: 10.1002/Jps.2600500606 |
0.608 |
|
| Low-probability matches (unlikely to be authored by this person) |
| 1971 |
MERTES MP, POWERS LJ, HAVA MM. ChemInform Abstract: DIE SYNTHESE UND DIE PHARMAKOLOGISCHE WIRKUNG VON DIHYDROBENZOFURANEN Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197130270 |
0.3 |
|
| 1979 |
Henderson JD, Partington CR, Mertes MP. Synthesis and pH effects on the hydrolysis of 5′-adenosyl phenylalaninate Journal of Organic Chemistry. 44: 1003-1006. DOI: 10.1021/Jo01320A027 |
0.297 |
|
| 1987 |
Hosseini MW, Lehn JM, Maggiora L, Mertes KB, Mertes MP. Supramolecular catalysis in the hydrolysis of ATP facilitated by macrocyclic polyamines: Mechanistic studies Journal of the American Chemical Society. 109: 537-544. DOI: 10.1021/Ja00236A036 |
0.296 |
|
| 1974 |
Woodford WJ, Swartz BA, Pillar CJ, Kampf A, Mertes MP. Synthesis of the alpha and beta anomers of 1-(2-deoxy-D-ribofuranosyl)-4-pyridone. Journal of Medicinal Chemistry. 17: 1027-9. PMID 4607149 DOI: 10.1002/Chin.197501423 |
0.296 |
|
| 1988 |
Chang G, Schwepler D, Decedue CJ, Balzarini J, De Clercq E, Mertes MP. Linear free energy relationship studies of enzyme active site binding: thymidylate synthase. Journal of Medicinal Chemistry. 31: 1141-7. PMID 3373483 DOI: 10.1021/Jm00401A013 |
0.293 |
|
| 1970 |
Mertes MP, Ai Jeng Lin. Cofactor inhibition of thymidylate synthetase. Tetrahydrofolic acid analogs. Journal of Medicinal Chemistry. 13: 77-82. PMID 4904497 DOI: 10.1021/Jm00295A020 |
0.293 |
|
| 1984 |
Conway GA, Park JS, Maggiora L, Mertes MP, Galton N, Michaelis EK. Palladium(II)-Catalyzed Olefin-Coupling of Kainic Acid: Effects of Substitution on the Isopropenyl Group on Receptor Binding. Cheminform. 15. DOI: 10.1002/Chin.198424183 |
0.287 |
|
| 1981 |
De Clercq E, Balzarini J, Descamps J, Bigge CF, Chang CT, Kalaritis P, Mertes MP. Antiviral, antitumor, and thymidylate synthetase inhibition studies of 5-substituted styryl derivatives of 2'-deoxyuridine and their 5'-phosphates. Biochemical Pharmacology. 30: 495-502. PMID 6261769 DOI: 10.1016/0006-2952(81)90635-3 |
0.286 |
|
| 1976 |
Barfknecht RL, Huet-Rose RA, Kampf A, Mertes MP. Letter: 5-iodoacetamidomethyl-2'-deoxyuridine 5'-phosphate. A selective inhibitor of mammalian thymidylate synthetases. Journal of the American Chemical Society. 98: 5041-3. PMID 950429 DOI: 10.1021/Ja00432A069 |
0.286 |
|
| 1991 |
Qian L, Sun Z, Mertes MP, Mertes KB. Synthesis of selectively protected polyaza macrocycles Journal of Organic Chemistry. 56: 4904-4907. DOI: 10.1021/Jo00016A018 |
0.285 |
|
| 1989 |
Hosseini MW, Lehn JM, Jones KC, Plute KE, Mertes KB, Mertes MP. Supramolecular catalysis: Polyammonium macrocycles as enzyme mimics for phosphoryl transfer in ATP hydrolysis Journal of the American Chemical Society. 111: 6330-6335. DOI: 10.1021/Ja00198A051 |
0.28 |
|
| 1981 |
Bansal PC, Pitman IH, Tam JNS, Mertes M, Kaminski JJ. N-hydroxymethyl derivatives of nitrogen heterocycles as possible prodrugs I: N-hydroxymethylation of uracils Journal of Pharmaceutical Sciences. 70: 850-854. PMID 7310649 DOI: 10.1002/Jps.2600700803 |
0.274 |
|
| 1983 |
Hosseini MW, Lehn J, Mertes MP. Efficient Molecular Catalysis of ATP-Hydrolysis by Protonated Macrocyclic Polyamines Helvetica Chimica Acta. 66: 2454-2466. DOI: 10.1002/Chin.198411086 |
0.274 |
|
| 1977 |
Maggiora L, Boguslawski S, Mertes MP. Polynucleotide analogues. Copolymers of vinyl bases with acrylic acid, methylacrylic acid, acrylamide, and 1-vinylpyrrolidone. Journal of Medicinal Chemistry. 20: 1283-7. PMID 333112 DOI: 10.1002/Chin.197812259 |
0.273 |
|
| 1983 |
Lizotte KE, Marecki PE, Mertes MP. Synthesis and conformational aspects of cis- and trans-3-carbomethoxy-6-oxabicyclo[3.1.0]hexane Journal of Organic Chemistry. 48: 3594-3597. DOI: 10.1002/Chin.198412182 |
0.272 |
|
| 1977 |
Edelman MS, Barfknecht RL, Huet-Rose R, Boguslawski S, Mertes MP. Thymidylate synthetase inhibitors. Synthesis of N-substituted 5-aminomethyl-2′-deoxyuridine 5′-phosphates Journal of Medicinal Chemistry. 20: 669-673. |
0.27 |
|
| 1973 |
LEWIS NJ, BARKER KK, FOX RM, MERTES MP. ChemInform Abstract: DIACETOXY-PIPERIDINIUM-ANALOGA VON ACETYL-CHOLIN Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/Chin.197321321 |
0.266 |
|
| 1969 |
Mertes MP, Coats EA. Charge-spatial models: cis- and trans-3- and -4-Substituted cyclohexyl phosphates as analogs of 2'-deoxyuridine 5'-phosphate. Journal of Medicinal Chemistry. 12: 828-32. PMID 4897901 DOI: 10.1021/Jm00305A025 |
0.265 |
|
| 1985 |
Yohannes PG, Mertes MP, Mertes KB. Pyrophosphate formation via a phosphoramidate intermediate in polyammonium macrocycle/metal ion-catalyzed hydrolysis of ATP Journal of the American Chemical Society. 107: 8288-8289. DOI: 10.1021/Ja00312A094 |
0.263 |
|
| 1971 |
Mertes MP, Powers LJ, Shefter E. Isolation and identification of the cis-trans stereoisomers of substituted 3-hydroxy- (or 3-acetoxy-) 2-methyl-2,3-dihydrobenzofurans. Dihydrobenzofurans Which obey the Karplus equation Journal of Organic Chemistry. 36: 1805-1807. DOI: 10.1021/Jo00812A018 |
0.263 |
|
| 1971 |
Mertes MP, Shipchandler MT. Charge-spatial models. 2. cis-and trans-3-and-4-carboxycyclohexyl phosphates and the carboxylate esters as analogs of 2'-deoxyuridine 5'-phosphate. Journal of Medicinal Chemistry. 14: 257-8. PMID 4994697 DOI: 10.1021/Jm00285A026 |
0.262 |
|
| 1973 |
Lewis NJ, Barker KK, Fox RM, Mertes MP. Diacetoxypiperidinium analogs of acetylcholine. Journal of Medicinal Chemistry. 16: 156-9. PMID 4683111 DOI: 10.1021/Jm00260A016 |
0.257 |
|
| 1987 |
Hosseini MW, Lehn JM, Duff SR, Gu K, Mertes MP. Synthesis of mono- and difunctionalized ditopic [24]N6O2 macrocyclic receptor molecules Journal of Organic Chemistry. 52: 1662-1666. DOI: 10.1021/Jo00385A003 |
0.256 |
|
| 1963 |
MERTES MP, SAHEB SE. Use of sulfur tetrafluoride in syntheses of potential anticancer agents. Journal of Pharmaceutical Sciences. 52: 508-9. PMID 13935069 DOI: 10.1002/Jps.2600520531 |
0.251 |
|
| 1974 |
Hes J, Mertes MP. Di(2-tert-butylphenyl) phosphorochloridate. A new selective phosphorylating agent Journal of Organic Chemistry. 39: 3767-3769. DOI: 10.1021/Jo00939A035 |
0.244 |
|
| 1981 |
Early SL, Michaelis EK, Mertes MP. Pharmacological specificity of synaptosomal and synaptic membrane gamma-aminobutyric acid (GABA) transport processes. Biochemical Pharmacology. 30: 1105-13. PMID 7259793 DOI: 10.1016/0006-2952(81)90449-4 |
0.243 |
|
| 1987 |
Yohannes PG, Plute KE, Mertes MP, Mertes KB. Specificity, catalysis, and regulation: Effects of metal ions on polyammonium macrocycle catalyzed dephosphorylation of ATP Inorganic Chemistry. 26: 1751-1755. DOI: 10.1021/Ic00258A023 |
0.241 |
|
| 1990 |
Mertes MP, Mertes KB. Polyammonium macrocycles as catalysts for phosphoryl transfer: The evolution of an enzyme mimic Accounts of Chemical Research. 23: 413-418. DOI: 10.1021/Ar00180A003 |
0.24 |
|
| 1963 |
Mertes MP, Saheb SB. Thymine analogs: The synthesis of 5-difluoromethyluracil [3] Journal of Medicinal Chemistry. 6: 619. |
0.24 |
|
| 1966 |
Mertes MP, Saheb SE, Miller D. Synthesis of fluorinated pyrimidines and triazines Journal of Medicinal Chemistry. 9: 876-881. |
0.239 |
|
| 1973 |
Wilson RS, Mertes MP. A chemical model for thymidylate synthetase catalysis. Biochemistry. 12: 2879-86. PMID 4719124 DOI: 10.1021/Bi00739A017 |
0.237 |
|
| 1987 |
Chang G, Mertes MP. Linear free energy relationship studies of 5-substituted 2,4-dioxopyrimidine nucleosides Journal of Organic Chemistry. 52: 3625-3631. DOI: 10.1021/Jo00392A023 |
0.235 |
|
| 1969 |
Mertes MP, Ramsey AA. Omega-dithiolano amino acids. Journal of Medicinal Chemistry. 12: 342-3. PMID 5783619 DOI: 10.1021/Jm00302A042 |
0.225 |
|
| 1968 |
Mertes MP, Borne RF, Hare LE. The synthesis of furo[2,3-c]pyridine derivatives Journal of Organic Chemistry. 33: 133-137. |
0.224 |
|
| 1982 |
Balzarini J, De Clercq E, Torrence PF, Mertes MP, Park JS, Schmidt CL, Shugar D, Barr PJ, Jones AS, Verhelst G, Walker RT. Role of thymidine kinase in the inhibitory activity of 5-substituted-2'-deoxyuridines on the growth of human and murine tumor cell lines. Biochemical Pharmacology. 31: 1089-95. PMID 7082363 DOI: 10.1016/0006-2952(82)90347-1 |
0.224 |
|
| 1987 |
Kagel JR, Mertes MP. Selective addition of methanol to 1,2-epoxy-1-vinylcyclopentane Journal of Organic Chemistry. 52: 2950-2953. DOI: 10.1021/Jo00389A065 |
0.223 |
|
| 1989 |
Jahansouz H, Jiang Z, Himes RH, Mertes MP, Mertes KB. Formate activation in neutral aqueous solution mediated by a polyammonium macrocycle Journal of the American Chemical Society. 111: 1409-1413. DOI: 10.1021/Ja00186A039 |
0.221 |
|
| 1970 |
Powers LJ, Mertes MP. Antibacterial activity of nitrobenzofurans. Journal of Medicinal Chemistry. 13: 1102-5. PMID 4991392 DOI: 10.1021/Jm00300A020 |
0.22 |
|
| 1987 |
Al-Razzak LA, Schwepler D, Decedue CJ, Mertes MP. Inactivation of thymidylate synthase at an alternate high-affinity binding site. Journal of Medicinal Chemistry. 30: 1705-6. PMID 3656346 DOI: 10.1021/Jm00393A001 |
0.217 |
|
| 1963 |
Mertes MP. The conformational preference of sulfur in hemithioketals Journal of Organic Chemistry. 28: 2320-2323. DOI: 10.1021/Jo01044A039 |
0.216 |
|
| 1968 |
Mertes MP, Nerurkar SA, Walaszek EJ. Bisquaternary ammonium indolines and perhydroindoles in ganglionic blockade. Journal of Medicinal Chemistry. 11: 106-11. PMID 5637152 DOI: 10.1021/Jm00307A024 |
0.213 |
|
| 1967 |
Mertes MP, Gilman Q. N-thymidylglycine and ethyl p-N-thymidylaminobenzoate. Journal of Medicinal Chemistry. 10: 965-6. PMID 6048515 DOI: 10.1021/Jm00317A056 |
0.204 |
|
| 1969 |
Mertes MP, Coats EA. Synthesis of carbonate analogs of dinucleosides. 3'-Thymidinyl 5'-thymidinyl carbonate, 3'-thymidinyl 5'-(5-fluoro-2'-deoxyuridinyl) carbonate, and 3'-(5-fluoro-2'-deoxyuridinyl) 5'-thymidinyl carbonate. Journal of Medicinal Chemistry. 12: 154-7. PMID 4883934 DOI: 10.1021/Jm00301A041 |
0.202 |
|
| 1970 |
MERTES MP, SHIPCHANDLER MT. ChemInform Abstract: SYNTH. VON 5-FORMYL-2′-DESOXYURIDIN UND DEM ALPHA-ANOMEREN Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/chin.197040377 |
0.196 |
|
| 1961 |
Mertes MP. Intramolecular hydrogen bonding to sulfur Journal of Organic Chemistry. 26: 5236-5238. DOI: 10.1021/Jo01070A532 |
0.193 |
|
| 1968 |
Mertes MP, Smrt J. Nucleic acid components and their analogues. CXV. Synthesis of N4-hydroxy-6-azacytidine 5'-phosphate and 5'-diphosphate Collection of Czechoslovak Chemical Communications. 33: 3304-3312. DOI: 10.1135/cccc19683304 |
0.193 |
|
| 1958 |
MERTES MP, WILSON CO. Glutarimides. V. Synthesis of 2-allyl-2-phenylglutarimide. Journal of the American Pharmaceutical Association. American Pharmaceutical Association. 47: 882-5. PMID 13610712 |
0.173 |
|
| 1980 |
BROUILLETTE CB, CHANG CT, MERTES MP. ChemInform Abstract: 5-(α-BROMOACETYL)-2′-DEOXYURIDINE 5′-PHOSPHATE: AN AFFINITY LABEL FOR THYMIDYLATE SYNTHETASE Chemischer Informationsdienst. 11. DOI: 10.1002/chin.198016303 |
0.17 |
|
| 1970 |
Mertes MP. The synthesis of the alpha and beta anomers of 1-(2-deoxy-D-ribofuranosyl)-2-pyridone. Journal of Medicinal Chemistry. 13: 149-51. PMID 5412096 |
0.163 |
|
| 1978 |
Partington CR, Mertes MP. The synthesis of 14C-labeled N-carbonylbenzyloxyphenylalanine methylorthoester Journal of Labelled Compounds and Radiopharmaceuticals. 14: 223-229. |
0.16 |
|
| 1968 |
Mertes MP, Holý A, Smrt J. Oligonucleotidic compounds. XXVI. Synthesis of uridylyl-(3'→5')-N4-hydroxy-6-azacytidine and N4-hydroxy-6-azacytidylyl-(3'→5')-uridine Collection of Czechoslovak Chemical Communications. 33: 3313-3323. DOI: 10.1135/cccc19683313 |
0.157 |
|
| 1984 |
HOSSEINI MW, LEHN J, MERTES MP. ChemInform Abstract: EFFICIENT MOLECULAR CATALYSIS OF ATP HYDROLYSIS BY PROTONATED MACROCYCLIC POLYAMINES Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198411086 |
0.153 |
|
| 1967 |
Mertes MP, Zielinski J, Pillar C. Approaches to the Synthesis of 1-Deazauridine and 2'-Deoxy-1-deazauridine. Journal of Medicinal Chemistry. 10: 320-5. PMID 22185123 DOI: 10.1021/jm00315a007 |
0.151 |
|
| 1970 |
MERTES MP, LIN AJ. ChemInform Abstract: COFAKTOR-INHIBITOREN DER THYMIDYLAT-SYNTHETASE, PIPERIDIN- UND TETRAHYDROCHINOLIN-ANALOGA DER TETRAHYDROFOLSAEURE Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/chin.197024309 |
0.141 |
|
| 1976 |
Boguslawski S, Olson PE, Mertes MP. Mechanims of stimulation of in vitro protein synthesis by some copolymers of styrene, vinyluracil, and vinyladenine with maleic acid and acrylic acid. Biochemistry. 15: 3536-40. PMID 782518 |
0.14 |
|
| 1981 |
De Clercq E, Balzarini J, Torrence PF, Mertes MP, Schmidt CL, Shugar D, Barr PJ, Jones AS, Verhelst G, Walker RT. Thymidylate synthetase as target enzyme for the inhibitory activity of 5-substituted 2'-deoxyuridines on mouse leukemia L1210 cell growth. Molecular Pharmacology. 19: 321-30. PMID 7231392 |
0.136 |
|
| 1971 |
MERTES MP, SHIPCHANDLER MT. ChemInform Abstract: SYNTH. VON DESOXYRIBOSIDEN VON 5-FORMYL-, 5-HYDROXYMETHYL- UND 5-BENZYLOXYMETHYL-URACIL Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/chin.197128327 |
0.136 |
|
| 1967 |
Mertes MP, Zielinski J, Pillars C. Approaches to the Synthesis of 1-Deazauridine and 2′-Deoxy-l-deazauridine Journal of Medicinal Chemistry. 10: 320-325. |
0.135 |
|
| 1970 |
MERTES MP, BORNE RF, BRIDEN RC. ChemInform Abstract: KERNMAGNETISCHE RESONANZSPEKTREN HYDRIERTER FURO(2,3-C)PYRIDINE Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/chin.197011030 |
0.131 |
|
| 1989 |
Mertes M, Mertes K, Paoletti P, Bianchi A. Atpase activity in polyammonium macrocycles: The influence of ring size and heteroatoms Journal of Inorganic Biochemistry. 36: 275. DOI: 10.1016/0162-0134(89)84378-8 |
0.129 |
|
| 1970 |
MERTES MP. ChemInform Abstract: SYNTH. DER ALPHA- UND BETA-ANOMEREN DES 1-(2-DESOXY-D-RIBOFURANOSYL)-2-PYRIDONS Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/chin.197019428 |
0.128 |
|
| 1971 |
MERTES MP, SHIPCHANDLER MT. ChemInform Abstract: LADUNGS- UND RAUMMODELLE 2. MITT. CIS- UND TRANS-3- BZW. -4-CARBOXYCYCLOHEXYLPHOSPHATE UND DIE CARBOXYLATESTER ALS ANALOGA VON 2′-DESOXY-URIDIN-5′-PHOSPHAT Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/chin.197126015 |
0.128 |
|
| 1972 |
Mertes M, Peters MA, Mahoney W, Yarus M. Isoleucylation of transfer RNAf Met (E. coli) by isoleucyl-transfer RNA synthetase from Escherichia coli Journal of Molecular Biology. 71: 671-685. PMID 4567469 DOI: 10.1016/S0022-2836(72)80031-7 |
0.123 |
|
| 1975 |
Olson PE, Fraher P, Boguslawski S, Mertes MP. Polynucleotide analogs: acrylic acid and maleic acid copolymers of 1-vinyluracil and 9-vinyladenine. Biochemistry. 14: 4892-6. PMID 1101958 |
0.118 |
|
| 1975 |
HES J, MERTES MP. ChemInform Abstract: DI(2-TERT.-BUTYLPHENYL)PHOSPHOROCHLORIDATE, A NEW SELECTIVE PHOSPHORYLATING AGENT Chemischer Informationsdienst. 6: no-no. DOI: 10.1002/chin.197513340 |
0.118 |
|
| 1974 |
Woodford WJ, Swartz BA, Pillar CJ, Kampf A, Mertes MP. Synthesis of the α and β anomers of 1-(2-deoxy-D-ribofuranosyl)-4-pyridone Journal of Medicinal Chemistry. 17: 1027-1029. |
0.11 |
|
| 1973 |
Baer TA, Mertes MP. Pericillinase inhibition. Journal of Medicinal Chemistry. 16: 85-7. PMID 4629666 |
0.105 |
|
| 1971 |
POWERS LJ, MERTES MP. ChemInform Abstract: BAKTERICIDE WIRKUNG VON NITROBENZOFURANEN Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/chin.197111297 |
0.105 |
|
| 1970 |
MERTES MP, LIN AJ. ChemInform Abstract: INHIBIERUNG DES COFAKTORS VON THYMIDYLAT-SYNTHETASE, TETRAHYDROFOLSAEUREANALOGA Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/chin.197019340 |
0.101 |
|
| 1970 |
MERTES MP, LIN AJ. ChemInform Abstract: SYNTH. UND RK. VON N-(P-CARBAETHOXY-PHENYL)-4-PIPERIDON Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/chin.197018250 |
0.093 |
|
| 1972 |
Wilson RS, Mertes MP. A chemical model for thymidylate synthetase catalysis [24] Journal of the American Chemical Society. 94: 7182-7183. |
0.092 |
|
| 1973 |
Yarus M, Mertes M. The variety of intraspecific misacylations carried out by isoleucyl transfer ribonucleic acid synthetase of Escherichia coli Journal of Biological Chemistry. 248: 6744-6749. PMID 4355506 |
0.083 |
|
| 1973 |
Hasbun JA, Barker KK, Mertes MP. Trimethylammonium phenyl ketones. Actions on the cholinereic receptor and acetylcholinesterase Journal of Medicinal Chemistry. 16: 847-849. PMID 4725932 |
0.077 |
|
| 1972 |
WILSON RS, MERTES MP. ChemInform Abstract: CHEMISCHES MODELL DER KATALYSE DURCH THYMIDYLATSYNTHETASE Chemischer Informationsdienst. 3: no-no. DOI: 10.1002/chin.197251124 |
0.071 |
|
| 1969 |
Mertes MP, Borne RF, Briden RC. The nuclear magnetic resonance spectra of furo[2,3-c] pyridine derivatives Spectrochimica Acta Part a: Molecular Spectroscopy. 25: 1953-1958. |
0.064 |
|
| 1969 |
Mertes MP, Lee HK, Schowen R. The conformational preferences of sulfur and oxygen in hemithioketals. The Journal of Physical Chemistry. 34: 2080-2. PMID 5788207 DOI: 10.1021/Jo01259A011 |
0.033 |
|
| 1969 |
Mertes MP, Lee HK, Schowen RL. The conformational preferences of sulfur and oxygen in hemithioketals Journal of Organic Chemistry. 34: 2080-2082. |
0.033 |
|
| 2014 |
Fischer F, Collange O, Mahoudeau G, Simon M, Moussa H, Thibaud A, Steib A, Pottecher T, Mertes M. [VENTILOP survey. Survey in peroperative mechanical ventilation]. Annales FrançAises D'AnesthèSie Et De RèAnimation. 33: 389-94. PMID 24930761 DOI: 10.1016/j.annfar.2014.05.002 |
0.01 |
|
| 2010 |
Chalot Y, Boileau S, Vedel M, Audibert G, Mertes MP, Bouaziz H. [Course of the anaesthesiology and intensive care unit residents in Lorraine, France]. Annales FrançAises D'AnesthèSie Et De RèAnimation. 29: 209-14. PMID 20189342 DOI: 10.1016/j.annfar.2009.11.011 |
0.01 |
|
| 1970 |
Mertes MP, Powers LJ, Shefter E. Dihydrobenzofurans in which Jcis-2,3 > Jtrans-2,3: Confirmation using X-ray diffraction analysis Journal of the Chemical Society D: Chemical Communications. 620a-620a. DOI: 10.1039/C2970000620a |
0.01 |
|
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