Year |
Citation |
Score |
2022 |
Wilson BS, Peiser-Oliver J, Gillis A, Evans S, Alamein C, Mostyn SN, Shimmon S, Rawling T, Christie MJ, Vandenberg RJ, Mohammadi SA. . The Journal of Pharmacology and Experimental Therapeutics. PMID 35779948 DOI: 10.1124/jpet.122.001265 |
0.611 |
|
2021 |
Wilson KA, Mostyn SN, Frangos ZJ, Shimmon S, Rawling T, Vandenberg RJ, O'Mara ML. The allosteric inhibition of glycine transporter 2 by bioactive lipid analgesics is controlled by penetration into a deep lipid cavity. The Journal of Biological Chemistry. 100282. PMID 33450225 DOI: 10.1016/j.jbc.2021.100282 |
0.647 |
|
2020 |
Mostyn SN, Sarker S, Muthuraman P, Raja A, Shimmon S, Rawling T, Cioffi CL, Vandenberg RJ. A photoswitchable ORG25543 congener enables optical control of glycine transporter 2. Acs Chemical Neuroscience. PMID 32191428 DOI: 10.1021/Acschemneuro.9B00655 |
0.709 |
|
2019 |
Mostyn SN, Wilson KA, Schumann-Gillett A, Frangos ZJ, Shimmon S, Rawling T, Ryan RM, O'Mara ML, Vandenberg RJ. Identification of an allosteric binding site on the human glycine transporter, GlyT2, for bioactive lipid analgesics. Elife. 8. PMID 31621581 DOI: 10.7554/Elife.47150 |
0.737 |
|
2019 |
Mostyn SN, Rawling T, Mohammadi S, Shimmon S, Frangos ZJ, Sarker S, Yousuf A, Vetter I, Ryan RM, Christie MJ, Vandenberg RJ. Development of an N-acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain. Journal of Medicinal Chemistry. PMID 30714733 DOI: 10.1021/Acs.Jmedchem.8B01775 |
0.678 |
|
2019 |
Mostyn SN, Wilson KA, Schumann-Gillett A, Frangos ZJ, Shimmon S, Rawling T, Ryan RM, O'Mara ML, Vandenberg RJ. Author response: Identification of an allosteric binding site on the human glycine transporter, GlyT2, for bioactive lipid analgesics Elife. DOI: 10.7554/Elife.47150.029 |
0.679 |
|
2017 |
Carland JE, Thomas M, Mostyn SN, Subramanian N, O'Mara ML, Ryan RM, Vandenberg RJ. Molecular Determinants for Substrate Interactions with the Glycine Transporter GlyT2. Acs Chemical Neuroscience. PMID 29120604 DOI: 10.1021/Acschemneuro.7B00407 |
0.694 |
|
2017 |
Mostyn SN, Carland JE, Shimmon S, Ryan RM, Rawling T, Vandenberg RJ. Synthesis and Characterization of Novel Acyl-Glycine Inhibitors of GlyT2. Acs Chemical Neuroscience. PMID 28574249 DOI: 10.1021/Acschemneuro.7B00105 |
0.715 |
|
2015 |
Vandenberg RJ, Mostyn SN, Carland JE, Ryan RM. Glycine Transporter2 Inhibitors: Getting the balance right. Neurochemistry International. PMID 26723543 DOI: 10.1016/J.Neuint.2015.12.007 |
0.677 |
|
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